Potential Tumor-Selective Nitroimidazolylmethyluracil Prodrug Derivatives:  Inhibitors of the Angiogenic Enzyme Thymidine Phosphorylase von Cole, Christian, Reigan, Philip, Gbaj, Abdul, Edwards, Philip N, Douglas, Kenneth T, Stratford, Ian J, Freeman, Sally, Jaffar, Mohammed

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Design, synthesis and enzymatic evaluation of 6-bridged imidazolyluracil derivatives as inhibitors of human thymidine phosphorylase von McNally, Virginia A., Rajabi, Mehdi, Gbaj, Abdul, Stratford, Ian J., Edwards, Philip N., Douglas, Kenneth T., Bryce, Richard A., Jaffar, Mohammed, Freeman, Sally

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Discovery of novel inhibitors of Trypanosoma cruzi trans-sialidase from in silico screening von Neres, João, Brewer, Mark L., Ratier, Laura, Botti, Horacio, Buschiazzo, Alejandro, Edwards, Philip N., Mortenson, Paul N., Charlton, Michael H., Alzari, Pedro M., Frasch, Alberto C., Bryce, Richard A., Douglas, Kenneth T.

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A kinetic, modeling and mechanistic re-analysis of thymidine phosphorylase and some related enzymes von Edwards, Philip N.

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Benzoic acid and pyridine derivatives as inhibitors of Trypanosoma cruzi trans-sialidase von Neres, João, Bonnet, Pascal, Edwards, Philip N., Kotian, Pravin L., Buschiazzo, Alejandro, Alzari, Pedro M., Bryce, Richard A., Douglas, Kenneth T.

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Aminoimidazolylmethyluracil Analogues as Potent Inhibitors of Thymidine Phosphorylase and Their Bioreductive Nitroimidazolyl Prodrugs von Reigan, Philip, Edwards, Philip N, Gbaj, Abdul, Cole, Christian, Barry, Simon T, Page, Ken M, Ashton, Susan E, Luke, Richard W. A, Douglas, Kenneth T, Stratford, Ian J, Jaffar, Mohammed, Bryce, Richard A, Freeman, Sally

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Thymidine phosphorylase from Escherichia coli: Tight-binding inhibitors as enzyme active-site titrants von Gbaj, Abdul, Edwards, Philip N., Reigan, Philip, Freeman, Sally, Jaffar, Mohammed, Douglas, Kenneth T.

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The preclinical pharmacology of “Arimidex” (Anastrozole; ZD1033) — a potent, selective aromatase inhibitor von Dukes, Michael, Edwards, Philip N., Large, Michael, Smith, Ian K., Boyle, Thomas

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Methoxytetrahydropyrans. A new series of selective and orally potent 5-lipoxygenase inhibitors von Crawley, Graham C, Dowell, Robert I, Edwards, Philip N, Foster, Stephen J, McMillan, Rodger M, Walker, Edward R. H, Waterson, David, Bird, T. Geoffrey C, Bruneau, Pierre, Girodeau, Jean Marc

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Reversible acylation of elastase by γ-lactam analogues of β-lactam inhibitors von Westwood, Nicholas J, Claridge, Timothy D.W, Edwards, Philip N, Schofield, Christopher J

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A kinetic, modeling and mechanistic re-analysis of thymidine phosphorylase and some related enzymes: REVIEW ARTICLE von Edwards, Philip N.

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4-Methoxy-2-methyltetrahydropyrans: chiral leukotriene biosynthesis inhibitors, related to ICI D2138, which display enantioselectivity von Crawley, Graham C, Briggs, Malcolm T, Dowell, Robert I, Edwards, Philip N, Hamilton, Patricia M, Kingston, John F, Oldham, Keith, Waterson, David, Whalley, David P

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Prodrugs based on masked lactones. Cyclization of .gamma.-hydroxy amides von Johnson, C. David, Lane, Simon, Edwards, Philip N, Taylor, Peter J

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Inhibition of prolyl 4-hydroxylase in vitro and in vivo by members of a novel series of phenanthrolinones von FRANKLIN, Trevor J., MORRIS, William P., EDWARDS, Philip N., LARGE, Michael S., STEPHENSON, Robert

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Inhibition of prolyl 4-hydroxylase in vitro and in vivo by members of a novel series of phenanthrolinones von Franklin, T J, Morris, W P, Edwards, P N, Large, M S, Stephenson, R

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Conformational and tautomeric studies of acylguanidines. Part 1. Synthesis, ultraviolet spectroscopy, tautomeric preference, and site of protonation in some model compounds von Greenhill, John V., Ismail, M. Jamil, Edwards, Philip N., Taylor, Peter J.

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Conformational and tautomeric studies of acylguanidines. Part 2. Vibrational and carbon-13 nuclear magnetic resonance spectroscopy von Greenhill, John V., Ismail, M. Jamil, Bedford, Geoffrey R., Edwards, Philip N., Taylor, Peter J.

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Reactions of tetrafluoroethene oligomers. Part 7. Some reactions of 4-diazo-1,1,1,2,2-pentafluoro-3-pentafluoroethyl-3-trifluoromethylbutane von Coe, Paul L., Cook, Michael I., Goodchild, Nicholas J., Edwards, Philip N.

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Biosynthesis of The Non-Tryptophan Derived Portion of Ajmaline von Leete, Edward, Ghosal, Shibnath, Edwards, Philip N

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Covalent hydrates as intermediates in heterocyclic rearrangements. Part 3. The alkali-catalysed transformations of 1,5-diamino-1H-s-triazolo[1,5-c]quinazolinium bromide von Bowie, Raymond A., Edwards, Philip N., Nicholson, Stuart, Taylor, Peter J., Thomson, Douglas A.

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