Intrathecal pertussis toxin produces hyperalgesia and allodynia in mice von Womer, Daniel E, DeLapp, Neil W, E. Shannon, Harlan

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The Minimum Significant Ratio: A Statistical Parameter to Characterize the Reproducibility of Potency Estimates from Concentration-Response Assays and Estimation by Replicate-Exper... von Eastwood, Brian J., Farmen, Mark W., Iversen, Philip W., Craft, Trelia J., Smallwood, Jeffrey K., Garbison, Kim E., Delapp, Neil W., Smith, Gerald F.

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Muscarinic receptor agonists decrease cocaine self-administration rates in drug-naive mice von Rasmussen, Thøger, Sauerberg, Per, Nielsen, Erik B, Swedberg, Michael D.B, Thomsen, Christian, Sheardown, Malcolm J, Jeppesen, Lone, Calligaro, David O, DeLapp, Neil W, Whitesitt, Celia, Ward, John S, Shannon, Harlan E, Bymaster, Frank P, Fink-Jensen, Anders

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Unexpected antipsychotic-like activity with the muscarinic receptor ligand (5 R,6 R)6-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane von Bymaster, Frank P, Shannon, Harlan E, Rasmussen, Kurt, Delapp, Neil W, Mitch, Charles H, Ward, John S, Calligaro, David O, Ludvigsen, Thomas S, Sheardown, Malcolm J, Olesen, Preben H, Swedberg, Michael D.B, Sauerberg, Per, Fink-Jensen, Anders

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M1 muscarinic receptor signaling in mouse hippocampus and cortex von Porter, Amy C, Bymaster, Frank P, DeLapp, Neil W, Yamada, Masahisa, Wess, Jürgen, Hamilton, Susan E, Nathanson, Neil M, Felder, Christian C

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Muscarinic Agonists with Antipsychotic-like Activity:  Structure−Activity Relationships of 1,2,5-Thiadiazole Analogues with Functional Dopamine Antagonist Activity von Sauerberg, Per, Jeppesen, Lone, Olesen, Preben H, Rasmussen, Thøger, Swedberg, Michael D. B, Sheardown, Malcolm J, Fink-Jensen, Anders, Thomsen, Christian, Thøgersen, Henning, Rimvall, Karin, Ward, John S, Calligaro, David O, DeLapp, Neil W, Bymaster, Frank P, Shannon, Harlan E

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Muscarinic agonists exhibit functional dopamine antagonism in unilaterally 6-OHDA lesioned rats von Fink-Jensen, Anders, Kristensen, Peter, Shannon, Harlan E, Calligaro, David O, Delapp, Neil W, Whitesitt, Cilia, Ward, John S, Thomsen, Christian, Rasmusseen, Thøger, Sheardown, Malcolm J, Jeppesen, Lone, Sauerberg, Per, Bymaster, Frank P

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Forskolin Stimulation of Cyclic AMP Accumulation in Rat Brain Cortex Slices Is Markedly Enhanced by Endogenous Adenosine von DeLapp, Neil W., Eckols, Kris

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Identification of side chains on 1,2,5-thiadiazole-azacycles optimal for muscarinic M1 receptor activation von Sauerberg, Per, Jeppesen, Lone, Olesen, Preben H, Sheardown, Malcolm J, Fink-Jensen, Anders, Rasmussen, Thøger, Rimvall, Karin, Shannon, Harlan E, Bymaster, Frank P, DeLapp, Neil W, Calligaro, Dave O, Ward, John S, Whitesitt, Celia A, Thomsen, Christian

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The muscarinic receptor agonist BuTAC, a novel potential antipsychotic, does not impair learning and memory in mouse passive avoidance von Rasmussen, Thøger, Fink-Jensen, Anders, Sauerberg, Per, Swedberg, Michael D.B., Thomsen, Christian, Sheardown, Malcolm J., Jeppesen, Lone, Calligaro, David O., DeLapp, Neil W., Whitesitt, Celia, Ward, John S., Shannon, Harlan E., Bymaster, Frank P.

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Potential role of muscarinic receptors in schizophrenia von Bymaster, Frank P., Shannon, Harlan E., Rasmussen, Kurt, DeLapp, Neil W., Ward, John S., Calligaro, David O., Mitch, Charles H., Whitesitt, Celia, Ludvigsen, Thomas S., Sheardown, Malcolm, Swedberg, Michael, Rasmussen, Thøger, Olesen, Preben H., Jeppesen, Lone, Sauerberg, Per, Fink-Jensen, Anders

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Receptor reserve of phosphoinositide-coupled muscarinic receptors in mouse hippocampus in vivo von Bymaster, Frank P, Carter, Petra A, DeLapp, Neil W, Calligaro, David O, Felder, Christian C

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1-(1,2,5-Thiadiazol-4-yl)-4-azatricyclo[2.2.1.02,6]heptanes as New Potent Muscarinic M1 Agonists:  Structure−Activity Relationship for 3-Aryl-2-propyn-1-yloxy and 3-Aryl-2-propyn-1... von Jeppesen, Lone, Olesen, Preben H, Hansen, Lena, Sheardown, Malcolm J, Thomsen, Christian, Rasmussen, Thøger, Jensen, Anders Fink, Christensen, Michael S, Rimvall, Karin, Ward, John S, Whitesitt, Celia, Calligaro, David O, Bymaster, Frank P, Delapp, Neil W, Felder, Christian C, Shannon, Harlan E, Sauerberg, Per

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The antibody-capture [ 35S]GTPγS scintillation proximity assay: a powerful emerging technique for analysis of GPCR pharmacology von DeLapp, Neil W.

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Antagonism by olanzapine of dopamine D1, serotonin2, muscarinic, histamine H1 and α1-adrenergic receptors in vitro von BYMASTER, F. P, NELSON, D. L, DELAPP, N. W, FALCONE, J. F, ECKOLS, K, TRUEX, L. L, FOREMAN, M. M, LUCAITES, V. L, CALLIGARO, D. O

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The muscarinic M1 agonist xanomeline increases soluble amyloid precursor protein release from chinese hamster ovary-m1 cells von Eckols, Kris, Bymaster, Frank P., Mitch, Charles H., Shannon, Harlan E., Ward, John S., DeLapp, Neil W.

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Effect of Basic Fibroblast Growth Factor (bFGF) and Insulin-Like Growth Factors Type I (IGF-I) and Type II (IGF-II) on Adult Human Keratinocyte Growth and Fibronectin Secretion von DeLapp, Neil W., Dieckman, Donna K.

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Conformationally Constrained Analogues of the Muscarinic Agonist 3-(4-(Methylthio)-1,2,5-thiadiazol-3-yl)-1,2,5,6-tetrahydro-1-methylpyridine. Synthesis, Receptor Affinity, and Ant... von Sauerberg, Per, Olesen, Preben H, Sheardown, Malcolm J, Rimvall, Karin, Thøgersen, Henning, Shannon, Harlan E, Sawyer, Barry D, Ward, John S, Bymaster, Frank P, DeLapp, Neil W, Calligaro, David O, Swedberg, Michael D. B

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Potent antagonism of 5-HT3 and 5-HT6 receptors by olanzapine von BYMASTER, Frank P, FALCONE, Julie F, BAUZON, Delbert, KENNEDY, John S, SCHENCK, Kathryn, DELAPP, Neil W, COHEN, Marlene L

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Muscarinic agonist inhibition of rat striatal adenylate cyclase is enhanced by dopamine stimulation von Delapp, Neil W., Eckols, Kris, Shannon, Harlan E.

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