Prospects for Antibacterial Discovery and Development von Privalsky, Thomas M, Soohoo, Alexander M, Wang, Jinhua, Walsh, Christopher T, Wright, Gerard D, Gordon, Eric M, Gray, Nathanael S, Khosla, Chaitan

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Orally Absorbed Derivatives of the β‑Lactamase Inhibitor Avibactam. Design of Novel Prodrugs of Sulfate Containing Drugs von Gordon, Eric M, Duncton, Matthew A. J, Gallop, Mark A

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In situ assembly of enzyme inhibitors using extended tethering von Erlanson, Daniel A., Lam, Joni W., Wiesmann, Christian, Luong, Tinh N., Simmons, Robert L., DeLano, Warren L., Choong, Ingrid C., Burdett, Matthew T., Flanagan, W. Michael, Lee, Dennis, Gordon, Eric M., O'Brien, Tom

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Applications of Combinatorial Technologies to Drug Discovery. 2. Combinatorial Organic Synthesis, Library Screening Strategies, and Future Directions von Gordon, Eric M, Barrett, Ronald W, Dower, William J, Fodor, Stephen P. A, Gallop, Mark A

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Applications of Combinatorial Technologies to Drug Discovery. 1. Background and Peptide Combinatorial Libraries von Gallop, Mark A, Barrett, Ronald W, Dower, William J, Fodor, Stephen P. A, Gordon, Eric M

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Approaches to Combinatorial Synthesis of Heterocycles:  A Solid-Phase Synthesis of 1,4-Dihydropyridines von Gordeev, Mikhail F, Patel, Dinesh V, Gordon, Eric M

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Exercise and rehabilitation of the cancer patient von Gordon, Eric M., P.T

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Combinatorial Organic Synthesis of Highly Functionalized Pyrrolidines: Identification of a Potent Angiotensin Converting Enzyme Inhibitor from a Mercaptoacyl Proline Library von Murphy, Martin M, Schullek, John R, Gordon, Eric M, Gallop, Mark A

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Combinatorial modification of natural products: Synthesis and in vitro analysis of derivatives of thiazole peptide antibiotic GE2270 A: A-ring modifications von CLOUGH, Jeffrey, SHAOQING CHEN, CIABATTI, Romeo, JACOBS, Jeffrey W, GORDON, Eric M, HACKBARTH, Corinne, LAM, Stuart, TRIAS, Joaquim, WHITE, Richard J, CANDIANI, Gianpaolo, DONADIO, Stefano, ROMANO, Gabriella

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Toward Orally Absorbed Prodrugs of the Antibiotic Aztreonam. Design of Novel Prodrugs of Sulfate Containing Drugs. Part 2 von Gordon, Eric M, Duncton, Matthew A. J, Wang, Brian J, Qi, Longwu, Fan, Dazhong, Li, Xianfeng, Ni, Zhi-Jie, Ding, Pingyu, Grygorash, Ruslan, Low, Eddy, Yu, Guijun, Sun, Jiawei

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Site-Directed Ligand Discovery von Erlanson, Daniel A., Braisted, Andrew C., Raphael, Darren R., Randal, Mike, Stroud, Robert M., Gordon, Eric M., Wells, James A.

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Aminoethylenes:  A Tetrahedral Intermediate Isostere Yielding Potent Inhibitors of the Aspartyl Protease BACE-1 von Yang, Wenjin, Lu, Wanli, Lu, Yafan, Zhong, Min, Sun, Jian, Thomas, Anila E, Wilkinson, Jennifer M, Fucini, Raymond V, Lam, Melissa, Randal, Mike, Shi, Xiao-Ping, Jacobs, Jeffrey W, McDowell, Robert S, Gordon, Eric M, Ballinger, Marcus D

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Selective Reduction of Peptide Isothiazolidin-3-ones von Shiau, Timothy P, Erlanson, Daniel A, Gordon, Eric M

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Farnesyl Diphosphate-Based Inhibitors of Ras Farnesyl Protein Transferase von Patel, Dinesh V, Schmidt, Robert J, Biller, Scott A, Gordon, Eric M, Robinson, Simon S, Manne, Veeraswamy

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Identification of Potent and Selective Small-Molecule Inhibitors of Caspase-3 through the Use of Extended Tethering and Structure-Based Drug Design von Choong, Ingrid C, Lew, Willard, Lee, Dennis, Pham, Phuongly, Burdett, Matthew T, Lam, Joni W, Wiesmann, Christian, Luong, Tinh N, Fahr, Bruce, DeLano, Warren L, McDowell, Robert S, Allen, Darin A, Erlanson, Daniel A, Gordon, Eric M, O'Brien, Tom

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Solid-Supported Combinatorial Synthesis of Structurally Diverse β-Lactams von Ruhland, Beatrice, Bhandari, Ashok, Gordon, Eric M, Gallop, Mark A

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Strategies for Combinatorial Organic Synthesis: Solution and Polymer-Supported Synthesis of 4-Thiazolidinones and 4-Metathiazanones Derived from Amino Acids von Holmes, Christopher P, Chinn, Jason P, Look, Gary C, Gordon, Eric M, Gallop, Mark A

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The first potent inhibitor of squalene synthase: a profound contribution of an ether oxygen to inhibitor-enzyme interaction von Biller, Scott A, Sofia, Michael J, DeLange, Barbara, Forster, Cornelia, Gordon, Eric M, Harrity, Thomas, Rich, Lois C, Ciosek, Carl P

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Approaches to combinatorial synthesis of heterocycles: Solid phase synthesis of pyridines and pyrido[2,3-d]pyrimidines von Gordeev, Mikhail F, Patel, Dinesh V, Wu, Jie, Gordon, Eric M

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Versatile Approach To Encoding Combinatorial Organic Syntheses Using Chemically Robust Secondary Amine Tags von Ni, Zhi-Jie, Maclean, Derek, Holmes, Christopher P, Murphy, Martin M, Ruhland, Beatrice, Jacobs, Jeffrey W, Gordon, Eric M, Gallop, Mark A

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