746P Synergistic antitumor efficacy of INV-71 ROR gamma agonist with immune checkpoint inhibitor anti-PD-1 in a murine orthotopic 4T1 breast cancer model von Sebesta, C., Chung, V., El-Khoueiry, A.B., Tilley, J., Windsor, W., Stouch, T., Ellingboe, J., Zhang, C., Gaweco, A.

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Parallel solid-phase synthesis of vitronectin receptor (αvβ3) inhibitors von Gopalsamy, Ariamala, Yang, Hui, Ellingboe, John W, Kees, Kenneth L, Yoon, Jeanne, Murrills, Richard

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Discovery of Pyrano[3,4-b]indoles as Potent and Selective HCV NS5B Polymerase Inhibitors von Gopalsamy, Ariamala, Lim, Kitae, Ciszewski, Gregory, Park, Kaapjoo, Ellingboe, John W, Bloom, Jonathan, Insaf, Shabana, Upeslacis, Janis, Mansour, Tarek S, Krishnamurthy, Girija, Damarla, Murthy, Pyatski, Yelena, Ho, Douglas, Howe, Anita Y. M, Orlowski, Mark, Feld, Boris, O'Connell, John

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Prodrugs of CL316243: a selective β3-adrenergic receptor agonist for treating obesity and diabetes von Sum, F.W., Gilbert, A., Venkatesan, A.M., Lim, K., Wong, V., O'Dell, M., Francisco, G., Chen, Z., Grosu, G., Baker, J., Ellingboe, J., Malamas, M., Gunawan, I., Primeau, J., Largis, E., Steiner, K.

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Metabolites of the Angiotensin II Antagonist Tasosartan:  The Importance of a Second Acidic Group von Ellingboe, John W, Collini, Michael D, Quagliato, Dominick, Chen, James, Antane, Madelene, Schmid, Jean, Hartupee, Dale, White, Valerie, Park, C. Hyung, Tanikella, Tarak, Bagli, Jehan F

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Novel and Selective Calcitonin-Inducing Agents von Gilbert, Adam M, Caltabiano, Stephen, Roberts, Denise, Sum, Sam F. W, Francisco, Gerardo D, Lim, Kitae, Asselin, Magda, Ellingboe, John W, Kharode, Yogendra, Cannistraci, Anna, Francis, Rita, TrailSmith, Mark, Gralnick, David

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Class III antiarrhythmic activity of novel substituted 4-[(methylsulfonyl)amino]benzamides and sulfonamides von Ellingboe, John W, Spinelli, Walter, Winkley, Michael W, Nguyen, Thomas T, Parsons, Roderick W, Moubarak, Issam F, Kitzen, Jan M, Von Engen, Donna, Bagli, Jehan F

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Pyrido[2,3-d]pyrimidine Angiotensin II Antagonists von Ellingboe, John W, Antane, Madelene, Nguyen, Thomas T, Collini, Michael D, Antane, Schuyler, Bender, Reinhold, Hartupee, Dale, White, Valerie, McCallum, John

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Discovery of 5-Arylsulfonamido-3- (pyrrolidin-2-ylmethyl)-1H-indole Derivatives as Potent, Selective 5-HT6 Receptor Agonists and Antagonists von Cole, Derek C, Lennox, William J, Lombardi, Sabrina, Ellingboe, John W, Bernotas, Ronald C, Tawa, Gregory J, Mazandarani, Hossein, Smith, Deborah L, Zhang, Guoming, Coupet, Joseph, Schechter, Lee E

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Antihyperglycemic activity of novel substituted 3H-1,2,3,5-oxathiadiazole 2-oxides von Ellingboe, John W, Alessi, Thomas R, Dolak, Terence M, Nguyen, Thomas T, Tomer, John D, Guzzo, Frieda, Bagli, Jehan F, McCaleb, Michael L

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Synthesis and Structure−Activity Relationship of N-Substituted 4-Arylsulfonylpiperidine-4-hydroxamic Acids as Novel, Orally Active Matrix Metalloproteinase Inhibitors for the Treat... von Aranapakam, Venkatesan, Davis, Jamie M, Grosu, George T, Baker, Ellingboe, John, Zask, Arie, Levin, Jeremy I, Sandanayaka, Vincent P, Du, Mila, Skotnicki, Jerauld S, DiJoseph, John F, Sung, Amy, Sharr, Michele A, Killar, Loran M, Walter, Thomas, Jin, Guixian, Cowling, Rebecca, Tillett, Jeff, Zhao, Weiguang, McDevitt, Joseph, Xu, Zhang Bao

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Synthesis and Structure−Activity Relationship of α-Sulfonylhydroxamic Acids as Novel, Orally Active Matrix Metalloproteinase Inhibitors for the Treatment of Osteoarthritis von Aranapakam, Venkatesan, Grosu, George T, Davis, Jamie M, Hu, Baihua, Ellingboe, John, Baker, Jannie L, Skotnicki, Jerauld S, Zask, Arie, DiJoseph, John F, Sung, Amy, Sharr, Michele A, Killar, Loran M, Walter, Thomas, Jin, Guixian, Cowling, Rebecca

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Synthesis and Structure−Activity Relationships of 4-alkynyloxy Phenyl Sulfanyl, Sulfinyl, and Sulfonyl Alkyl Hydroxamates as Tumor Necrosis Factor-α Converting Enzyme and Matrix Me... von Venkatesan, Aranapakam M, Davis, Jamie M, Grosu, George T, Baker, Jannie, Zask, Arie, Levin, Jeremy I, Ellingboe, John, Skotnicki, Jerauld S, DiJoseph, John F, Sung, Amy, Jin, Guixian, Xu, Weixin, McCarthy, Diane Joseph, Barone, Dauphine

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Antihyperglycemic activity of novel naphthalenyl 3H-1,2,3,5-oxathiadiazole 2-oxides von ELLINGBOE, J. W, LOMBARDO, L. J, STEINER, K, MCCALEB, M. L, ALESSI, T. R, NGUYEN, T. T, GUZZO, F, GUINOSSO, C. J, BULLINGTON, J, BROWNE, E. N. C, BAGLI, J. F, WRENN, J

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Anterior pituitary, adrenal, and gonadal hormones during cocaine withdrawal von MENDELSON, J. H, TEOH, S. K, LANGE, U, MELLO, N. K, WEISS, R, SKUPNY, A, ELLINGBOE, J

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Synthesis and SAR of bis-statine based peptides as BACE 1 inhibitors von Hu, Baihua, Fan, Kristi Yi, Bridges, Kristie, Chopra, Rajiv, Lovering, Frank, Cole, Derek, Zhou, Ping, Ellingboe, John, Jin, Guixiang, Cowling, Rebecca, Bard, Jonathan

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Pyrazolo[1,5- a]pyrimidin-7-yl phenyl amides as novel anti-proliferative agents: parallel synthesis for lead optimization of amide region von Gopalsamy, Ariamala, Yang, Hui, Ellingboe, John W., Tsou, Hwei-Ru, Zhang, Nan, Honores, Erick, Powell, Dennis, Miranda, Miriam, McGinnis, John P., Rabindran, Sridhar K.

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Prolactin and cortisol levels following acute alcohol challenges in women with and without a family history of alcoholism von Lex, Barbara W., Ellingboe, James E., Siew Koon Teoh, Mendelson, Jack H., Rhoades, Erin

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Ion channel screening plates: design, construction, and maintenance von Mayer, Scott C, Butera, John A, Diller, David J, Dunlop, John, Ellingboe, John, Fan, Kristi Yi, Kaftan, Edward, Mekonnen, Belew, Mobilio, Dominick, Paslay, Jeff, Tawa, Gregory, Vasilyev, Dmitry, Bowlby, Mark R

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The Solid Phase Synthesis of Tri-Substituted Indoles von Collini, Michael D, Ellingboe, John W

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