A Nonpeptide Antagonist Reveals a Highly Glycosylated State of the Rabbit Kinin B1 Receptor von Fortin, Jean-Philippe, Dziadulewicz, Edward K, Gera, Lajos, Marceau, François

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Potent and Orally Bioavailable Non-Peptide Antagonists at the Human Bradykinin B1 Receptor Based on a 2-Alkylamino-5-sulfamoylbenzamide Core von Ritchie, Timothy J, Dziadulewicz, Edward K, Culshaw, Andrew J, Müller, Werner, Burgess, Gillian M, Bloomfield, Graham C, Drake, Gillian S, Dunstan, Andrew R, Beattie, David, Hughes, Glyn A, Ganju, Pam, McIntyre, Peter, Bevan, Stuart J, Davis, Clare, Yaqoob, Mohammed

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Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone:  A Potent, Orally Bioavailable Human CB1/CB2 Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous Sys... von Dziadulewicz, Edward K, Bevan, Stuart J, Brain, Christopher T, Coote, Paul R, Culshaw, Andrew J, Davis, Andrew J, Edwards, Lee J, Fisher, Adrian J, Fox, Alyson J, Gentry, Clive, Groarke, Alex, Hart, Terance W, Huber, Werner, James, Iain F, Kesingland, Adam, La Vecchia, Luigi, Loong, Yvonne, Lyothier, Isabelle, McNair, Kara, O'Farrell, Cathal, Peacock, Marcus, Portmann, Robert, Schopfer, Ulrich, Yaqoob, Mohammed, Zadrobilek, Jiri

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Non-peptide ligands for bradykinin receptors 1995 - 2004 von Dziadulewicz, Edward K

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Identification and Biological Characterization of 6-Aryl-7-isopropylquinazolinones as Novel TRPV1 Antagonists that Are Effective in Models of Chronic Pain von Culshaw, Andrew J, Bevan, Stuart, Christiansen, Martin, Copp, Prafula, Davis, Andrew, Davis, Clare, Dyson, Alex, Dziadulewicz, Edward K, Edwards, Lee, Eggelte, Hendrikus, Fox, Alyson, Gentry, Clive, Groarke, Alex, Hallett, Allan, Hart, Terance W, Hughes, Glyn A, Knights, Sally, Kotsonis, Peter, Lee, Wai, Lyothier, Isabelle, McBryde, Andrew, McIntyre, Peter, Paloumbis, George, Panesar, Moh, Patel, Sadhana, Seiler, Max-Peter, Yaqoob, Mohammed, Zimmermann, Kaspar

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Bradyzide, a potent non‐peptide B2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia von Burgess, Gillian M, Perkins, Martin N, Rang, Humphrey P, Campbell, Elizabeth A, Brown, Michael C, McIntyre, Peter, Urban, Laszlo, Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Wrigglesworth, Roger, Lee, Wai, Davis, Clare, Phagoo, Steve B, Davis, Andrew J, Phillips, Elsa, Drake, Gillian S, Hughes, Glyn A, Dunstan, Andrew, Bloomfield, Graham C

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A non-peptide antagonist unusually selective for the human form of the bradykinin B2 receptor von MARCEAU, Francois, FORTIN, Jean-Philippe, MORISSETTE, Guillaume, DZIADULEWICZ, Edward K

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Nonpeptide Bradykinin B2 Receptor Antagonists:  Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B2 Receptor Antagonists von Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Davies, John W, Wrigglesworth, Roger, Dunstan, Andrew R, Bloomfield, Graham C, Drake, Gillian S, McIntyre, Peter, Brown, Michael C, Burgess, Gillian M, Lee, Wai, Davis, Clare, Yaqoob, Mohammed, Phagoo, Steve B, Phillips, Elsa, Perkins, Martin N, Campbell, Elizabeth A, Davis, Andrew J, Rang, Humphrey P

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Bradyzide, a potent non‐peptide B 2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia von Burgess, Gillian M, Perkins, Martin N, Rang, Humphrey P, Campbell, Elizabeth A, Brown, Michael C, McIntyre, Peter, Urban, Laszlo, Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Wrigglesworth, Roger, Lee, Wai, Davis, Clare, Phagoo, Steve B, Davis, Andrew J, Phillips, Elsa, Drake, Gillian S, Hughes, Glyn A, Dunstan, Andrew, Bloomfield, Graham C

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1-(2-Nitrophenyl)thiosemicarbazides:  A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B2 Receptor von Dziadulewicz, Edward K, Ritchie, Timothy J, Hallett, Allan, Snell, Christopher R, Ko, Soo Y, Wrigglesworth, Roger, Hughes, Glyn A, Dunstan, Andrew R, Bloomfield, Graham C, Drake, Gillian S, Brown, Michael C, Lee, Wai, Burgess, Gillian M, Davis, Clare, Yaqoob, Mohammed, Perkins, Martin N, Campbell, Elizabeth A, Davis, Andrew J, Rang, Humphrey P

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Concise and regiospecific syntheses of tri-substituted 1,2,4-triazoles von Dunstan, Andrew R, Weber, Hans-Peter, Rihs, Grety, Widmer, Hans, Dziadulewicz, Edward K

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Mitsunobu alkylation of imidazole: a convenient route to chiral ionic liquids von Kim, Eun Jin, Ko, Soo Y., Dziadulewicz, Edward K.

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A Nonpeptide Antagonist Reveals a Highly Glycosylated State of the Rabbit Kinin B 1 Receptor von Fortin, Jean-Philippe, Dziadulewicz, Edward K., Gera, Lajos, Marceau, François

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Design of non-peptide CCK2 and NK1 peptidomimetics using 1-(2-nitrophenyl)thiosemicarbazide as a novel common scaffold von DZIADULEWICZ, Edward K, WALPOLE, Christopher S, SNELL, Christopher R, WRIGGLESWORTH, Roger, HUGHES, Glyn A, BEATTIE, David, WOOD, John N, BEECH, Margaret M, COOTE, Paul R

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Potent and Orally Bioavailable Non-Peptide Antagonists at the Human Bradykinin B 1 Receptor Based on a 2-Alkylamino-5-sulfamoylbenzamide Core von Ritchie, Timothy J., Dziadulewicz, Edward K., Culshaw, Andrew J., Müller, Werner, Burgess, Gillian M., Bloomfield, Graham C., Drake, Gillian S., Dunstan, Andrew R., Beattie, David, Hughes, Glyn A., Ganju, Pam, McIntyre, Peter, Bevan, Stuart J., Davis, Clare, Yaqoob, Mohammed

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The design of non-peptide human bradykinin B2 receptor antagonists employing the benzodiazepine peptidomimetic scaffold von DZIADULEWICZ, E. K, BROWN, M. C, DUNSTAN, A. R, WAI LEE, SAID, N. B, GARRATT, P. J

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A non-peptide antagonist unusually selective for the human form of the bradykinin B 2 receptor von Marceau, François, Fortin, Jean-Philippe, Morissette, Guillaume, Dziadulewicz, Edward K.

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Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone:  A Potent, Orally Bioavailable Human CB 1 /CB 2 Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous... von Dziadulewicz, Edward K., Bevan, Stuart J., Brain, Christopher T., Coote, Paul R., Culshaw, Andrew J., Davis, Andrew J., Edwards, Lee J., Fisher, Adrian J., Fox, Alyson J., Gentry, Clive, Groarke, Alex, Hart, Terance W., Huber, Werner, James, Iain F., Kesingland, Adam, La Vecchia, Luigi, Loong, Yvonne, Lyothier, Isabelle, McNair, Kara, O'Farrell, Cathal, Peacock, Marcus, Portmann, Robert, Schopfer, Ulrich, Yaqoob, Mohammed, Zadrobilek, Jiri

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Nonpeptide Bradykinin B 2 Receptor Antagonists:  Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B 2 Receptor Antagonists von Dziadulewicz, Edward K., Ritchie, Timothy J., Hallett, Allan, Snell, Christopher R., Davies, John W., Wrigglesworth, Roger, Dunstan, Andrew R., Bloomfield, Graham C., Drake, Gillian S., McIntyre, Peter, Brown, Michael C., Burgess, Gillian M., Lee, Wai, Davis, Clare, Yaqoob, Mohammed, Phagoo, Steve B., Phillips, Elsa, Perkins, Martin N., Campbell, Elizabeth A., Davis, Andrew J., Rang, Humphrey P.

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Identification and biological characterization of 6-aryl-7-isopropylquinazolinones as novel TRPV1 antagonists that are effective in models of chronicpain von CULSHAW, Andrew J, BEVAN, Stuart, FOX, Alyson, GENTRY, Clive, GROARKE, Alex, HALLETT, Allan, HART, Terance W, HUGHES, Glyn A, KNIGHTS, Sally, KOTSONIS, Peter, LEE, Wai, LYOTHIER, Isabelle, CHRISTIANSEN, Martin, MCBRYDE, Andrew, MCINTYRE, Peter, PALOUMBIS, George, PANESAR, Moh, PATEL, Sadhana, SEILER, Max-Peter, YAQOOB, Mohammed, ZIMMERMANN, Kaspar, COPP, Prafula, DAVIS, Andrew, DAVIS, Clare, DYSON, Alex, DZIADULEWICZ, Edward K, EDWARDS, Lee, EGGELTE, Hendrikus

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