Molecular basis for cooperative binding and synergy of ATP-site and allosteric EGFR inhibitors von Beyett, Tyler S., To, Ciric, Heppner, David E., Rana, Jaimin K., Schmoker, Anna M., Jang, Jaebong, De Clercq, Dries J. H., Gomez, Gabriel, Scott, David A., Gray, Nathanael S., Jänne, Pasi A., Eck, Michael J.

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Discovery of a Highly Potent and Broadly Effective Epidermal Growth Factor Receptor and HER2 Exon 20 Insertion Mutant Inhibitor von Jang, Jaebong, Son, Jieun, Park, Eunyoung, Kosaka, Takayuki, Saxon, Jamie A., De Clercq, Dries J. H., Choi, Hwan Geun, Tanizaki, Junko, Eck, Michael J., Jänne, Pasi A., Gray, Nathanael S.

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Mutant‐Selective Allosteric EGFR Degraders are Effective Against a Broad Range of Drug‐Resistant Mutations von Jang, Jaebong, To, Ciric, De Clercq, Dries J. H., Park, Eunyoung, Ponthier, Charles M., Shin, Bo Hee, Mushajiang, Mierzhati, Nowak, Radosław P., Fischer, Eric S., Eck, Michael J., Jänne, Pasi A., Gray, Nathanael S.

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Discovery and Optimization of Dibenzodiazepinones as Allosteric Mutant-Selective EGFR Inhibitors von De Clercq, Dries J. H, Heppner, David E, To, Ciric, Jang, Jaebong, Park, Eunyoung, Yun, Cai-Hong, Mushajiang, Mierzhati, Shin, Bo Hee, Gero, Thomas W, Scott, David A, Jänne, Pasi A, Eck, Michael J, Gray, Nathanael S

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Single and Dual Targeting of Mutant EGFR with an Allosteric Inhibitor von To, Ciric, Jang, Jaebong, Chen, Ting, Park, Eunyoung, Mushajiang, Mierzhati, De Clercq, Dries J H, Xu, Man, Wang, Stephen, Cameron, Michael D, Heppner, David E, Shin, Bo Hee, Gero, Thomas W, Yang, Annan, Dahlberg, Suzanne E, Wong, Kwok-Kin, Eck, Michael J, Gray, Nathanael S, Jänne, Pasi A

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Proteome-scale Binary Interactomics in Human Cells von Lievens, Sam, Van der Heyden, José, Masschaele, Delphine, De Ceuninck, Leentje, Petta, Ioanna, Gupta, Surya, De Puysseleyr, Veronic, Vauthier, Virginie, Lemmens, Irma, De Clercq, Dries J.H., Defever, Dieter, Vanderroost, Nele, De Smet, Anne-Sophie, Eyckerman, Sven, Van Calenbergh, Serge, Martens, Lennart, De Bosscher, Karolien, Libert, Claude, Hill, David E., Vidal, Marc, Tavernier, Jan

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Chemical Dimerizers in Three-Hybrid Systems for Small Molecule–Target Protein Profiling von De Clercq, Dries J. H, Tavernier, Jan, Lievens, Sam, Van Calenbergh, Serge

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Kinase Substrate Sensor (KISS), a Mammalian In Situ Protein Interaction Sensor von Lievens, Sam, Gerlo, Sarah, Lemmens, Irma, De Clercq, Dries J.H., Risseeuw, Martijn D.P., Vanderroost, Nele, De Smet, Anne-Sophie, Ruyssinck, Elien, Chevet, Eric, Van Calenbergh, Serge, Tavernier, Jan

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A "Clickable" MTX Reagent as a Practical Tool for Profiling Small-Molecule-Intracellular Target Interactions via MASPIT von Risseeuw, Martijn D. P., De Clercq, Dries J. H., Lievens, Sam, Hillaert, Ulrik, Sinnaeve, Davy, Van den Broeck, Freya, Martins, José C., Tavernier, Jan, Van Calenbergh, Serge

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Alternative Reagents for Methotrexate as Immobilizing Anchor Moieties in the Optimization of MASPIT: Synthesis and Biological Evaluation von De Clercq, Dries J. H., Risseeuw, Martijn D. P., Karalic, Izet, De Smet, Anne-Sophie, Defever, Dieter, Tavernier, Jan, Lievens, Sam, Van Calenbergh, Serge

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Mutant‐Selective Allosteric EGFR Degraders are Effective Against a Broad Range of Drug‐Resistant Mutations von Jang, Jaebong, To, Ciric, De Clercq, Dries J. H., Park, Eunyoung, Ponthier, Charles M., Shin, Bo Hee, Mushajiang, Mierzhati, Nowak, Radosław P., Fischer, Eric S., Eck, Michael J., Jänne, Pasi A., Gray, Nathanael S.

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Discovery of a Highly Potent and Broadly Effective Epidermal Growth Factor Receptor and HER2 Exon 20 Insertion Mutant Inhibitor von Jang, Jaebong, Son, Jieun, Park, Eunyoung, Kosaka, Takayuki, Saxon, Jamie A., De Clercq, Dries J. H., Choi, Hwan Geun, Tanizaki, Junko, Eck, Michael J., Jänne, Pasi A., Gray, Nathanael S.

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