The histamine H 3 receptor: an attractive target for the treatment of cognitive disorders von Esbenshade, T A, Browman, K E, Bitner, R S, Strakhova, M, Cowart, M D, Brioni, J D

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Antibody Drug Conjugates for Cancer Therapy von Polakis, Paul

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Synthetic oleanane triterpenoids: multifunctional drugs with a broad range of applications for prevention and treatment of chronic disease von Liby, Karen T, Sporn, Michael B

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The histamine H3 receptor: an attractive target for the treatment of cognitive disorders von Esbenshade, T A, Browman, K E, Bitner, R S, Strakhova, M, Cowart, M D, Brioni, J D

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Therapeutic Potential of α 7 Nicotinic Acetylcholine Receptors von Bertrand, Daniel, Lee, Chih-Hung L., Flood, Dorothy, Marger, Fabrice, Donnelly-Roberts, Diana

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Minimization of potential hERG liability in histamine H3 receptor antagonists von Black, L. A., Liu, H., Diaz, G. J., Fox, G. B., Browman, K. E., Wetter, J., Marsh, K. C., Miller, T. R., Esbenshade, T. A., Brioni, J., Cowart, M. D.

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Use of the H3 receptor antagonist radioligand [3H]‐A‐349821 to reveal in vivo receptor occupancy of cognition enhancing H3 receptor antagonists von Miller, TR, Milicic, I, Bauch, J, Du, J, Surber, B, Browman, KE, Marsh, K, Cowart, M, Brioni, JD, Esbenshade, TA

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Pharmacological classification of histamine H3 receptor agents across species is attributable to transmembrane 3 sequence differences von Esbenshade, T A, Estvander, B R, Miller, T R, Baranowski, J L, Sharma, R, Hancock, A A, Krueger, K M

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Pharmacologically active drug metabolites: impact on drug discovery and pharmacotherapy von Obach, R Scott

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Cognitive Effects of MDMA in Laboratory Animals: A Systematic Review Focusing on Dose von Pantoni, Madeline M, Anagnostaras, Stephan G

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Molecular modeling and pharmacological analysis of species-related histamine H3 receptor heterogeneity von YAO, B. B, HUTCHINS, C. W, CARR, T. L, CASSAR, S, MASTERS, J. N, BENNANI, Y. L, ESBENSHADE, T. A, HANCOCK, A. A

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In vitro and in vivo characterization of A‐940894: a potent histamine H 4 receptor antagonist with anti‐inflammatory properties von Strakhova, MI, Cuff, CA, Manelli, AM, Carr, TL, Witte, DG, Baranowski, JL, Vortherms, TA, Miller, TR, Rundell, L, McPherson, MJ, Adair, RM, Brito, AA, Bettencourt, BM, Yao, BB, Wetter, JM, Marsh, KC, Liu, H, Cowart, MD, Brioni, JD, Esbenshade, TA

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Use of the H 3 receptor antagonist radioligand [ 3 H]‐A‐349821 to reveal in vivo receptor occupancy of cognition enhancing H 3 receptor antagonists von Miller, TR, Milicic, I, Bauch, J, Du, J, Surber, B, Browman, KE, Marsh, K, Cowart, M, Brioni, JD, Esbenshade, TA

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Structure-activity relationships of A-331440: a new histamine-3 antagonist with anti-obesity properties von Faghih, R, Esbenshade, T A, Krueger, K M, Yao, B B, Witte, D G, Miller, T M, Kang, C H, Fox, G B, Cowart, M, Bennani, Y L, Hancock, A A

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Use of an inverse agonist radioligand [3H]A-317920 reveals distinct pharmacological profiles of the rat histamine H3 receptor von Yao, B Bei, Witte, D G, Miller, T R, Carr, T L, Kang, C H, Cassar, S, Faghih, R, Bennani, Y L, Surber, B W, Hancock, A A, Esbenshade, T A

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Fluorescent benzofuran histamine H3 receptor antagonists with sub-nanomolar potency von Cowart, M., Gfesser, G. A., Bhatia, K., Esser, R., Sun, M., Miller, T. R., Krueger, K., Witte, D., Esbenshade, T. A., Hancock, A. A.

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A new family of histamine H3 receptor antagonists based on a natural product: discovery, SAR, and properties of the series von Cowart, M, Sun, M, Zhao, C, Witte, D G, Miller, T R, Krueger, K M, Browman, K, Fox, G B, Bennani, Y L, Esbenshade, T A, Hancock, A A

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Antiobesity evaluation of histamine H3 receptor (H3R) antagonist analogs of A-331440 with improved safety and efficacy von Hancock, A A, Diehl, M S, Fey, T A, Bush, E N, Faghih, R, Miller, T R, Krueger, K M, Pratt, J K, Cowart, M D, Dickinson, R W, Shapiro, R, Knourek-Segel, V E, Droz, B A, McDowell, C A, Krishna, G, Brune, M E, Esbenshade, T A, Jacobson, P B

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Differential CNS expression and functional activity of multiple human H3 receptor isoforms von Esbenshade, T. A., Strakhova, M. I., Carr, T. L., Sharma, R., Witte, D. G., Yao, B. B., Miller, T. R., Hancock, A. A.

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In vitro and in vivo characterization of A‐940894: a potent histamine H4 receptor antagonist with anti‐inflammatory properties von Strakhova, MI, Cuff, CA, Manelli, AM, Carr, TL, Witte, DG, Baranowski, JL, Vortherms, TA, Miller, TR, Rundell, L, McPherson, MJ, Adair, RM, Brito, AA, Bettencourt, BM, Yao, BB, Wetter, JM, Marsh, KC, Liu, H, Cowart, MD, Brioni, JD, Esbenshade, TA

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