Crystallization-Induced Diastereomer Transformations von Brands, Karel M. J, Davies, Antony J

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A Novel Approach to 3-Methylindoles by a Heck/Cyclization/Isomerization Process von Baxter, Carl A, Cleator, Ed, Alam, Mahbub, Davies, Antony J, Goodyear, Adrian, O’Hagan, Michael

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Process Development and Multikilogram-Scale Synthesis of a TRPV1 Antagonist von Cleator, Ed, Scott, Jeremy P, Avalle, Paulo, Bio, Matthew M, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Sheen, Faye J, Stewart, Gavin W, Wallace, Debra J, Wilson, Robert D

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Efficient One-Pot Synthesis of the 2-Aminocarbonylpyrrolidin-4-ylthio-Containing Side Chain of the New Broad-Spectrum Carbapenem Antibiotic Ertapenem von Brands, Karel M. J, Jobson, Ronald B, Conrad, Karen M, Williams, J. Michael, Pipik, Brenda, Cameron, Mark, Davies, Antony J, Houghton, Peter G, Ashwood, Michael S, Cottrell, Ian F, Reamer, Robert A, Kennedy, Derek J, Dolling, Ulf-H, Reider, Paul J

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Process Development and Large-Scale Synthesis of a c-Met Kinase Inhibitor von Stewart, Gavin W, Brands, Karel M. J, Brewer, Sarah E, Cowden, Cameron J, Davies, Antony J, Edwards, John S, Gibson, Andrew W, Hamilton, Simon E, Katz, Jason D, Keen, Stephen P, Mullens, Peter R, Scott, Jeremy P, Wallace, Debra J, Wise, Christopher S

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Practical Asymmetric Synthesis of a γ-Secretase Inhibitor Exploiting Substrate-Controlled Intramolecular Nitrile Oxide−Olefin Cycloaddition von Scott, Jeremy P, Oliver, Steven F, Brands, Karel M. J, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Hands, David, Keen, Stephen P, Sheen, Faye J, Reamer, Robert A, Wilson, Robert D, Dolling, Ulf-H

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A Practical Synthesis of a γ-Secretase Inhibitor von Scott, Jeremy P, Lieberman, David R, Beureux, Olivier M, Brands, Karel M. J, Davies, Antony J, Gibson, Andrew W, Hammond, Deborah C, McWilliams, Chris J, Stewart, Gavin W, Wilson, Robert D, Dolling, Ulf-H

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A Double Ring Closing Metathesis Reaction in the Rapid, Enantioselective Synthesis of NK-1 Receptor Antagonists von Wallace, Debra J, Goodman, Jonathan M, Kennedy, Derek J, Davies, Antony J, Cowden, Cameron J, Ashwood, Michael S, Cottrell, Ian F, Dolling, Ulf-H, Reider, Paul J

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A Practical and Scaleable Synthesis of 1R,5S-Bicyclo[3.1.0]hexan-2-one:  The Development of a Catalytic Lithium 2,2,6,6-Tetramethylpiperidide (LTMP) Mediated Intramolecular Cyclopr... von Alorati, Anthony D, Bio, Matthew M, Brands, Karel M. J, Cleator, Ed, Davies, Antony J, Wilson, Robert D, Wise, Chris S

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A Novel Crystallization-Induced Diastereomeric Transformation Based on a Reversible Carbon−Sulfur Bond Formation. Application to the Synthesis of a γ-Secretase Inhibitor von Davies, Antony J, Scott, Jeremy P, Bishop, Brian C, Brands, Karel M. J, Brewer, Sarah E, DaSilva, Jimmy O, Dormer, Peter G, Dolling, Ulf-H, Gibb, Andrew D, Hammond, Deborah C, Lieberman, David R, Palucki, Michael, Payack, Joseph F

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Development of a Scaleable Synthesis of a Partial Nicotinic Acid Receptor Agonist von Wilson, Robert D, Cleator, Ed, Ashwood, Michael S, Bio, Matthew M, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf-H, Emerson, Khateeta M, Gibb, Andrew D, Hands, David, McKeown, Arlene E, Oliver, Steven F, Reamer, Robert A, Sheen, Faye J, Stewart, Gavin W, Zhou, George X

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An investigation into the alkylation of 1,2,4-triazole von Bulger, Paul G, Cottrell, Ian F, Cowden, Cameron J, Davies, Antony J, Dolling, Ulf-H

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An efficient and general synthesis of 3-substituted propionaldehydes using the Suzuki–Miyaura coupling von Cowden, Cameron J, Hammond, Deborah C, Bishop, Brian C, Brands, Karel M.J, Davies, Antony J, Dolling, Ulf-H, Brewer, Sarah E

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Development of a Scaleable Synthesis of a 3-Aminopyrazinone Acetamide Thrombin Inhibitor von Ashwood, Michael S, Alabaster, Ramon J, Cottrell, Ian F, Cowden, Cameron J, Davies, Antony J, Dolling, Ulf H, Emerson, Khateeta M, Gibb, Andrew D, Hands, David, Wallace, Debra J, Wilson, Robert D

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The conformational bias of aryl, arylsulfonyl geminally substituted tertiary carbon centers: applications in substrate-based stereocontrol von Scott, Jeremy P, Mullens, Peter R, Brewer, Sarah E, Brands, Karel M J, Chilenski, Jennifer R, Davies, Antony J, Gibb, Andrew D, Lieberman, David R, Oliver, Steven F, Dolling, Ulf-H

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Practical Asymmetric Synthesis of a Non-Peptidic αvβ3 Antagonist von Keen, Stephen P, Cowden, Cameron J, Bishop, Brian C, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf H, Lieberman, David R, Stewart, Gavin W

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Regioselective coupling reactions of 2,4-diaminopyridine derivatives with aryl halides: the synthesis of elaborated pyridines von Bio, Matthew M., Cleator, Ed, Davies, Antony J., Hamilton, Simon E., Lawrence, Andrew, Sheen, Faye J., Stewart, Gavin W., Wilson, Robert D.

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Practical Asymmetric Synthesis of a Non-Peptidic α v β 3 Antagonist von Keen, Stephen P., Cowden, Cameron J., Bishop, Brian C., Brands, Karel M. J., Davies, Antony J., Dolling, Ulf H., Lieberman, David R., Stewart, Gavin W.

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Regioselective coupling reactions of 2,4-diaminopyridine derivatives with aryl halides: the synthesis of elaborated pyridines: Modern Applications of Transition Metal Catalysis in... von BIO, Matthew M, CLEATOR, Ed, DAVIES, Antony J, HAMILTON, Simon E, LAWRENCE, Andrew, SHEEN, Faye J, STEWART, Gavin W, WILSON, Robert D

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Regioselective synthesis of N-substituted-4-substituted isothiazolidine-1,1-dioxides von Cleator, Ed, Sheen, Faye J., Bio, Matthew M., Jos Brands, K.M., Davies, Antony J., Dolling, Ulf-H.

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