Negative allosteric modulation of GluN1/GluN3 NMDA receptors von Zhu, Zongjian, Yi, Feng, Epplin, Matthew P., Liu, Ding, Summer, Samantha L., Mizu, Ruth, Shaulsky, Gil, XiangWei, Wenshu, Tang, Weiting, Burger, Pieter B., Menaldino, David S., Myers, Scott J., Liotta, Dennis C., Hansen, Kasper B., Yuan, Hongjie, Traynelis, Stephen F.

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An NMDAR positive and negative allosteric modulator series share a binding site and are interconverted by methyl groups von Perszyk, Riley, Katzman, Brooke M, Kusumoto, Hirofumi, Kell, Steven A, Epplin, Matthew P, Tahirovic, Yesim A, Moore, Rhonda L, Menaldino, David, Burger, Pieter, Liotta, Dennis C, Traynelis, Stephen F

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Biased modulators of NMDA receptors control channel opening and ion selectivity von Perszyk, Riley E., Swanger, Sharon A., Shelley, Chris, Khatri, Alpa, Fernandez-Cuervo, Gabriela, Epplin, Matthew P., Zhang, Jing, Le, Phuong, Bülow, Pernille, Garnier-Amblard, Ethel, Gangireddy, Pavan Kumar Reddy, Bassell, Gary J., Yuan, Hongjie, Menaldino, David S., Liotta, Dennis C., Liebeskind, Lanny S., Traynelis, Stephen F.

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Discovery of Dihydropyrrolo[1,2‑a]pyrazin-3(4H)‑one-Based Second-Generation GluN2C- and GluN2D-Selective Positive Allosteric Modulators (PAMs) of the N‑Methyl‑d‑Aspartate (NMDA) Re... von Epplin, Matthew P, Mohan, Ayush, Harris, Lynnea D, Zhu, Zongjian, Strong, Katie L, Bacsa, John, Le, Phuong, Menaldino, David S, Traynelis, Stephen F, Liotta, Dennis C

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The Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA Receptor von Kaiser, Thomas M., Kell, Steven A., Kusumoto, Hirofumi, Shaulsky, Gil, Bhattacharya, Subhrajit, Epplin, Matthew P., Strong, Katie L., Miller, Eric J., Cox, Bryan D., Menaldino, David S., Liotta, Dennis C., Traynelis, Stephen F., Burger, Pieter B.

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The Structure–Activity Relationship of a Tetrahydroisoquinoline Class of N‑Methyl‑d‑Aspartate Receptor Modulators that Potentiates GluN2B-Containing N‑Methyl‑d‑Aspartate Receptors... von Strong, Katie L, Epplin, Matthew P, Bacsa, John, Butch, Christopher J, Burger, Pieter B, Menaldino, David S, Traynelis, Stephen F, Liotta, Dennis C

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Distinct GluN1 and GluN2 Structural Determinants for Subunit-Selective Positive Allosteric Modulation of N-Methyl-D-aspartate Receptors von Strong, Katie L., Epplin, Matthew P., Ogden, Kevin K., Burger, Pieter B., Kaiser, Thomas M., Wilding, Timothy J., Kusumoto, Hiro, Camp, Chad R., Shaulsky, Gil, Bhattacharya, Subhrajit, Perszyk, Riley E., Menaldino, David S., McDaniel, Miranda J., Zhang, Jing, Phuong Le, Banke, Tue G., Hansen, Kasper B., Huettner, James E., Liotta, Dennis C., Traynelis, Stephen F.

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N-methyl-D-aspartic Acid Receptor Modulators von Liotta, Dennis, Epplin, Matthew, Traynelis, Stephen F, Menaldino, David

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N-methyl-D-aspartic acid receptor modulators von Liotta, Dennis, Epplin, Matthew, Traynelis, Stephen F, Menaldino, David

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N-methyl-D-aspartic Acid Receptor Modulators von Liotta, Dennis, Epplin, Matthew, Traynelis, Stephen F, Menaldino, David

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Negative Allosteric Modulation of GluN3-Containing N-Methyl-D-Aspartate Receptors von Yuan, Hongjie, McCallum, Adam, Liotta, Dennis C, Epplin, Matthew, Jacobs, Leon, Traynelis, Stephen, Summer, Samantha, Menaldino, David

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Process for preparing tetralin compounds von Gal, Balint, Yu, Kai, Mata, Guillaume, Epplin, Matthew, Kalisiak, Jaroslaw, Mailyan, Artur Karenovich, Hardman, Clayton, Lawson, Kenneth Victor, Rosen, Brandon Reid, Drew, Samuel Lawrie, Haelsig, Karl T, Wang, Zhang, Fournier, Jeremy, Leleti, Manmohan Reddy, Beatty, Joel Worley

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INHIBITORS OF HIF-2ALPHA AND METHODS OF USE THEREOF von LELETI, Manmohan Reddy, DREW, Samuel Lawrie, EPPLIN, Matthew, PODUNAVAC, Masa, MATA, Guillaume, ROSEN, Brandon Reid, HARDMAN, Clayton, FOURNIER, Jeremy, LIU, Dongdong, LAWSON, Kenneth Victor, YU, Kai, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich

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Inhibitors of HIF-2α and methods of use thereof von Gal, Balint, Yu, Kai, Liu, Dongdong, Mata, Guillaume, Epplin, Matthew, Mailyan, Artur Karenovich, Hardman, Clayton, Lawson, Kenneth Victor, Rosen, Brandon Reid, Podunavac, Ma{hacek over (s)}a, Drew, Samuel Lawrie, Powers, Jay Patrick, Fournier, Jeremy, Leleti, Manmohan Reddy, Beatty, Joel Worley

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Inhibitors of hif-2alpha and methods of use thereof von BEATTY Joel Worley, FOURNIER Jeremy, LIU Dongdong, YU Kai, LELETI Manmohan Reddy, HARDMAN Clayton, MATA Guillaume, GAL Balint, POWERS Jay Patrick, ROSEN Brandon Reid, MAILYAN Artur Karenovich, EPPLIN Matthew, LAWSON Kenneth Victor, DREW Samuel Lawrie, PODUNAVAC Ma?a

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INHIBITORS OF HIF-2ALPHA AND METHODS OF USE THEREOF von LELETI, Manmohan Reddy, DREW, Samuel Lawrie, EPPLIN, Matthew, MATA, Guillaume, ROSEN, Brandon Reid, HARDMAN, Clayton, FOURNIER, Jeremy, LIU, Dongdong, PODUNAVAC, Maša, LAWSON, Kenneth Victor, YU, Kai, POWERS, Jay Patrick, BEATTY, Joel Worley, GAL, Balint, MAILYAN, Artur Karenovich

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N-METHYL-D-ASPARTIC ACID RECEPTOR MODULATORS von TRAYNELIS, Stephen F, EPPLIN, Matthew, MENALDINO, David, LIOTTA, Dennis C

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Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2alpha von Su, Yongli, Yan, Xuelei, Mailyan, Artur Karenovich, Rosen, Brandon Reid, Drew, Samuel Lawrie, Haelsig, Karl T, Lindsey, Erick Allen, Powers, Jay Patrick, Wang, Zhang, Fournier, Jeremy Thomas Andre, Leleti, Manmohan Reddy, Jeffrey, Jenna Leigh, Beatty, Joel Worley, Gal, Balint, Yu, Kai, Mata, Guillaume, Epplin, Matthew, Kalisiak, Jaroslaw, Hardman, Clayton, Lawson, Kenneth Victor, Mandal, Debashis, Guney, Tezcan, Tran, Anh Thu, Jacob, Steven Donald, Moon, Hyunyoung

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NEGATIVE ALLOSTERIC MODULATION OF GLUN3-CONTAINING N-METHYL-D-ASPARTATE RECEPTORS von SUMMER, Samantha, TRAYNELIS, Stephen F, JACOBS, Leon, EPPLIN, Matthew, MCCALLUM, Adam, YUAN, Hongjie, MENALDINO, David, LIOTTA, Dennis C

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NEGATIVE ALLOSTERIC MODULATION OF GLUN3-CONTAINING N-METHYL-D-ASPARTATE RECEPTORS von SUMMER, Samantha, TRAYNELIS, Stephen F, JACOBS, Leon, EPPLIN, Matthew, MCCALLUM, Adam, YUAN, Hongjie, MENALDINO, David, LIOTTA, Dennis C

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