Discovery of novel benzohydroxamate-based histone deacetylase 6 (HDAC6) inhibitors with the ability to potentiate anti-PD-L1 immunotherapy in melanoma von Peng, Xiaopeng, Yu, Ziwen, Surineni, Goverdhan, Deng, Bulian, Zhang, Meizhu, Li, Chuan, Sun, Zhiqiang, Pan, Wanyi, Liu, Yao, Liu, Shenglan, Yu, Bin, Chen, Jianjun

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Discovery of pomalidomide-based PROTACs for selective degradation of histone deacetylase 8 von Sun, Zhiqiang, Deng, Bulian, Yang, Zichao, Mai, Ruiyao, Huang, Junli, Ma, Zeli, Chen, Ting, Chen, Jianjun

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Design, Synthesis, and Bioevaluation of Novel Enzyme-Triggerable Cell Penetrating Peptide-Based Dendrimers for Targeted Delivery of Camptothecin and Cancer Therapy von Mai, Ruiyao, Deng, Bulian, Zhao, Huiting, Li, Ling, Fang, Yuyu, Li, Siming, Deng, Xin, Chen, Jianjun

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Discovery of Novel HDAC3 Inhibitors with PD-L1 Downregulating/Degrading and Antitumor Immune Effects von Sun, Zhiqiang, Xu, Chenglong, Cheng, Jinmei, Yang, Zichao, Liu, Ting, Deng, Bulian, Zhang, Xuewen, Peng, Xiaopeng, Chen, Jianjun

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Novel CRBN-Recruiting Proteolysis-Targeting Chimeras as Degraders of Stimulator of Interferon Genes with In Vivo Anti-Inflammatory Efficacy von Liu, Jin, Yuan, Lin, Ruan, Yong, Deng, Bulian, Yang, Zicao, Ren, Yichang, Li, Ling, Liu, Ting, Zhao, Huiting, Mai, Ruiyao, Chen, Jianjun

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Design, synthesis, and bioevaluation of imidazo [1,2–a] pyrazine derivatives as tubulin polymerization inhibitors with potent anticancer activities von Deng, Bulian, Sun, Zhiqiang, Wang, Yuxi, Mai, Ruiyao, Yang, Zichao, Ren, Yichang, Liu, Jin, Huang, Junli, Ma, Zeli, Chen, Ting, Zeng, Canjun, Chen, Jianjun

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Discovery of Thieno[2,3-d]pyrimidine-based KRAS G12D inhibitors as potential anticancer agents via combinatorial virtual screening von Li, Ling, Liu, Jin, Yang, Zichao, Zhao, Huiting, Deng, Bulian, Ren, Yichang, Mai, Ruiyao, Huang, Junli, Chen, Jianjun

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