Discovery of MK-8153, a Potent and Selective ROMK Inhibitor and Novel Diuretic/Natriuretic von Jiang, Jinlong, Ding, Fa-Xiang, Zhou, Xiaoyan, Bateman, Thomas J, Dong, Shuzhi, Gu, Xin, Keh deJesus, Reynalda, Pio, Barbara, Tang, Haifeng, Chobanian, Harry R, Levorse, Dorothy, Hu, Mengwei, Thomas-Fowlkes, Brande, Margulis, Michael, Koehler, Martin, Weinglass, Adam, Gibson, Jack, Houle, Kevin, Yudkovitz, Joel, Hampton, Caryn, Pai, Lee-Yuh, Samuel, Koppara, Cutarelli, Timothy, Sullivan, Kathleen, Parmee, Emma R, Davies, Ian, Pasternak, Alexander

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Discovery and optimization of novel 4-[(aminocarbonyl)amino]- N-[4-(2-aminoethyl)phenyl]benzenesulfonamide ghrelin receptor antagonists von Pasternak, Alexander, Goble, Stephen D., deJesus, Reynalda K., Hreniuk, Donna L., Chung, Christine C., Tota, Michael R., Mazur, Paul, Feighner, Scott D., Howard, Andrew D., Mills, Sander G., Yang, Lihu

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Structure Guided Discovery of Novel Pan Metallo-β-Lactamase Inhibitors with Improved Gram-Negative Bacterial Cell Penetration von Dong, Shuzhi, Zhao, Zhiqiang, Tang, Haiqun, Li, Guoqing, Pan, Jianping, Gu, Xin, Jiang, Jinlong, Xiao, Li, Scapin, Giovanna, Hunter, David N., Yang, Dexi, Huang, Yuhua, Bennett, Frank, Yang, Shu-Wei, Mandal, Mihirbaran, Tang, Haifeng, Su, Jing, Tudge, Clare, deJesus, Reynalda Keh, Ding, Fa-Xiang, Lombardo, Matthew, Hicks, Jacqueline D., Fischmann, Thierry, Mirza, Asra, Dayananth, Priya, Painter, Ronald E., Villafania, Artjohn, Garlisi, Charles G., Zhang, Rumin, Mayhood, Todd W., Si, Qian, Li, Nianyu, Amin, Rupesh P., Bhatt, Bhavana, Chen, Feifei, Regan, Christopher P., Regan, Hillary, Lin, Xinjie, Wu, Jin, Leithead, Andrew, Pollack, Scott R., Scott, Jack D., Nargund, Ravi P., Therien, Alex G., Black, Todd, Young, Katherine, Pasternak, Alexander

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Quantitation of wall teichoic acid in Staphylococcus aureus by direct measurement of monomeric units using LC-MS/MS von Berejnaia, Olga, Wang, Hao, Labroli, Marc, Yang, Christine, Gill, Charles, Xiao, Jianying, Hesk, David, DeJesus, Reynalda, Su, Jing, Tan, Christopher M., Sheth, Payal R., Kavana, Michael, McLaren, David G.

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Can We Make Small Molecules Lean? Optimization of a Highly Lipophilic TarO Inhibitor von Mandal, Mihirbaran, Tan, Zheng, Madsen-Duggan, Christina, Buevich, Alexei V, Caldwell, John P, Dejesus, Reynalda, Flattery, Amy, Garlisi, Charles G, Gill, Charles, Ha, Sookhee Nicole, Ho, Ginny, Koseoglu, Sandra, Labroli, Marc, Basu, Kallol, Lee, Sang Ho, Liang, Lianzhu, Liu, Jenny, Mayhood, Todd, McGuinness, Debra, McLaren, David G, Wen, Xiujuan, Parmee, Emma, Rindgen, Diane, Roemer, Terry, Sheth, Payal, Tawa, Paul, Tata, James, Yang, Christine, Yang, Shu-Wei, Xiao, Li, Wang, Hao, Tan, Christopher, Tang, Haifeng, Walsh, Paul, Walsh, Erika, Wu, Jin, Su, Jing

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The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes von He, Shuwen, Ye, Zhixiong, Truong, Quang, Shah, Shrenik, Du, Wu, Guo, Liangqin, Dobbelaar, Peter H, Lai, Zhong, Liu, Jian, Jian, Tianying, Qi, Hongbo, Bakshi, Raman K, Hong, Qingmei, Dellureficio, James, Pasternak, Alexander, Feng, Zhe, deJesus, Reynalda, Yang, Lihu, Reibarkh, Mikhail, Bradley, Scott A, Holmes, Mark A, Ball, Richard G, Ruck, Rebecca T, Huffman, Mark A, Wong, Frederick, Samuel, Koppara, Reddy, Vijay B, Mitelman, Stan, Tong, Sharon X, Chicchi, Gary G, Tsao, Kwei-Lan, Trusca, Dorina, Wu, Margaret, Shao, Qing, Trujillo, Maria E, Eiermann, George J, Li, Cai, Zhang, Bei B, Howard, Andrew D, Zhou, Yun-Ping, Nargund, Ravi P, Hagmann, William K

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Diaminoindanes as Microsomal Triglyceride Transfer Protein Inhibitors von Ksander, Gary M, deJesus, Reynalda, Yuan, Andrew, Fink, Cynthia, Moskal, Michael, Carlson, Eric, Kukkola, Paivi, Bilci, Natalie, Wallace, Eli, Neubert, Alan, Feldman, David, Mogelesky, Therese, Poirier, Kevin, Jeune, Michael, Steele, Ronald, Wasvery, Jong, Stephan, Zouhair, Cahill, Edna, Webb, Randy, Navarrete, Aida, Lee, Warren, Gibson, Joyce, Alexander, Natalya, Sharif, Haamid, Hospattankar, Ashok

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BICYCLIC ARYL MONOBACTAM COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF BACTERIAL INFECTIONS von HUANG, Xianhai, DING, Fa-Xiang, JIAN, Jinlong, TANG, Haifeng, DEJESUS, Reynalda, Keh, LIU, Weiguo, SUN, Wanying, WANG, Hongwu, GUO, Yan

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Inhibitors of the renal outer medullary potassium channel von Jiang, Jinlong, Fu, Qinghong, deJesus, Reynalda K, Tang, Haifeng

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POLYCYCLIC CAP-DEPENDENT ENDONUCLEASE INHIBITORS FOR TREATING OR PREVENTING INFLUENZA von MCCAULEY, John A, GUO, Liangqin, CHOBANIAN, Harry R, DEJESUS, Reynalda Keh, PLOTKIN, Michael A, FELLS, James, SU, Hua, DE LERA RUIZ, Manuel, ZHAO, Kake, CROWLEY, Brendan M, ZHANG, Yonglian, LO, Michael Man-Chu, EMBREY, Mark, W, SHURTLEFF, Valerie W, KIM, Ronald M, BENNETT, Frank, MORRIELLO, Gregori, J

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Dicarboxylic Acid Dipeptide Neutral Endopeptidase Inhibitors von Ksander, Gary M, Ghai, Raj D, deJesus, Reynalda, Diefenbacher, Clive, Yuan, Andrew, Berry, Carol, Sakane, Yumi, Trapani, Angelo

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POLYCYCLIC CAP-DEPENDENT ENDONUCLEASE INHIBITORS FOR TREATING OR PREVENTING INFLUENZA von Fells, James, Bennett, Frank, Plotkin, Michael, Embrey, Mark W, Crowley, Brendan M, Zhao, Kake, Guo, Liangqin, DeJesus, Reynalda Keh, de Lera Ruiz, Manuel, Chobanian, Harry R, Morriello, Gregori J, Lo, Michael Man-Chu, Kim, Ronald M, McCauley, John A, Su, Hua, Shurtleff, Valerie W, Zhang, Yonglian

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Bicyclic aryl monobactam compounds and methods of use thereof for the treatment of bacterial infections von Dejesus, Reynalda Keh, Wang, Hongwu, Ding, Fa-Xiang, Huang, Xianhai, Liu, Weiguo, Guo, Yan, Jian, Jinlong, Sun, Wanying, Tang, Haifeng

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INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL von Jiang Jinlong, deJesus Reynalda K, Tang Haifeng, Fu Qinghong

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INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL von JIANG, Jinlong, TANG, Haifeng, FU, Qinghong, DEJESUS, Reynalda, K

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POLYCYCLIC CAP-DEPENDENT ENDONUCLEASE INHIBITORS FOR TREATING OR PREVENTING INFLUENZA von MCCAULEY, John A, GUO, Liangqin, CHOBANIAN, Harry R, DEJESUS, Reynalda Keh, PLOTKIN, Michael A, FELLS, James, SU, Hua, DE LERA RUIZ, Manuel, ZHAO, Kake, CROWLEY, Brendan M, ZHANG, Yonglian, LO, Michael Man-Chu, EMBREY, Mark, W, SHURTLEFF, Valerie W, KIM, Ronald M, BENNETT, Frank, MORRIELLO, Gregori, J

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Polycyclic cap-dependent endonuclease inhibitors for treating or preventing influenza von MCCAULEY, John A, GUO, Liangqin, CHOBANIAN, Harry R, DEJESUS, Reynalda Keh, PLOTKIN, Michael A, FELLS, James, SU, Hua, DE LERA RUIZ, Manuel, ZHAO, Kake, CROWLEY, Brendan M, ZHANG, Yonglian, MORRIELLO, Gregori J, LO, Michael Man-Chu, SHURTLEFF, Valerie W, KIM, Ronald M, EMBREY, Mark W, BENNETT, Frank

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Polycyclic cap-dependent endonuclease inhibitors for treating or preventing influenza von MCCAULEY, John A, GUO, Liangqin, CHOBANIAN, Harry R, DEJESUS, Reynalda Keh, PLOTKIN, Michael A, FELLS, James, SU, Hua, DE LERA RUIZ, Manuel, ZHAO, Kake, CROWLEY, Brendan M, ZHANG, Yonglian, MORRIELLO, Gregori J, LO, Michael Man-Chu, SHURTLEFF, Valerie W, KIM, Ronald M, EMBREY, Mark W, BENNETT, Frank

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Bicyclic aryl monobactam compounds and methods of use thereof for the treatment of bacterial infections von Dejesus, Reynalda Keh, Jiang, Jinlong, Wang, Hongwu, Ding, Fa-Xiang, Huang, Xianhai, Liu, Weiguo, Guo, Yan, Sun, Wanying, Tang, Haifeng

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BICYCLIC ARYL MONOBACTAM COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF BACTERIAL INFECTIONS von HUANG, Xianhai, DING, Fa-Xiang, JIAN, Jinlong, TANG, Haifeng, DEJESUS, Reynalda, Keh, LIU, Weiguo, SUN, Wanying, WANG, Hongwu, GUO, Yan

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