Intermolecular Enolate Heterocoupling: Scope, Mechanism, and Application von DeMartino, Michael P, Chen, Ke, Baran, Phil S

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Model-Based Virtual PK/PD Exploration and Machine Learning Approach to Define PK Drivers in Early Drug Discovery von Chen, Emile P., Dutta, Shayoni, Ho, Ming-Hsun, DeMartino, Michael P.

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Applications of Model-Based Target Pharmacology Assessment in Defining Drug Design and DMPK Strategies: GSK Experiences von Chen, Emile P., Bondi, Robert W., Zhang, Carolyn, Price, Daniel J., Ho, Ming-Hsun, Armacost, Kira A., DeMartino, Michael P.

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Intermolecular Oxidative Enolate Heterocoupling von Baran, Phil S., DeMartino, Michael P.

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Exploring the Potential of RET Kinase Inhibition for Irritable Bowel Syndrome: A Preclinical Investigation in Rodent Models of Colonic Hypersensitivity von Russell, John P, Mohammadi, Ehsan, Ligon, Casey O, Johnson, Anthony C, Gershon, Michael D, Rao, Meenakshi, Shen, Yuhong, Chan, Chi-Chung, Eidam, Hilary S, DeMartino, Michael P, Cheung, Mui, Oliff, Allen I, Kumar, Sanjay, Greenwood-Van Meerveld, Beverley

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TLR2 agonism reverses chemotherapy-induced neutropenia in Macaca fascicularis von Laping, Nicholas J., DeMartino, Michael P., Cottom, Joshua E., Axten, Jeffrey M., Emery, John G., Guss, Jeffrey H., Burman, Miriam, Foley, James J., Cheung, Mui, Oliff, Allen, Kumar, Sanjay

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Understanding Pharmacokinetic Disconnect in Preclinical Species for 4-Aminoquinolines: Consequences of Low Permeability and High P-glycoprotein Efflux Ratio on Rat and Dog Oral Pha... von Mahajan, Mukesh K., Rivera, Elizabeth J., Sun, Helen H., Nagilla, Rakesh, DeMartino, Michael P., Haile, Pamela A., Casillas, Linda N., Marquis, Robert W., Votta, Bartholomew J., Bertin, John, Reilly, Michael A.

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Overcoming the Pregnane X Receptor Liability: Rational Design to Eliminate PXR-Mediated CYP Induction von Ramanjulu, Joshi M, Williams, Shawn P, Lakdawala, Ami S, DeMartino, Michael P, Lan, Yunfeng, Marquis, Robert W

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Enteric RET inhibition attenuates gastrointestinal secretion and motility via cholinergic signaling in rat colonic mucosal preparations von Russell, John P., Mohammadi, Ehsan, Ligon, Casey, Latorre, Rocco, Johnson, Anthony C., Hoang, Bao, Krull, David, Ho, Melisa W.‐Y., Eidam, Hilary S., DeMartino, Michael P., Cheung, Mui, Oliff, Allen I., Kumar, Sanjay, Greenwood‐Van Meerveld, Beverley

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Titanium(IV) Isopropoxide Mediated Synthesis of Pyrimidin-4-ones von Ramanjulu, Joshi M, DeMartino, Michael P, Lan, Yunfeng, Marquis, Robert

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Identification of Quinoline-Based RIP2 Kinase Inhibitors with an Improved Therapeutic Index to the hERG Ion Channel von Haile, Pamela A, Casillas, Linda N, Bury, Michael J, Mehlmann, John F, Singhaus, Robert, Charnley, Adam K, Hughes, Terry V, DeMartino, Michael P, Wang, Gren Z, Romano, Joseph J, Dong, Xiaoyang, Plotnikov, Nikolay V, Lakdawala, Ami S, Convery, Maire A, Votta, Bartholomew J, Lipshutz, David B, Desai, Biva M, Swift, Barbara, Capriotti, Carol A, Berger, Scott B, Mahajan, Mukesh K, Reilly, Michael A, Rivera, Elizabeth J, Sun, Helen H, Nagilla, Rakesh, LePage, Carol, Ouellette, Michael T, Totoritis, Rachel D, Donovan, Brian T, Brown, Barry S, Chaudhary, Khuram W, Gough, Peter J, Bertin, John, Marquis, Robert W

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Identification of a Ret Kinase Inhibitor, GSK589, as a Peripheral Analgesic for the Treatment Visceral Pain Associated with Irritable Bowel Syndrome von Russell, John, Mohammadi, Ehsan, Ligon, Casey O, Latorre, Rocco, Joberty, Gerard, Zinn, Nico, Castellino, Steve, Hoang, Bao, Krull, David L, DeMartino, Michael P, Cheung, Mui, Oliff, Allen, Meerveld, Beverley Greenwood-Van, Kumar, Sanjay

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RIP3 Induces Apoptosis Independent of Pronecrotic Kinase Activity von Mandal, Pratyusha, Berger, Scott B., Pillay, Sirika, Moriwaki, Kenta, Huang, Chunzi, Guo, Hongyan, Lich, John D., Finger, Joshua, Kasparcova, Viera, Votta, Bart, Ouellette, Michael, King, Bryan W., Wisnoski, David, Lakdawala, Ami S., DeMartino, Michael P., Casillas, Linda N., Haile, Pamela A., Sehon, Clark A., Marquis, Robert W., Upton, Jason, Daley-Bauer, Lisa P., Roback, Linda, Ramia, Nancy, Dovey, Cole M., Carette, Jan E., Chan, Francis Ka-Ming, Bertin, John, Gough, Peter J., Mocarski, Edward S., Kaiser, William J.

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Mo1602 - Identification of a Ret Kinase Inhibitor, GSK589, as a Peripheral Analgesic for the Treatment Visceral Pain Associated with Irritable Bowel Syndrome von Russell, John, Mohammadi, Ehsan, Ligon, Casey O., Latorre, Rocco, Joberty, Gerard, Zinn, Nico, Castellino, Steve, Hoang, Bao, Krull, David L., DeMartino, Michael P., Cheung, Mui, Oliff, Allen, Meerveld, Beverley Greenwood-Van, Kumar, Sanjay

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Identification of Quinoline-Based RIP2 Kinase Inhibitors with an Improved Therapeutic Index to the hERG Ion Channel (vol 9, pg 1039, 2018) von Haile, Pamela A., Casillas, Linda N., Bury, Michael J., Mehlmann, John F., Singhaus, Robert, Charnley, Adam K., Hughes, Terry V., DeMartino, Michael P., Wang, Gren Z., Romano, Joseph J., Dong, Xiaoyang, Plotnikov, Nikolay V., Lakdawala, Ami S., Duraiswami, Chaya, Convery, Maire A., Votta, Bartholomew J., Lipshutz, David B., Desai, Biva M., Swift, Barbara, Capriotti, Carol A., Berger, Scott B., Mahajan, Mukesh K., Reilly, Michael A., Rivera, Elizabeth J., Sun, Helen H., Nagilla, Rakesh, LePage, Carol, Ouellette, Michael T., Totoritis, Rachel D., Donovan, Brian T., Brown, Barry S., Chaudhary, Khuram W., Gough, Peter J., Bertin, John, Marquis, Robert W.

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Correction to Identification of Quinoline-Based RIP2 Kinase Inhibitors with an Improved Therapeutic Index to the hERG Ion Channel von Haile, Pamela A., Casillas, Linda N., Bury, Michael J., Mehlmann, John F., Singhaus, Robert, Charnley, Adam K., Hughes, Terry V., DeMartino, Michael P., Wang, Gren Z., Romano, Joseph J., Dong, Xiaoyang, Plotnikov, Nikolay V., Lakdawala, Ami S., Duraiswami, Chaya, Convery, Maire A., Votta, Bartholomew J., Lipshutz, David B., Desai, Biva M., Swift, Barbara, Capriotti, Carol A., Berger, Scott B., Mahajan, Mukesh K., Reilly, Michael A., Rivera, Elizabeth J., Sun, Helen H., Nagilla, Rakesh, LePage, Carol, Ouellette, Michael T., Totoritis, Rachel D., Donovan, Brian T., Brown, Barry S., Chaudhary, Khuram W., Gough, Peter J., Bertin, John, Marquis, Robert W.

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RIP3 induces apoptosis independent of pro-necrotic kinase activity von Mandal, Pratyusha, Berger, Scott B., Pillay, Sirika, Moriwaki, Kenta, Huang, Chunzi, Guo, Hongyan, Lich, John D., Finger, Joshua, Kasparcova, Viera, Votta, Bart, Ouellette, Michael, King, Bryan W., Wisnoski, David, Lakdawala, Ami S., DeMartino, Michael P., Casillas, Linda N., Haile, Pamela A., Sehon, Clark A., Marquis, Robert W., Upton, Jason, Daley-Bauer, Lisa P., Roback, Linda, Ramia, Nancy, Dovey, Cole M., Carette, Jan E., Chan, Francis, Bertin, John, Gough, Peter J., Mocarski, Edward S., Kaiser, William J.

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Intra- vs. intermolecular configurations in the three-legged, piano-stool compounds ( o, m and p-xylene)Mo(CO) 3 von DeMartino, Michael P., Read, Stephen M., Rheingold, Arnold L.

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N-(3-(2-(4-CHLOROPHENOXY)ACETAMIDO)BICYCLO[1.1.1] PENTAN-1-YL)-2-CYCLOBUTANE-1- CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS ATF4 INHIBITORS FOR TREATING CANCER AND OTHER DISEA... von KALITA, Biswajit, CHEUNG, Mui, DEMARTINO, Michael P

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Piridinonas como inhibidores reordenados durante la transfección (RET) von GUAN, Huiping Amy, DEMARTINO, Michael P

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