The design of non-peptide human bradykinin B2 receptor antagonists employing the benzodiazepine peptidomimetic scaffold von DZIADULEWICZ, E. K, BROWN, M. C, DUNSTAN, A. R, WAI LEE, SAID, N. B, GARRATT, P. J

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Bradyzide, a potent non‐peptide B 2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia von Burgess, Gillian M, Perkins, Martin N, Rang, Humphrey P, Campbell, Elizabeth A, Brown, Michael C, McIntyre, Peter, Urban, Laszlo, Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Wrigglesworth, Roger, Lee, Wai, Davis, Clare, Phagoo, Steve B, Davis, Andrew J, Phillips, Elsa, Drake, Gillian S, Hughes, Glyn A, Dunstan, Andrew, Bloomfield, Graham C

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Bradyzide, a potent non‐peptide B2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia von Burgess, Gillian M, Perkins, Martin N, Rang, Humphrey P, Campbell, Elizabeth A, Brown, Michael C, McIntyre, Peter, Urban, Laszlo, Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Wrigglesworth, Roger, Lee, Wai, Davis, Clare, Phagoo, Steve B, Davis, Andrew J, Phillips, Elsa, Drake, Gillian S, Hughes, Glyn A, Dunstan, Andrew, Bloomfield, Graham C

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Design of non-peptide CCK2 and NK1 peptidomimetics using 1-(2-nitrophenyl)thiosemicarbazide as a novel common scaffold von DZIADULEWICZ, Edward K, WALPOLE, Christopher S, SNELL, Christopher R, WRIGGLESWORTH, Roger, HUGHES, Glyn A, BEATTIE, David, WOOD, John N, BEECH, Margaret M, COOTE, Paul R

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Non-peptide ligands for bradykinin receptors 1995 - 2004 von Dziadulewicz, Edward K

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A Nonpeptide Antagonist Reveals a Highly Glycosylated State of the Rabbit Kinin B1 Receptor von Fortin, Jean-Philippe, Dziadulewicz, Edward K, Gera, Lajos, Marceau, François

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Identification and Biological Characterization of 6-Aryl-7-isopropylquinazolinones as Novel TRPV1 Antagonists that Are Effective in Models of Chronic Pain von Culshaw, Andrew J, Bevan, Stuart, Christiansen, Martin, Copp, Prafula, Davis, Andrew, Davis, Clare, Dyson, Alex, Dziadulewicz, Edward K, Edwards, Lee, Eggelte, Hendrikus, Fox, Alyson, Gentry, Clive, Groarke, Alex, Hallett, Allan, Hart, Terance W, Hughes, Glyn A, Knights, Sally, Kotsonis, Peter, Lee, Wai, Lyothier, Isabelle, McBryde, Andrew, McIntyre, Peter, Paloumbis, George, Panesar, Moh, Patel, Sadhana, Seiler, Max-Peter, Yaqoob, Mohammed, Zimmermann, Kaspar

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Mitsunobu alkylation of imidazole: a convenient route to chiral ionic liquids von Kim, Eun Jin, Ko, Soo Y., Dziadulewicz, Edward K.

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A Nonpeptide Antagonist Reveals a Highly Glycosylated State of the Rabbit Kinin B 1 Receptor von Fortin, Jean-Philippe, Dziadulewicz, Edward K., Gera, Lajos, Marceau, François

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Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone: A Potent, Orally Bioavailable Human CB sub(1)/CB sub(2) Dual Agonist with Antihyperalgesic Properties and Restricted Central... von Dziadulewicz, E K, Bevan, S J, Brain, C T, Coote, PR, Culshaw, A J, Davis, A J, Edwards, L J, Fisher, A J, Fox, A J, Gentry, C, Groarke, A, Hart, T W, Huber, W, James, I F

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A non-peptide antagonist unusually selective for the human form of the bradykinin B sub(2) receptor von Marceau, F, tin, J-P, Morissette, G, Dziadulewicz, E K

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1-(2-Nitrophenyl)thiosemicarbazides:  A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B2 Receptor von Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Ko, Soo Y, Wrigglesworth, Roger, Hughes, Glyn A, Dunstan, Andrew R, Bloomfield, Graham C, Drake, Gillian S, Brown, Michael C, Lee, Wai, Burgess, Gillian M, Davis, Clare, Yaqoob, Mohammed, Perkins, Martin N, Campbell, Elizabeth A, Davis, Andrew J, Rang, Humphrey P

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Potent and Orally Bioavailable Non-Peptide Antagonists at the Human Bradykinin B 1 Receptor Based on a 2-Alkylamino-5-sulfamoylbenzamide Core von Ritchie, Timothy J., Dziadulewicz, Edward K., Culshaw, Andrew J., Müller, Werner, Burgess, Gillian M., Bloomfield, Graham C., Drake, Gillian S., Dunstan, Andrew R., Beattie, David, Hughes, Glyn A., Ganju, Pam, McIntyre, Peter, Bevan, Stuart J., Davis, Clare, Yaqoob, Mohammed

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A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor von MARCEAU, Francois, FORTIN, Jean-Philippe, MORISSETTE, Guillaume, DZIADULEWICZ, Edward K

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Effects of two novel non-peptide antagonists at the rabbit bradykinin B2 receptor von Marceau, F, Houle, S, Bouthillier, J, Said, N B, Garratt, P J, Dziadulewicz, E K

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A non-peptide antagonist unusually selective for the human form of the bradykinin B 2 receptor von Marceau, François, Fortin, Jean-Philippe, Morissette, Guillaume, Dziadulewicz, Edward K.

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Concise and regiospecific syntheses of tri-substituted 1,2,4-triazoles von Dunstan, Andrew R, Weber, Hans-Peter, Rihs, Grety, Widmer, Hans, Dziadulewicz, Edward K

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Nonpeptide Bradykinin B 2 Receptor Antagonists:  Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B 2 Receptor Antagonists von Dziadulewicz, Edward K., Ritchie, Timothy J., Hallett, Allan, Snell, Christopher R., Davies, John W., Wrigglesworth, Roger, Dunstan, Andrew R., Bloomfield, Graham C., Drake, Gillian S., McIntyre, Peter, Brown, Michael C., Burgess, Gillian M., Lee, Wai, Davis, Clare, Yaqoob, Mohammed, Phagoo, Steve B., Phillips, Elsa, Perkins, Martin N., Campbell, Elizabeth A., Davis, Andrew J., Rang, Humphrey P.

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1-(2-Nitrophenyl)thiosemicarbazides:  A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B 2 Receptor von Dziadulewicz, Edward K., Ritchie, Timothy J., Hallett, Allan, Snell, Christopher R., Ko, Soo Y., Wrigglesworth, Roger, Hughes, Glyn A., Dunstan, Andrew R., Bloomfield, Graham C., Drake, Gillian S., Brown, Michael C., Lee, Wai, Burgess, Gillian M., Davis, Clare, Yaqoob, Mohammed, Perkins, Martin N., Campbell, Elizabeth A., Davis, Andrew J., Rang, Humphrey P.

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Potent and orally bioavailable non-peptide antagonists at the human bradykinin B(1) receptor based on a 2-alkylamino-5-sulfamoylbenzamide core von Ritchie, Timothy J, Dziadulewicz, Edward K, Culshaw, Andrew J, Müller, Werner, Burgess, Gillian M, Bloomfield, Graham C, Drake, Gillian S, Dunstan, Andrew R, Beattie, David, Hughes, Glyn A, Ganju, Pam, McIntyre, Peter, Bevan, Stuart J, Davis, Clare, Yaqoob, Mohammed

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