Synthesis and Activity of New Aryl- and Heteroaryl-Substituted Pyrazole Inhibitors of the Transforming Growth Factor-β Type I Receptor Kinase Domain von Sawyer, J. Scott, Anderson, Bryan D, Beight, Douglas W, Campbell, Robert M, Jones, Michael L, Herron, David K, Lampe, John W, McCowan, Jefferson R, McMillen, William T, Mort, Nicholas, Parsons, Stephen, Smith, Edward C. R, Vieth, Michal, Weir, Leonard C, Yan, Lei, Zhang, Faming, Yingling, Jonathan M

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Design and Synthesis of a Novel Series of 1,2-Disubstituted Cyclopentanes as Small, Potent Potentiators of 2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propanoic Acid (AMPA) Recepto... von Shepherd, Timothy A, Aikins, James A, Bleakman, David, Cantrell, Buddy E, Rearick, John P, Simon, Richard L, Smith, Edward C. R, Stephenson, Gregory A, Zimmerman, Dennis M, Mandelzys, Allan, Jarvie, Keith R, Ho, Ken, Deverill, Michelle, Kamboj, Rajender K

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Carbocyclic[g]indole Inhibitors of Human Nonpancreatic s-PLA2 von Sawyer, J. Scott, Beight, Douglas W, Smith, Edward C. R, Snyder, David W, Chastain, Marcia K, Tielking, Richard L, Hartley, Lawrence W, Carlson, Donald G

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Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain von SAWYER, J. Scott, BEIGHT, Douglas W, PARSONS, Stephen, SMITH, Edward C. R, WAGNER, Jill R, LEI YAN, FAMING ZHANG, YINGLING, Jonathan M, BRITT, Karen S, ANDERSON, Bryan D, CAMPBELL, Robert M, GOODSON, Theodore JR, HERRON, David K, LI, Hong-Yu, MCMILLEN, William T, MORT, Nicholas

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3-Phenyl-4-hydroxyquinolin-2(1H)-ones: potent and selective antagonists at the strychnine-insensitive glycine site on the N-methyl-D-aspartate receptor complex von McQuaid, Loretta A, Smith, Edward C. R, Lodge, David, Pralong, Etienne, Wikel, James H, Calligaro, David O, O'Malley, Patrick J

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Diethyl 2,4-dioxoimidazolidine-5-phosphonates: Horner-Wadsworth-Emmons reagents for the mild and efficient preparation of C-5 unsaturated hydantoin derivatives von Meanwell, Nicholas A, Roth, Herbert R, Smith, Edward C. R, Wedding, Donald L, Wright, J. J. Kim

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Synthesis and excitatory amino acid pharmacology of a series of heterocyclic-fused quinoxalinones and quinazolinones von McQuaid, Loretta A, Smith, Edward C. R, South, Kimberly K, Mitch, Charles H, Schoepp, Darryle D, True, Rebecca A, Calligaro, David O, O'Malley, Patrick J, Lodge, David, Ornstein, Paul L

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1,3-Dihydro-2H-imidazo[4,5-b]quinolin-2-ones - inhibitors of blood platelet cAMP phosphodiesterase and induced aggregation von Meanwell, Nicholas A, Roth, Herbert R, Smith, Edward C. R, Wedding, Donald L, Wright, J. J. Kim, Fleming, J. Stuart, Gillespie, Elizabeth

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An enantioselective synthesis of D-(-)- and L-(+)-2-amino-3-phosphonopropanoic acid von Smith, Edward C. R, McQuaid, Loretta A, Paschal, Jonathan W, DeHoniesto, Juel

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Synthesis and biological activity of structural analogs of the anticancer benzophenanthridine alkaloid nitidine chloride von Cushman, Mark, Mohan, Prem, Smith, Edward C. R

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Inhibitors of blood platelet cAMP phosphodiesterase. 2. Structure-activity relationships associated with 1,3-dihydro-2H-imidazo[4,5-b]quinolin-2-ones substituted with functionalize... von Meanwell, Nicholas A, Pearce, Bradley C, Roth, Herbert R, Smith, Edward C. R, Wedding, Donald L, Wright, J. J. Kim, Buchanan, John O, Baryla, Urzula M, Gamberdella, Marianne

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2-Amino- and 2-guanidino-1,2,3,4-tetrahydro-1,4-epoxynaphthalenes as conformationally defined analogs of .alpha.-adrenergic agents von Smith, Edward C. R, Riley, Thomas N, Borne, Ronald F, Waters, I. W

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Carbocyclic[ g ]indole Inhibitors of Human Nonpancreatic s-PLA 2 von Sawyer, J. Scott, Beight, Douglas W., Smith, Edward C. R., Snyder, David W., Chastain, Marcia K., Tielking, Richard L., Hartley, Lawrence W., Carlson, Donald G.

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Substituerte karboksamider, farmasøytiske sammensetninger omfattende slike og anvendelse von Smith, Edward C R, Backer, Ryan Thomas, Takeuchi, Kumiko, Kuklish, Steven Lee, Hollinshead, Sean Patrick, Fisher, Matthew Joseph

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composto ou um sal farmaceuticamente aceitável do mesmo, composição farmacêutica, e, uso de composto von PRABHAKAR KONDAJI JADHAV, DAVID ANDREW NEEL, EDWARD C. R. SMITH, DONALD PAUL MATTHEWS, JONATHAN EDWARD GREEN, KEVIN ROBERT FALES

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CARBOXAMIDES SUBSTITUES von TAKEUCHI, KUMIKO, BACKER, RYAN, THOMAS, HOLLINSHEAD, SEAN, PATRICK, FISHER, MATTHEW, JOSEPH, KUKLISH, STEVEN, LEE, SMITH, EDWARD, C, R

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Novel pyrrole derivatives as pharmaceutical agents von R,CIAPETTI PAOLA,SMITH EDWARD C. R, HERRON DAVID KENT,MORT NICOLAS ANTHONY,MCMILLEN WILLIAM THOMAS,DECOLLO TODD VINCENT,SAWYER JASON SCOTT,LIAO JUNKAI,GOODSON JR. THEODORE,GODFREY ALEXANDER GLENN,BEIGHT DOUGLAS WADE,YINGLING JONATHAN MI

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SUBSTITUTED CARBOXAMIDES AS GROUP 1 METABOTROPIC RECEPTOR ANTAGONISTS von KUKLISH, STEVEN LEE, BACKER, RYAN THOMAS, TAKEUCHI, KUMIKO, HOLLINSHEAD, SEAN PATRICK, FISHER, MATTHEW JOSEPH, SMITH, EDWARD C. R

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SUBSTITUTED CARBOXAMIDES AS GROUP I METABOTROPIC RECEPTOR ANTAGONISTS von TAKEUCHI, KUMIKO, BACKER, RYAN, THOMAS, HOLLINSHEAD, SEAN, PATRICK, FISHER, MATTHEW, JOSEPH, SMITH, EDWARD C. R, KUKLISH, STEVEN, LEE

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Tetrahydrocarbazole derivatives useful as androgen receptor modulators (SARM) von GREEN, JONATHAN EDWARD, MATTHEWS, DONALD PAUL, SMITH, EDWARD C R, JADHAV, PRABHAKAR KONDAJI, NEEL, DAVID ANDREW, FALES, KEVIN ROBERT

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