Molecular mechanism of 7TM receptor activation : A global toggle switch model von SCHWARTZ, Thue W, FRIMURER, Thomas M, HOIST, Birgitte, ROSENKILDE, Mette M, ELLING, Christian E

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Common Structural Basis for Constitutive Activity of the Ghrelin Receptor Family von Holst, Birgitte, Holliday, Nicholas D., Bach, Anders, Elling, Christian E., Cox, Helen M., Schwartz, Thue W.

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The Cannabinoid CB1 Antagonist TM38837 With Limited Penetrance to the Brain Shows Reduced Fear-Promoting Effects in Mice von Micale, Vincenzo, Drago, Filippo, Noerregaard, Pia K, Elling, Christian E, Wotjak, Carsten T

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Peripheral selectivity of the novel cannabinoid receptor antagonist TM38837 in healthy subjects von Klumpers, Linda E., Fridberg, Marianne, Kam, Marieke L., Little, Paul B., Jensen, Niels Ole, Kleinloog, Hendrik D., Elling, Christian E., Gerven, Joop M. A.

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Metal Ion Site Engineering Indicates a Global Toggle Switch Model for Seven-transmembrane Receptor Activation von Elling, Christian E., Frimurer, Thomas M., Gerlach, Lars-Ole, Jorgensen, Rasmus, Holst, Birgitte, Schwartz, Thue W.

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Metal Ion-mediated Agonism and Agonist Enhancement in Melanocortin MC1 and MC4 Receptors von Holst, Birgitte, Elling, Christian E., Schwartz, Thue W.

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Efficacy in diet‐induced obese mice of the hepatotropic, peripheral cannabinoid 1 receptor inverse agonist TM38837 von Cooper, Martin E., Nørregaard, Pia K., Högberg, Thomas, Andersson, Gunnar, Receveur, Jean‐Marie, Linget, Jean‐Michel, Elling, Christian E.

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A physicogenetic method to assign ligand-binding relationships between 7TM receptors von Frimurer, Thomas M., Ulven, Trond, Elling, Christian E., Gerlach, Lars-Ole, Kostenis, Evi, Högberg, Thomas

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Characterization of G-Protein Coupled Receptor Kinase Interaction with the Neurokinin-1 Receptor Using Bioluminescence Resonance Energy Transfer von Jorgensen, Rasmus, Holliday, Nicholas D, Hansen, Jakob L, Vrecl, Milka, Heding, Anders, Schwartz, Thue W, Elling, Christian E

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Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation von Bellmann-Sickert, Kathrin, Elling, Christian E, Madsen, Andreas N, Little, Paul B, Lundgren, Karsten, Gerlach, Lars-Ole, Bergmann, Ralf, Holst, Birgitte, Schwartz, Thue W, Beck-Sickinger, Annette G

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Conversion of antagonist-binding site to metal-ion site in the tachykinin NK-1 receptor von Elling, Christian E, Nielsen, Søren Møller, Schwartz, Thue W

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Low brain CB1 receptor occupancy by a second generation CB1 receptor antagonist TM38837 in comparison with rimonabant in nonhuman primates: A PET study von Takano, Akihiro, Gulyás, Balázs, Varnäs, Katarina, Little, Paul Brian, Noerregaard, Pia K., Jensen, Niels Ole, Elling, Christian e., Halldin, Christer

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Characterization of Glucagon-Like Peptide-1 Receptor β-Arrestin 2 Interaction: A High-Affinity Receptor Phenotype von Jorgensen, Rasmus, Martini, Lene, Schwartz, Thue W, Elling, Christian E

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Beta-Arrestin2 as a Competitor for GRK2 Interaction with the GLP-1 Receptor upon Receptor Activation von Jorgensen, Rasmus, Norklit Roed, Sarah, Heding, Anders, Elling, Christian E.

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Conversion of agonist site to metal-ion chelator site in the β2-adrenergic receptor von Elling, Christian E., Thirstrup, Kenneth, Holst, Birgitte, Schwartz, Thue W.

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Partial Agonism through a Zinc-Ion Switch Constructed between Transmembrane Domains III and VII in the Tachykinin NK1 Receptor von Birgitte Holst, Christian E. Elling, Thue W. Schwartz

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Construction of covalently coupled, concatameric dimers of 7TM receptors von Terpager, Marie, Scholl, D. Jason, Kubale, Valentina, Martini, Lene, Elling, Christian E., Schwartz, Thue W.

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Steric Hindrance Mutagenesis versus Alanine Scan in Mapping of Ligand Binding Sites in the Tachykinin NK1 Receptor von Holst, B, Zoffmann, S, Elling, C E, Hjorth, S A, Schwartz, T W

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Disulfide Bridge Engineering in the Tachykinin NK1 Receptor von Elling, Christian E, Raffetseder, Ute, Nielsen, Søren Møller, Schwartz, Thue W

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Peripheral selectivity of the novel cannabinoid receptor antagonist TM 38837 in healthy subjects von Klumpers, Linda E., Fridberg, Marianne, de Kam, Marieke L., Little, Paul B., Jensen, Niels Ole, Kleinloog, Hendrik D., Elling, Christian E., van Gerven, Joop M. A.

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