Conformationally constrained opioid ligands: The Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffold von Ballet, Steven, Feytens, Debby, Wachter, Rien De, Vlaeminck, Magali De, Marczak, Ewa D., Salvadori, Severo, Graaf, Chris de, Rognan, Didier, Negri, Lucia, Lattanzi, Roberta, Lazarus, Lawrence H., Tourwé, Dirk, Balboni, Gianfranco

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Asymmetric Synthesis and Conformational Analysis by NMR Spectroscopy and MD of Aba- and α-MeAba-Containing Dermorphin Analogues von Vandormael, Bart, De Wachter, Rien, Martins, José C., Hendrickx, Pieter M. S., Keresztes, Attila, Ballet, Steven, Mallareddy, Jayapal R., Tóth, Fanni, Tóth, Géza, Tourwé, Dirk

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Synthesis, Biological Evaluation, and Automated Docking of Constrained Analogues of the Opioid Peptide H-Dmt- d -Ala-Phe-Gly-NH 2 Using the 4- or 5-Methyl Substituted 4-Amino-1,2,4... von De Wachter, Rien, de Graaf, Chris, Keresztes, Atilla, Vandormael, Bart, Ballet, Steven, Tóth, Géza, Rognan, Didier, Tourwé, Dirk

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Synthesis, Biological Evaluation, and Automated Docking of Constrained Analogues of the Opioid Peptide H-Dmt-d-Ala-Phe-Gly-NH2 Using the 4- or 5-Methyl Substituted 4-Amino-1,2,4,5-... von De Wachter, Rien, de Graaf, Chris, Keresztes, Atilla, Vandormael, Bart, Ballet, Steven, Tóth, Géza, Rognan, Didier, Tourwé, Dirk

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Influence of ring substitution on the conformation and β-turn mimicry of 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one peptide mimetics von De Wachter, Rien, Brans, Luc, Ballet, Steven, Van den Eynde, Isabelle, Feytens, Debby, Keresztes, Attila, Toth, Geza, Urbanczyk-Lipkowska, Zofia, Tourwé, Dirk

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Synthesis of 4-amino-3-oxo-tetrahydroazepino[3,4- b]indoles: new conformationally constrained Trp analogs von Pulka, Karolina, Feytens, Debby, Van den Eynde, Isabelle, De Wachter, Rien, Kosson, Piotr, Misicka, Aleksandra, Lipkowski, Andrzej, Chung, Nga N., Schiller, Peter W., Tourwé, Dirk

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Synthesis and Evaluation of the β-Turn Properties of 4-Amino-1,2,4,5-tetrahydro-2-benzazepin-3-ones and of Their Spirocyclic Derivative von Van Rompaey, Karolien, Ballet, Steven, Tömböly, Csaba, De Wachter, Rien, Vanommeslaeghe, Kenno, Biesemans, Monique, Willem, Rudolph, Tourwé, Dirk

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Derivatization of 1-phenyl substituted 4-amino-2-benzazepin-3-ones: evaluation of Pd-catalyzed coupling reactions von Ballet, Steven, De Wachter, Rien, Maes, Bert U.W., Tourwé, Dirk

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Conformationally constrained opioid ligands: The Dmt-Aba and Dmt-Aia vs. Dmt-Tic scaffold von Ballet, Steven, Feytens, Debby, De Wachter, Rien, De Vlaeminck, Magali, Marczak, Ewa D., Salvadori, Severo, de Graaf, Chris, Rognan, Didier, Negri, Lucia, Lattanzi, Roberta, Lazarus, Lawrence H., Tourwé, Dirk, Balboni, Gianfranco

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High-performance liquid chromatographic separation of stereoisomers of N-phthaloyl-protected amino acids and dipeptidomimetics von Ilisz, István, Ballet, Steven, Van Rompaey, Karolien, De Wachter, Rien, Tourwé, Dirk, Armstrong, Daniel W., Péter, Antal

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