PK 11195, an antagonist of peripheral benzodiazepine receptors, reduces ventricular arrhythmias during myocardial ischemia and reperfusion in the dog von Mestre, Michel, Bouetard, Giséle, Uzan, André, Gueremy, Claude, Renault, Christian, Dubroeucq, Marie-Christine, Le Fur, Gérard

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Labelling of “Peripheral‐Type” Benzodiazepine Binding Sites in the Rat Brain By Using [3H]PK 11195, an Isoquinoline Carboxamide Derivative: Kinetic Studies and Autoradiographic Loc... von Benavides, J., Quarteronet, D., Imbault, F., Malgouris, C., Uzan, A., Renault, C., Dubroeucq, M. C., Gueremy, C., Fur, G. Le

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Photoaffinity labeling of peripheral-type benzodiazepine-binding sites von DOBLE, A, FERRIS, O, BURGEVIN, M. C, MENAGER, J, UZAN, A, DUBRŒUCQ, M. C, RENAULT, C, GUEREMY, C, LE FUR, G

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Peripheral benzodiazepine binding sites: Effect of PK 11195, 1-(2-chlorophenyl)-n-methyl-n-(1-methylpropyl)-3-isoquinolinecarboxamide: I. In vitro studies von Le Fur, G., Perrier, M.L., Vaucher, N., Imbault, F., Flamier, A., Benavides, J., Uzan, A., Renault, C., Dubroeucq, M.C., Guérémy, C.

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Modulation of voltage-operated, but not receptor-operated, calcium channels in the rabbit aorta by PK 11195, an antagonist of peripheral-type benzodiazepine receptors von MESTRE, M, BELIN, C, UZAN, A, RENAULT, C, DUBRŒUCQ, M.-C, GUEREMY, C, LE FUR, G

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Electrophysiological and pharmacological evidence that peripheral type benzodiazepine receptors are coupled to calcium channels in the heart von Mestre, M., Carriot, T., Belin, C., Uzan, A., Renault, C., Dubroeucq, M.C., Guérémy, C., Doble, A., Le Fur, G.

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In vivo labelling in several rat tissues of ‘peripheral type’ benzodiazepine binding sites von Benavides, Jesus, Guilloux, Françoise, Rufat, Pierre, Uzan, Andre, Renault, Christian, Dubroeucq, Marie-Christine, Gueremy, Claude, Le Fur, Gerard

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Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation von Mestre, M., Carriot, T., Belin, C., Uzan, A., Renault, C., Dubroeucq, M.C., Guérémy, C., Le Fur, G.

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Synthesis and pharmacological properties of 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, a new competitive AMPA/KA receptor antagonist von Mignani, Serge, Aloup, Jean-Claude, Barreau, Michel, Blanchard, Jean Charles, Böhme, Georg Andrees, Boireau, Alain, Damour, Dominique, Debono, Marc-Williams, Dubroeucq, Marie-Christine, Genevois-Borella, Arielle, Imperato, Assunta, Jimonet, Patrick, Pratt, Jeremy, Randle, John C.R., Reibaud, Michel, Ribeill, Yves, Stutzmann, Jean-Marie

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Peripheral benzodiazepine binding sites: Effect of PK 11195, 1-(2-chlorophenyl)-n-methyl-(1-methylpropyl)-3 isoquinolinecarboxamide: II. In vivo studies von Le Fur, G., Guilloux, F., Rufat, P., Benavides, J., Uzan, A., Renault, C., Dubroeucq, M.C., Guérémy, C.

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The Ureidoacetamides, a Novel Family of Non-peptide CCK-B/Gastrin Antagonists von BÖHME, G. A., BERTRAND, P., GUYON, C., CAPET, M., PENDLEY, C., STUTZMANN, J. M., DOBLE, A., DUBROEUCQ, M. C., MARTIN, G., BLANCHARD, J. C.

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Partial Purification and Pharmacology of Peripheral-Type Benzodiazepine Receptors von Doble, A., Burgevin, M. C., MÉNager, J., Ferris, O., BÉGassat, F., Renault, C., Dubroeucq, M. C., GuÉRÉMy, C., Uzan, A., Fur, G. Le

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Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat von Mizoule, J., Gauthier, A., Uzan, A., Renault, C., Dubroeucq, M.C., Guéremy, C., Le Fur, G.

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Opposite effects of an agonist, RO5-4864, and an antagonist, PK 11195, of the peripheral type benzodiazepine binding sites on audiogenic seizures in DBA/2J mice von Bénavidès, J, Guilloux, F, Allam, D E, Uzan, A, Mizoule, J, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G

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Autoradiographic localization of peripheral benzodiazepine binding sites in the cat brain with [ 3H]PK 11195 von Bénavidès, J., Savaki, H.E., Malgouris, C., Laplace, C., Daniel, M., Begassat, F., Desban, M., Uzan, A., Dubroeucq, M.C., Renault, C., Guérémy, C., Le Fur, G.

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Stereoselective inhibition of the binding of [ 3H]PK 11195 to peripheral-type benzodiazepine binding sites by a quinolinepropanamide derivative von Dubroeucq, Marie-Christine, Bénavidès, Jesus, Doble, Adam, Guilloux, Françoise, Allam, Djamal, Vaucher, Nadine, Bertrand, Philippe, Guérémy, Claude, Renault, Christian, Uzan, Andre, Le Fur, Gérard

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Evaluation of Brain Penetration of CCK-B Antagonists von DBROEUCQ, M. C., GUYON, C., MANFRÉ, F., CAPET, M., BARREAU, M., BERTRAND, P., JEANTAUD, B., DOBLE, A., BLANCHARD, J.-C.

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PK 11195, an antagonist of peripheral type benzodiazepine receptors, modulates bay K8644 sensitive but not β- or H2-receptor sensitive voltage operated calcium channels in the guin... von MESTRE, M, CARRIOT, T, NELIAT, G, UZAN, A, RENAULT, C, DUBRŒUCQ, M. C, GUEREMY, C, DOBLE, A, LE FUR, G

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Histidine modification with diethylpyrocarbonate induces a decrease in the binding of an antagonist, PK 11195, but not of an agonist, RO5-4864, of the peripheral benzodiazepine rec... von Bénavidès, J, Begassat, F, Phan, T, Tur, C, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G

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Differentiation between two ligands for peripheral benzodiazepine binding sites, [ 3H]R05-4864 and [ 3H]PK 11195, by thermodynamic studies von Le Fur, G., Vaucher, N., Perrier, M.L., Flamier, A., Benavides, J., Renault, C., Dubroeucq, M.C., Guérémy, C., Uzan, A.

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