Total Synthesis and Antimalarial Activity of 2‑(p‑Hydroxybenzyl)-prodigiosins, Isoheptylprodigiosin, and Geometric Isomers of Tambjamine MYP1 Isolated from Marine Bacteria von Kancharla, Papireddy, Li, Yuexin, Yeluguri, Monish, Dodean, Rozalia A, Reynolds, Kevin A, Kelly, Jane X

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Boron trifluoride etherate promoted microwave-assisted synthesis of antimalarial acridones von Kancharla, Papireddy, Dodean, Rozalia A, Li, Yuexin, Kelly, Jane X

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Optimization of B‑Ring-Functionalized Antimalarial Tambjamines and Prodiginines von Kumar, Amrendra, Chithanna, Sivanna, Li, Yuexin, Zhang, Xiaowei, Dodean, Rozalia A., Caridha, Diana, Madejczyk, Michael S., Lee, Patricia J., Jin, Xiannu, Chetree, Ravi, Blount, Cameron, Dennis, William E., DeLuca, Jesse, Vuong, Chau, Pannone, Kristina, Dinh, Hieu T., Leed, Susan, Roth, Alison, Reynolds, Kevin A., Kelly, Jane X., Kancharla, Papireddy

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Babesia duncani as a Model Organism to Study the Development, Virulence, and Drug Susceptibility of Intraerythrocytic Parasites In Vitro and In Vivo von Pal, Anasuya C, Renard, Isaline, Singh, Pallavi, Vydyam, Pratap, Chiu, Joy E, Pou, Sovitj, Winter, Rolf W, Dodean, Rozalia, Frueh, Lisa, Nilsen, Aaron C, Riscoe, Michael K, Doggett, J Stone, Ben Mamoun, Choukri

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Long-acting intramuscular injections of ELQ-331, an antimalarial agent von Karunakaran, Dipu, Mutyam, Shravan K., Fu, Melody, Chen, Jiaming, Pham, Kim Hue Nicky, Pou, Sovitj, Winter, Rolf W., Nilsen, Aaron, Dodean, Rozalia A., Smilkstein, Martin J., Riscoe, Michael K., Shankar, Gita

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Discovery of dual function acridones as a new antimalarial chemotype von Hinrichs, David J, Wittlin, Sergio, Cooper, Roland A, Riscoe, Michael K, Dodean, Rozalia A, Kelly, Jane X, Winter, Rolf, Smilkstein, Martin J, Janowsky, Aaron, Lane, Kristin D, Johnson, Robert A, Brun, Reto

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Endochin-like quinolone-300 and ELQ-316 inhibit Babesia bovis, B. bigemina, B. caballi and Theileria equi von Silva, Marta G, Bastos, Reginaldo G, Stone Doggett, J, Riscoe, Michael K, Pou, Sovitj, Winter, Rolf, Dodean, Rozalia A, Nilsen, Aaron, Suarez, Carlos E

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Discovery and Optimization of Tambjamines as a Novel Class of Antileishmanial Agents von Kancharla, Papireddy, Ortiz, Diana, Fargo, Corinne M., Zhang, Xiaowei, Li, Yuexin, Sanchez, Marco, Kumar, Amrendra, Yeluguri, Monish, Dodean, Rozalia A., Caridha, Diana, Madejczyk, Michael S., Martin, Monica, Jin, Xiannu, Blount, Cameron, Chetree, Ravi, Pannone, Kristina, Dinh, Hieu T., DeLuca, Jesse, Evans, Martin, Nadeau, Robert, Vuong, Chau, Leed, Susan, Dennis, William E., Roncal, Norma, Pybus, Brandon S., Lee, Patricia J., Roth, Alison, Reynolds, Kevin A., Kelly, Jane X., Landfear, Scott M.

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New Scalable Synthetic Routes to ELQ-300, ELQ-316, and Other Antiparasitic Quinolones von Pou, Sovitj, Dodean, Rozalia A, Frueh, Lisa, Liebman, Katherine M, Gallagher, Rory T, Jin, Haihong, Jacobs, Robert T, Nilsen, Aaron, Stuart, David R, Doggett, J. Stone, Riscoe, Michael K, Winter, Rolf W

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ELQ-331 as a prototype for extremely durable chemoprotection against malaria von Smilkstein, Martin J, Pou, Sovitj, Krollenbrock, Alina, Bleyle, Lisa A, Dodean, Rozalia A, Frueh, Lisa, Hinrichs, David J, Li, Yuexin, Martinson, Thomas, Munar, Myrna Y, Winter, Rolf W, Bruzual, Igor, Whiteside, Samantha, Nilsen, Aaron, Koop, Dennis R, Kelly, Jane X, Kappe, Stefan H I, Wilder, Brandon K, Riscoe, Michael K

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Targeted Structure-Activity Analysis of Endochin-like Quinolones Reveals Potent Qi and Qo Site Inhibitors of Toxoplasma gondii and Plasmodium falciparum Cytochrome bc1 and Identifi... von McConnell, Erin V, Bruzual, Igor, Pou, Sovitj, Winter, Rolf, Dodean, Rozalia A, Smilkstein, Martin J, Krollenbrock, Alina, Nilsen, Aaron, Zakharov, Lev N, Riscoe, Michael K, Doggett, J Stone

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A New Scalable Synthesis of ELQ-300, ELQ-316, and other Antiparasitic Quinolones von Pou, Sovitj, Dodean, Rozalia A, Frueh, Lisa, Liebman, Katherine M, Gallagher, Rory T, Jin, Haihong, Jacobs, Robert T, Nilsen, Aaron, Stuart, David R, Doggett, J Stone, Riscoe, Michael K, Winter, Rolf W

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Lead Optimization of Second-Generation Acridones as Broad-Spectrum Antimalarials von Kancharla, Papireddy, Dodean, Rozalia A, Li, Yuexin, Pou, Sovitj, Pybus, Brandon, Melendez, Victor, Read, Lisa, Bane, Charles E, Vesely, Brian, Kreishman-Deitrick, Mara, Black, Chad, Li, Qigui, Sciotti, Richard J, Olmeda, Raul, Luong, Thu-Lan, Gaona, Heather, Potter, Brittney, Sousa, Jason, Marcsisin, Sean, Caridha, Diana, Xie, Lisa, Vuong, Chau, Zeng, Qiang, Zhang, Jing, Zhang, Ping, Lin, Hsiuling, Butler, Kirk, Roncal, Norma, Gaynor-Ohnstad, Lacy, Leed, Susan E, Nolan, Christina, Ceja, Frida G, Rasmussen, Stephanie A, Tumwebaze, Patrick K, Rosenthal, Philip J, Mu, Jianbing, Bayles, Brett R, Cooper, Roland A, Reynolds, Kevin A, Smilkstein, Martin J, Riscoe, Michael K, Kelly, Jane X

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Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials von Dodean, Rozalia A, Kancharla, Papireddy, Li, Yuexin, Melendez, Victor, Read, Lisa, Bane, Charles E, Vesely, Brian, Kreishman-Deitrick, Mara, Black, Chad, Li, Qigui, Sciotti, Richard J, Olmeda, Raul, Luong, Thu-Lan, Gaona, Heather, Potter, Brittney, Sousa, Jason, Marcsisin, Sean, Caridha, Diana, Xie, Lisa, Vuong, Chau, Zeng, Qiang, Zhang, Jing, Zhang, Ping, Lin, Hsiuling, Butler, Kirk, Roncal, Norma, Gaynor-Ohnstad, Lacy, Leed, Susan E, Nolan, Christina, Huezo, Stephanie J, Rasmussen, Stephanie A, Stephens, Melissa T, Tan, John C, Cooper, Roland A, Smilkstein, Martin J, Pou, Sovitj, Winter, Rolf W, Riscoe, Michael K, Kelly, Jane X

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3‑Position Biaryl Endochin-like Quinolones with Enhanced Antimalarial Performance von Pou, Sovitj, Winter, Rolf W., Dodean, Rozalia A., Liebman, Katherine, Li, Yuexin, Mather, Michael W., Nepal, Binod, Nilsen, Aaron, Handford, Mason J., Riscoe, Teresa M., Laxson, Sydney, Kirtley, Payton J., Aleshnick, Maya, Zakharov, Lev N., Kelly, Jane X., Smilkstein, Martin J., Wilder, Brandon K., Kortagere, Sandhya, Vaidya, Akhil B., Alday, P. Holland, Doggett, J. Stone, Riscoe, Michael K.

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Tambjamines as Fast-Acting Multistage Antimalarials von Kumar, Amrendra, Li, Yuexin, Dodean, Rozalia A., Roth, Alison, Caridha, Diana, Madejczyk, Michael S., Jin, Xiannu, Dennis, William E., Lee, Patricia J., Pybus, Brandon S., Martin, Monica, Pannone, Kristina, Dinh, Hieu T., Blount, Cameron, Chetree, Ravi, DeLuca, Jesse, Evans, Martin, Nadeau, Robert, Vuong, Chau, Leed, Susan, Black, Chad, Sousa, Jason, Nolan, Christina, Ceja, Frida G., Rasmussen, Stephanie A., Tumwebaze, Patrick K., Rosenthal, Philip J., Cooper, Roland A., Rottmann, Matthias, Orjuela-Sanchez, Pamela, Meister, Stephan, Winzeler, Elizabeth A., Delves, Michael J., Matthews, Holly, Baum, Jake, Kirby, Robert W., Burrows, Jeremy N., Duffy, James, Peyton, David H., Reynolds, Kevin A., Kelly, Jane X., Kancharla, Papireddy

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Acridones Are Highly Potent Inhibitors of Toxoplasma gondii Tachyzoites von Alday, P. Holland, McConnell, Erin V, Boitz Zarella, Jan M, Dodean, Rozalia A, Kancharla, Papireddy, Kelly, Jane X, Doggett, J. Stone

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Design, Synthesis, and Evaluation of 10-N-Substituted Acridones as Novel Chemosensitizers in Plasmodium falciparum von KELLY, Jane X, SMILKSTEIN, Martin J, COOPER, Roland A, LANE, Kristin D, JOHNSON, Robert A, JANOWSKY, Aaron, DODEAN, Rozalia A, HINRICHS, David J, WINTER, Rolf, RISCOE, Michael

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Diphenylether-Modified 1,2-Diamines with Improved Drug Properties for Development against Mycobacterium tuberculosis von Foss, Marie H, Pou, Sovitj, Davidson, Patrick M, Dunaj, Jennifer L, Winter, Rolf W, Pou, Sovijja, Licon, Meredith H, Doh, Julia K, Li, Yuexin, Kelly, Jane X, Dodean, Rozalia A, Koop, Dennis R, Riscoe, Michael K, Purdy, Georgiana E

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Targeted Structure–Activity Analysis of Endochin-like Quinolones Reveals Potent Qi and Qo Site Inhibitors of Toxoplasma gondii and Plasmodium falciparum Cytochrome bc 1 and Identif... von McConnell, Erin V, Bruzual, Igor, Pou, Sovitj, Winter, Rolf, Dodean, Rozalia A, Smilkstein, Martin J, Krollenbrock, Alina, Nilsen, Aaron, Zakharov, Lev N, Riscoe, Michael K, Doggett, J. Stone

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