Kinetics of Avibactam Inhibition against Class A, C, and D β-Lactamases von Ehmann, David E., Jahić, Haris, Ross, Philip L., Gu, Rong-Fang, Hu, Jun, Durand-Réville, Thomas F., Lahiri, Sushmita, Thresher, Jason, Livchak, Stephania, Gao, Ning, Palmer, Tiffany, Walkup, Grant K., Fisher, Stewart L.

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Rational design of a new antibiotic class for drug-resistant infections von Durand-Reville, Thomas F., Miller, Alita A., O’Donnell, John P., Wu, Xiaoyun, Sylvester, Mark A., Guler, Satenig, Iyer, Ramkumar, Shapiro, Adam B., Carter, Nicole M., Velez-Vega, Camilo, Moussa, Samir H., McLeod, Sarah M., Chen, April, Tanudra, Angela M., Zhang, Jing, Comita-Prevoir, Janelle, Romero, Jan A., Huynh, Hoan, Ferguson, Andrew D., Horanyi, Peter S., Mayclin, Stephen J., Heine, Henry S., Drusano, George L., Cummings, Jason E., Slayden, Richard A., Tommasi, Ruben A.

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Discovery and Characterization of New Hydroxamate Siderophores, Baumannoferrin A and B, produced by Acinetobacter baumannii von Penwell, William F., DeGrace, Nancy, Tentarelli, Sharon, Gauthier, Lise, Gilbert, Catherine M., Arivett, Brock A., Miller, Alita A., Durand-Reville, Thomas F., Joubran, Camil, Actis, Luis A.

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Structural Insight into Potent Broad-Spectrum Inhibition with Reversible Recyclization Mechanism: Avibactam in Complex with CTX-M-15 and Pseudomonas aeruginosa AmpC β-Lactamases von LAHIRI, Sushmita D, MANGANI, Stefano, DURAND-REVILLE, Thomas, BENVENUTI, Manuela, DE LUCA, Filomena, SANYAL, Gautam, DOCQUIER, Jean-Denis

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Spiropyrimidinetriones: a Class of DNA Gyrase Inhibitors with Activity against Mycobacterium tuberculosis and without Cross-Resistance to Fluoroquinolones von Basarab, Gregory S, Ghorpade, Sandeep, Gibhard, Liezl, Mueller, Rudolf, Njoroge, Mathew, Peton, Nashied, Govender, Preshendren, Massoudi, Lisa M, Robertson, Gregory Thomas, Lenaerts, Anne J, Boshoff, Helena Ingrid, Joerss, Douglas, Parish, Tanya, Durand-Reville, Thomas F, Perros, Manos, Singh, Vinayak, Chibale, Kelly

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Molecular Basis of Selective Inhibition and Slow Reversibility of Avibactam against Class D Carbapenemases: A Structure-Guided Study of OXA-24 and OXA-48 von Lahiri, Sushmita D, Mangani, Stefano, Jahić, Haris, Benvenuti, Manuela, Durand-Reville, Thomas F, De Luca, Filomena, Ehmann, David E, Rossolini, Gian Maria, Alm, Richard A, Docquier, Jean-Denis

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Discovery of an Orally Available Diazabicyclooctane Inhibitor (ETX0282) of Class A, C, and D Serine β‑Lactamases von Durand-Réville, Thomas F, Comita-Prevoir, Janelle, Zhang, Jing, Wu, Xiaoyun, May-Dracka, Tricia L, Romero, Jan Antoinette C, Wu, Frank, Chen, April, Shapiro, Adam B, Carter, Nicole M, McLeod, Sarah M, Giacobbe, Robert A, Verheijen, Jeroen C, Lahiri, Sushmita D, Sacco, Michael D, Chen, Yu, O’Donnell, John P, Miller, Alita A, Mueller, John P, Tommasi, Rubén A

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N-Hydroxyformamide LpxC inhibitors, their in vivo efficacy in a mouse Escherichia coli infection model, and their safety in a rat hemodynamic assay von Furuya, Takeru, Shapiro, Adam B., Comita-Prevoir, Janelle, Kuenstner, Eric J., Zhang, Jing, Ribe, Seth D., Chen, April, Hines, Daniel, Moussa, Samir H., Carter, Nicole M., Sylvester, Mark A., Romero, Jan A.C., Vega, Camilo V., Sacco, Michael D., Chen, Yu, O'Donnell, John P., Durand-Reville, Thomas F., Miller, Alita A., Tommasi, Ruben A.

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Acinetobacter baumannii OmpA Is a Selective Antibiotic Permeant Porin von Iyer, Ramkumar, Moussa, Samir H, Durand-Réville, Thomas F, Tommasi, Ruben, Miller, Alita

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Durlobactam, a New Diazabicyclooctane β-Lactamase Inhibitor for the Treatment of Acinetobacter Infections in Combination With Sulbactam von Shapiro, Adam B., Moussa, Samir H., McLeod, Sarah M., Durand-Réville, Thomas, Miller, Alita A.

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Whole-Cell-Based Assay To Evaluate Structure Permeation Relationships for Carbapenem Passage through the Pseudomonas aeruginosa Porin OprD von Iyer, Ramkumar, Sylvester, Mark A, Velez-Vega, Camilo, Tommasi, Ruben, Durand-Reville, Thomas F, Miller, Alita A

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ETX2514 is a broad-spectrum β-lactamase inhibitor for the treatment of drug-resistant Gram-negative bacteria including Acinetobacter baumannii von Durand-Réville, Thomas F., Guler, Satenig, Comita-Prevoir, Janelle, Chen, Brendan, Bifulco, Neil, Huynh, Hoan, Lahiri, Sushmita, Shapiro, Adam B., McLeod, Sarah M., Carter, Nicole M., Moussa, Samir H., Velez-Vega, Camilo, Olivier, Nelson B., McLaughlin, Robert, Gao, Ning, Thresher, Jason, Palmer, Tiffany, Andrews, Beth, Giacobbe, Robert A., Newman, Joseph V., Ehmann, David E., de Jonge, Boudewijn, O'Donnell, John, Mueller, John P., Tommasi, Rubén A., Miller, Alita A.

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Discovery of Efficacious Pseudomonas aeruginosa-Targeted Siderophore-Conjugated Monocarbams by Application of a Semi-mechanistic Pharmacokinetic/Pharmacodynamic Model von Murphy-Benenato, Kerry E, Bhagunde, Pratik R, Chen, April, Davis, Hajnalka E, Durand-Réville, Thomas F, Ehmann, David E, Galullo, Vincent, Harris, Jennifer J, Hatoum-Mokdad, Holia, Jahić, Haris, Kim, Aryun, Manjunatha, M. R, Manyak, Erika L, Mueller, John, Patey, Sara, Quiroga, Olga, Rooney, Michael, Sha, Li, Shapiro, Adam B, Sylvester, Mark, Tan, Beesan, Tsai, Andy S, Uria-Nickelsen, Maria, Wu, Ye, Zambrowski, Mark, Zhao, Shannon X

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Enantioselective Synthesis and Profiling of Two Novel Diazabicyclooctanone β‑Lactamase Inhibitors von Xiong, Hui, Chen, Brendan, Durand-Réville, Thomas F, Joubran, Camil, Alelyunas, Yun W, Wu, Dedong, Huynh, Hoan

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SAR and Structural Analysis of Siderophore-Conjugated Monocarbam Inhibitors of Pseudomonas aeruginosa PBP3 von Murphy-Benenato, Kerry E, Dangel, Brian, Davis, Hajnalka E, Durand-Réville, Thomas F, Ferguson, Andrew D, Gao, Ning, Jahić, Haris, Mueller, John P, Manyak, Erika L, Quiroga, Olga, Rooney, Michael, Sha, Li, Sylvester, Mark, Wu, Frank, Zambrowski, Mark, Zhao, Shannon X

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Highly Selective Entry to the Azadirachtin Skeleton via a Claisen Rearrangement/Radical Cyclization Sequence von Durand-Reville, Thomas, Gobbi, Luca B, Gray, Brian Lawrence, Ley, Steven V, Scott, James S

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The Synthesis of Azadirachtin: A Potent Insect Antifeedant von Ley, Steven V., Abad-Somovilla, Antonio, Anderson, James C., Ayats, Carles, Bänteli, Rolf, Beckmann, Edith, Boyer, Alistair, Brasca, Maria G., Brice, Abigail, Broughton, Howard B., Burke, Brenda J., Cleator, Ed, Craig, Donald, Denholm, Alastair A., Denton, Ross M., Durand-Reville, Thomas, Gobbi, Luca B., Göbel, Michael, Gray, Brian Lawrence, Grossmann, Robert B., Gutteridge, Claire E., Hahn, Norbert, Harding, Sarah L., Jennens, David C., Jennens, Lynn, Lovell, Peter J., Lovell, Helen J., de la Puente, Mary L., Kolb, Hartmuth C., Koot, Win-Jan, Maslen, Sarah L., McCusker, Catherine F., Mattes, Amos, Pape, Andrew R., Pinto, Andrea, Santafianos, Dinos, Scott, James S., Smith, Stephen C., Somers, Andrew Q., Spilling, Christopher D., Stelzer, Frank, Toogood, Peter L., Turner, Richard M., Veitch, Gemma E., Wood, Anthony, Zumbrunn, Cornelia

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ChemInform Abstract: Tungsten(0) Alkylidene Complexes Stabilized as Pyridinium Ylides: New Aspects of Their Synthesis and Reactivity von Rudler, Henri, Durand-Reville, Thomas

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Combination therapy for treatment of resistant bacterial infections von Durand-Reville, Thomas, Tommasi, Ruben, Dejonge, Boudewijn, Mueller, John, Verheijen, Jeroen

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METHOD OF CALCINING A CLAY MATERIAL von DION, Pascal, DURAND-REVILLE, Thomas

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