Degradation of Polycomb Repressive Complex 2 with an EED-Targeted Bivalent Chemical Degrader von Potjewyd, Frances, Turner, Anne-Marie W., Beri, Joshua, Rectenwald, Justin M., Norris-Drouin, Jacqueline L., Cholensky, Stephanie H., Margolis, David M., Pearce, Kenneth H., Herring, Laura E., James, Lindsey I.

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Identification of a cell-active chikungunya virus nsP2 protease inhibitor using a covalent fragment-based screening approach von Merten, Eric M, Sears, John D, Leisner, Tina M, Hardy, P Brian, Ghoshal, Anirban, Hossain, Mohammad Anwar, Asressu, Kesatebrhan Haile, Brown, Peter J, Tse, Edwin G, Stashko, Michael A, Li, Kelin, Norris-Drouin, Jacqueline L, Herring, Laura E, Mordant, Angie L, Webb, Thomas S, Mills, Christine A, Barker, Natalie K, Streblow, Zachary J, Perveen, Sumera, Arrowsmith, Cheryl H, Couñago, Rafael Miguez, Arnold, Jamie J, Cameron, Craig E, Streblow, Daniel N, Moorman, Nathaniel J, Heise, Mark T, Willson, Timothy M, Popov, Konstantin I, Pearce, Kenneth H

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Identification of Covalent Cyclic Peptide Inhibitors in mRNA Display von Iskandar, Sabrina E., Chiou, Lilly F., Leisner, Tina M., Shell, Devan J., Norris-Drouin, Jacqueline L., Vaziri, Cyrus, Pearce, Kenneth H., Bowers, Albert A.

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Discovery of CHD1 Antagonists for PTEN-Deficient Prostate Cancer von Johnson, Rebecca L., Graboski, Amanda L., Li, Fengling, Norris-Drouin, Jacqueline L., Walton, William G., Arrowsmith, Cheryl H., Redinbo, Matthew R., Frye, Stephen V., James, Lindsey I.

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Discovery and Structural Basis of the Selectivity of Potent Cyclic Peptide Inhibitors of MAGE-A4 von Fleming, Matthew C., Chiou, Lilly F., Tumbale, Percy P., Droby, Gaith N., Lim, Jiwoong, Norris-Drouin, Jacqueline L., Williams, Jason G., Pearce, Kenneth H., Williams, R. Scott, Vaziri, Cyrus, Bowers, Albert A.

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Comparisons between Manual Lymph Drainage, Abdominal Massage, and Electrical Stimulation on Functional Constipation Outcomes: A Randomized, Controlled Trial von Drouin, Jacqueline S., Pfalzer, Lucinda, Shim, Jung Myo, Kim, Seong Jung

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IRE1α Is a Therapeutic Target for Cystic Fibrosis Airway Inflammation von Hull-Ryde, Emily A, Minges, John T, Martino, Mary E B, Kato, Takafumi, Norris-Drouin, Jacqueline L, Ribeiro, Carla M P

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Discovery of an H3K36me3-Derived Peptidomimetic Ligand with Enhanced Affinity for Plant Homeodomain Finger Protein 1 (PHF1) von Engelberg, Isabelle A, Liu, Jiuyang, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Ottavi, Samantha A, Frye, Stephen V, Kutateladze, Tatiana G, James, Lindsey I

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Discovery of a 53BP1 Small Molecule Antagonist Using a Focused DNA-Encoded Library Screen von Shell, Devan J., Foley, Caroline A., Wang, Qinhong, Smith, Chelsea M., Guduru, Shiva K. R., Zeng, Hong, Dong, Aiping, Norris-Drouin, Jacqueline L., Axtman, Matthew, Hardy, P. Brian, Gupta, Gaorav, Halabelian, Levon, Frye, Stephen V., James, Lindsey I., Pearce, Kenneth H.

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PROTAC Linkerology Leads to an Optimized Bivalent Chemical Degrader of Polycomb Repressive Complex 2 (PRC2) Components von Bashore, Frances M., Foley, Caroline A., Ong, Han Wee, Rectenwald, Justin M., Hanley, Ronan P., Norris-Drouin, Jacqueline L., Cholensky, Stephanie H., Mills, Christine A., Pearce, Kenneth H., Herring, Laura E., Kireev, Dmitri, Frye, Stephen V., James, Lindsey I.

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Structure–Activity Relationships and Kinetic Studies of Peptidic Antagonists of CBX Chromodomains von Stuckey, Jacob I, Simpson, Catherine, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Lee, Junghyun, Pasca, Ryan, Cheng, Nancy, Dickson, Bradley M, Pearce, Kenneth H, Frye, Stephen V, James, Lindsey I

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Design and Construction of a Focused DNA-Encoded Library for Multivalent Chromatin Reader Proteins von Rectenwald, Justin M, Guduru, Shiva Krishna Reddy, Dang, Zhao, Collins, Leonard B, Liao, Yi-En, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Kaufmann, Kyle W, Hammond, Scott M, Kireev, Dmitri B, Frye, Stephen V, Pearce, Kenneth H

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Cdyl Deficiency Brakes Neuronal Excitability and Nociception through Promoting Kcnb1 Transcription in Peripheral Sensory Neurons von Sun, Zhao‐Wei, Waybright, Jarod M., Beldar, Serap, Chen, Lu, Foley, Caroline A., Norris‐Drouin, Jacqueline L., Lyu, Tian‐Jie, Dong, Aiping, Min, Jinrong, Wang, Yu‐Pu, James, Lindsey I., Wang, Yun

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Cdyl Deficiency Brakes Neuronal Excitability and Nociception through Promoting Kcnb1 Transcription in Peripheral Sensory Neurons von Sun, Zhao‐Wei, Waybright, Jarod M., Beldar, Serap, Chen, Lu, Foley, Caroline A., Norris‐Drouin, Jacqueline L., Lyu, Tian‐Jie, Dong, Aiping, Min, Jinrong, Wang, Yu‐Pu, James, Lindsey I., Wang, Yun

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SETDB1 Triple Tudor Domain Ligand, (R,R)‑59, Promotes Methylation of Akt1 in Cells von Uguen, Mélanie, Deng, Yu, Li, Fengling, Shell, Devan J., Norris-Drouin, Jacqueline L., Stashko, Michael A., Ackloo, Suzanne, Arrowsmith, Cheryl H., James, Lindsey I., Liu, Pengda, Pearce, Kenneth H., Frye, Stephen V.

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Discovery of Peptidomimetic Ligands of EED as Allosteric Inhibitors of PRC2 von Barnash, Kimberly D, The, Juliana, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Worley, Beau M, Li, Fengling, Stuckey, Jacob I, Brown, Peter J, Vedadi, Masoud, Arrowsmith, Cheryl H, Frye, Stephen V, James, Lindsey I

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Magnitude of late effects of breast cancer treatments on shoulder function: a systematic review von Levangie, Pamela K, Drouin, Jacqueline

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A Peptidomimetic Ligand Targeting the Chromodomain of MPP8 Reveals HRP2’s Association with the HUSH Complex von Waybright, Jarod M, Clinkscales, Sarah E, Barnash, Kimberly D, Budziszewski, Gabrielle R, Rectenwald, Justin M, Chiarella, Anna M, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Pearce, Kenneth H, Herring, Laura E, McGinty, Robert K, Hathaway, Nathaniel A, James, Lindsey I

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Discovery of Macrocyclic Pyrimidines as MerTK‐Specific Inhibitors von McIver, Andrew L., Zhang, Weihe, Liu, Qingyang, Jiang, Xinpeng, Stashko, Michael A., Nichols, James, Miley, Michael J., Norris‐Drouin, Jacqueline, Machius, Mischa, DeRyckere, Deborah, Wood, Edgar, Graham, Douglas K., Earp, H. Shelton, Kireev, Dmitri, Frye, Stephen V., Wang, Xiaodong

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Discovery and Characterization of Peptide Inhibitors for Calcium and Integrin Binding Protein 1 von Puhl, Ana C, Bogart, Jonathan W, Haberman, Victoria A, Larson, Jacob E, Godoy, Andre S, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Leisner, Tina M, Frye, Stephen V, Parise, Leslie V, Bowers, Albert A, Pearce, Kenneth H

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