Synthesis and Evaluation of Bicyclic Hydroxypyridones as Inhibitors of Catechol O‑Methyltransferase von Ernst, Glen, Akuma, Daniel, Au, Vinh, Buchler, Ingrid P, Byers, Spencer, Carr, Gregory V, Defays, Sabine, de León, Pablo, Demaude, Thierry, DePasquale, Michael, Durieu, Véronique, Huang, Yifang, Jigorel, Emilie, Kimos, Martha, Kolobova, Anna, Montel, Florian, Moureau, Florence, Poslusney, Michael, Swinnen, Dominique, Vandergeten, Marie-Christine, Van houtvin, Nathalie, Wei, Huijun, White, Noelle, Wood, Martyn, Barrow, James C

Volltext

Lead Optimization of Thiazolo[5,4-c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H3R Inverse Agonists von Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie

Volltext

Acetamide Scanning around Bicyclic Thiazoles: SAR at the H 3 Receptor von Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean‐Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent

Volltext

Phenyl‐oxazoles, a New Family of Inverse Agonists at the H 3 Histamine Receptor von Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie‐Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent

Volltext

Discovery of a New Class of Non‐imidazole Oxazoline‐Based Histamine H 3 Receptor (H 3 R) Inverse Agonists von Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean‐Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent

Volltext

First dual M sub(3) antagonists-PDE4 inhibitors: Synthesis and SAR of 4,6- diaminopyrimidine derivatives von Provins, Laurent, Christophe, Bernard, Danhaive, Pierre, Dulieu, Jacques, Durieu, Veronique, Gillard, Michel, Lebon, Florence, Lengele, Sebastien, Quere, Luc, Van Keulen, BerendJan

Volltext

Phenyl-oxazoles, a New Family of Inverse Agonists at the H3 Histamine Receptor von Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent

Volltext

First dual M3 antagonists-PDE4 inhibitors : Synthesis and SAR of 4,6-diaminopyrimidine derivatives von PROVINS, Laurent, CHRISTOPHE, Bernard, DANHAIVE, Pierre, DULIEU, Jacques, DURIEU, Véronique, GILLARD, Michel, LEBON, Florence, LENGELE, Sébastien, QUERE, Luc, VAN KEULEN, Berendjan

Volltext

Lead Optimization of Thiazolo[5,4‐ c ]piperidines: 3‐Cyclobutoxy Linker as a Key Spacer for H 3 R Inverse Agonists von Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie

Volltext

First dual M 3 antagonists-PDE4 inhibitors: Synthesis and SAR of 4,6-diaminopyrimidine derivatives von Provins, Laurent, Christophe, Bernard, Danhaive, Pierre, Dulieu, Jacques, Durieu, Véronique, Gillard, Michel, Lebon, Florence, Lengelé, Sébastien, Quéré, Luc, van Keulen, BerendJan

Volltext

Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor von Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean-Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent

Volltext

Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists von Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van Houtvin, Nathalie

Volltext

Discovery of a New Class of Non-imidazole Oxazoline-Based Histamine H3 Receptor (H3R) Inverse Agonists von Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean-Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent

Volltext

COMPOUNDS COMPRISING A CYCLOBUTOXY GROUP von DENONNE, FREDERIC, VALADE, ANNE, DEFAYS, SABINE, CELANIRE, SYLVAIN, DURIEU, VERONIQUE

Volltext bestellen

Fused tricyclic benzimidazoles derivatives as modulators of TNF activity von Deligny Michael, Jackson Victoria Elizabeth, Selby Matthew Duncan, Keyaerts Jean, Durieu Veronique, Alexander Rikki Peter, Heer Jag Paul, Kroeplien Boris, Sabnis Yogesh Anil, Calmiano Mark Daniel, Heinelt Uwe, Swinnen Dominique Louis Leon, Van Houtvin Nathalie, Wehner Volkmar, Mac Coss Malcolm, Defays Sabine, Zhu Zhaoning

Volltext bestellen

Compounds Comprising A Cyclobutoxy Group von CELANIRE SYLVAIN, DENONNE FREDERIC, DEFAYS SABINE, DURIEU VERONIQUE, VALADE ANNE

Volltext bestellen

COMPOUNDS COMPRISING A CYCLOBUTOXY GROUP von DENONNE, FREDERIC, VALADE, ANNE, DEFAYS, SABINE, CELANIRE, SYLVAIN, DURIEU, VERONIQUE

Volltext bestellen

Compounds comprising a cyclobutoxy group von SYLVAIN CELANIRE, ANNE VALADE, FREDERIC DENONNE, SABINE DEFAYS, VERONIQUE DURIEU

Volltext bestellen

Phenyl-oxazoles, a new family of inverse agonists at the H(3) histamine receptor von Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van Houtvin, Nathalie, Verbois, Valérie, Provins, Laurent

Volltext

Fused Tricyclic Benzimidazoles Derivatives As Modulators of TNF Activity von Deligny Michael, Jackson Victoria Elizabeth, Selby Matthew Duncan, Keyaerts Jean, Durieu Veronique, Alexander Rikki Peter, Heer Jag Paul, Kroeplien Boris, Sabnis Yogesh Anil, Calmiano Mark Daniel, Heinelt Uwe, Swinnen Dominique Louis Leon, Van Houtvin Nathalie, Wehner Volkmar, Mac Coss Malcolm, Defays Sabine, Zhu Zhaoning

Volltext bestellen