Unprecedented Catalytic Three Component One-Pot Condensation Reaction:  An Efficient Synthesis of 5-Alkoxycarbonyl- 4-aryl-3,4-dihydropyrimidin-2(1H)-ones von Hu, Essa H, Sidler, Daniel R, Dolling, Ulf-H

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The Expedient Synthesis of 4,2‘-Difluoro-5‘-(7-trifluoromethyl- imidazo[1,2-a]pyrimidin-3-yl)biphenyl-2-carbonitrile, a GABA α2/3 Agonist von Cameron, Mark, Foster, Bruce S, Lynch, Joseph E, Shi, Yao-Jun, Dolling, Ulf-H

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Practical Synthesis of Aryl Triflates under Aqueous Conditions von Frantz, Doug E, Weaver, Damian G, Carey, James P, Kress, Michael H, Dolling, Ulf H

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Development of a Phase Transfer Catalyzed Asymmetric Synthesis for an Estrogen Receptor Beta Selective Agonist von Scott, Jeremy P, Ashwood, Michael S, Brands, Karel M. J, Brewer, Sarah E, Cowden, Cameron J, Dolling, Ulf-H, Emerson, Khateeta M, Gibb, Andrew D, Goodyear, Adrian, Oliver, Steven F, Stewart, Gavin W, Wallace, Debra J

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Practical Asymmetric Synthesis of a γ-Secretase Inhibitor Exploiting Substrate-Controlled Intramolecular Nitrile Oxide−Olefin Cycloaddition von Scott, Jeremy P, Oliver, Steven F, Brands, Karel M. J, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Hands, David, Keen, Stephen P, Sheen, Faye J, Reamer, Robert A, Wilson, Robert D, Dolling, Ulf-H

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Synthesis of a NO-Releasing Prodrug of Rofecoxib von Engelhardt, F. Conrad, Shi, Yao-Jun, Cowden, Cameron J, Conlon, David A, Pipik, Brenda, Zhou, George, McNamara, James M, Dolling, Ulf-H

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A new general method for preparation of N-methoxy- N-methylamides. Application in direct conversion of an ester to a ketone von Williams, J.Michael, Jobson, Ronald B., Yasuda, Nobuyoshi, Marchesini, George, Dolling, Ulf-H., Grabowski, Edward J.J.

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Stereoselective Synthesis of a Potent Thrombin Inhibitor by a Novel P2−P3 Lactone Ring Opening von Nelson, Todd D, LeBlond, Carl R, Frantz, Doug E, Matty, Louis, Mitten, Jeffrey V, Weaver, Damian G, Moore, Jeffrey C, Kim, Jaehon M, Boyd, Russell, Kim, Pei-Yi, Gbewonyo, Kodzo, Brower, Mark, Sturr, Michael, McLaughlin, Kathleen, McMasters, Daniel R, Kress, Michael H, McNamara, James M, Dolling, Ulf H

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A Double Ring Closing Metathesis Reaction in the Rapid, Enantioselective Synthesis of NK-1 Receptor Antagonists von Wallace, Debra J, Goodman, Jonathan M, Kennedy, Derek J, Davies, Antony J, Cowden, Cameron J, Ashwood, Michael S, Cottrell, Ian F, Dolling, Ulf-H, Reider, Paul J

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A Practical Synthesis of a γ-Secretase Inhibitor von Scott, Jeremy P, Lieberman, David R, Beureux, Olivier M, Brands, Karel M. J, Davies, Antony J, Gibson, Andrew W, Hammond, Deborah C, McWilliams, Chris J, Stewart, Gavin W, Wilson, Robert D, Dolling, Ulf-H

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Practical and efficient synthesis of N-halo compounds von Zhong, Yong-Li, Zhou, Hua, Gauthier, Donald R., Lee, Jaemoon, Askin, David, Dolling, Ulf H., Volante, Ralph P.

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Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction von Zhao, Matthew M, McNamara, James M, Ho, Guo-Jie, Emerson, Khateeta M, Song, Zhiguo J, Tschaen, David M, Brands, Karel M. J, Dolling, Ulf-H, Grabowski, Edward J. J, Reider, Paul J, Cottrell, Ian F, Ashwood, Michael S, Bishop, Brian C

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Practical Synthesis of the New Carbapenem Antibiotic Ertapenem Sodium von Williams, J. Michael, Brands, Karel M. J, Skerlj, Renato T, Jobson, Ronald B, Marchesini, George, Conrad, Karen M, Pipik, Brenda, Savary, Kimberly A, Tsay, Fuh-Rong, Houghton, Peter G, Sidler, D. Richard, Dolling, Ulf-H, DiMichele, Lisa M, Novak, Thomas J

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Practical Asymmetric Synthesis of an Endothelin Receptor Antagonist von Song, Zhiguo J, Zhao, Mangzhu, Desmond, Richard, Devine, Paul, Tschaen, David M, Tillyer, Richard, Frey, Lisa, Heid, Richard, Xu, Feng, Foster, Bruce, Li, Jing, Reamer, Robert, Volante, Ralph, Dolling, Ulf H, Reider, Paul J, Okada, Shigemitsu, Kato, Yoshiaki, Mano, Eiichi

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Asymmetric Synthesis of MK-0499 von Tschaen, David M, Abramson, Lee, Cai, Dongwei, Desmond, Richard, Dolling, Ulf-H, Frey, Lisa, Karady, Sandor, Shi, Yao-Jun, Verhoeven, Thomas R

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Stereoselective double ring closing metathesis reactions in the synthesis of spirocyclic compounds von Wallace, Debra J, Cowden, Cameron J, Kennedy, Derek J, Ashwood, Michael S, Cottrell, Ian F, Dolling, Ulf-H

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Efficient One-Pot Synthesis of the 2-Aminocarbonylpyrrolidin-4-ylthio-Containing Side Chain of the New Broad-Spectrum Carbapenem Antibiotic Ertapenem von Brands, Karel M. J, Jobson, Ronald B, Conrad, Karen M, Williams, J. Michael, Pipik, Brenda, Cameron, Mark, Davies, Antony J, Houghton, Peter G, Ashwood, Michael S, Cottrell, Ian F, Reamer, Robert A, Kennedy, Derek J, Dolling, Ulf-H, Reider, Paul J

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A Novel Crystallization-Induced Diastereomeric Transformation Based on a Reversible Carbon−Sulfur Bond Formation. Application to the Synthesis of a γ-Secretase Inhibitor von Davies, Antony J, Scott, Jeremy P, Bishop, Brian C, Brands, Karel M. J, Brewer, Sarah E, DaSilva, Jimmy O, Dormer, Peter G, Dolling, Ulf-H, Gibb, Andrew D, Hammond, Deborah C, Lieberman, David R, Palucki, Michael, Payack, Joseph F

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Development of a Scaleable Synthesis of a Partial Nicotinic Acid Receptor Agonist von Wilson, Robert D, Cleator, Ed, Ashwood, Michael S, Bio, Matthew M, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf-H, Emerson, Khateeta M, Gibb, Andrew D, Hands, David, McKeown, Arlene E, Oliver, Steven F, Reamer, Robert A, Sheen, Faye J, Stewart, Gavin W, Zhou, George X

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Practical synthesis of a highly functionalized thiazole ketone von Frey, Lisa F, Marcantonio, Karen M, Chen, Cheng-yi, Wallace, Debra J, Murry, Jerry A, Tan, Lushi, Chen, Weirong, Dolling, Ulf H, Grabowski, Edward J.J

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