Large-Scale Applications of Transition Metal-Catalyzed Couplings for the Synthesis of Pharmaceuticals von Magano, Javier, Dunetz, Joshua R

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Large-Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals von Dunetz, Joshua R, Magano, Javier, Weisenburger, Gerald A

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Large-Scale Carbonyl Reductions in the Pharmaceutical Industry von Magano, Javier, Dunetz, Joshua R

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Synthesis of Highly Substituted Indolines and Indoles via Intramolecular [4 + 2] Cycloaddition of Ynamides and Conjugated Enynes von Dunetz, Joshua R, Danheiser, Rick L

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Copper-Mediated N-Alkynylation of Carbamates, Ureas, and Sulfonamides. A General Method for the Synthesis of Ynamides von Dunetz, Joshua R, Danheiser, Rick L

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Discovery and Preclinical Characterization of 1‑Methyl‑3-(4‑methylpyridin‑3‑yl)‑6‑(pyridin‑2‑ylmethoxy)‑1H‑pyrazolo-[3,4‑b]­pyrazine (PF470): A Highly Potent, Selective, and Effica... von Zhang, Lei, Balan, Gayatri, Barreiro, Gabriela, Boscoe, Brian P, Chenard, Lois K, Cianfrogna, Julie, Claffey, Michelle M, Chen, Laigao, Coffman, Karen J, Drozda, Susan E, Dunetz, Joshua R, Fonseca, Kari R, Galatsis, Paul, Grimwood, Sarah, Lazzaro, John T, Mancuso, Jessica Y, Miller, Emily L, Reese, Matthew R, Rogers, Bruce N, Sakurada, Isao, Skaddan, Marc, Smith, Deborah L, Stepan, Antonia F, Trapa, Patrick, Tuttle, Jamison B, Verhoest, Patrick R, Walker, Daniel P, Wright, Ann S, Zaleska, Margaret M, Zasadny, Kenneth, Shaffer, Christopher L

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General and Scalable Amide Bond Formation with Epimerization-Prone Substrates Using T3P and Pyridine von Dunetz, Joshua R, Xiang, Yanqiao, Baldwin, Aaron, Ringling, Justin

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Total Syntheses of (+)-Tedanolide and (+)-13-Deoxytedanolide von Dunetz, Joshua R, Julian, Lisa D, Newcom, Jason S, Roush, William R

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Mapping Polymorphic Behavior of Process Intermediates, an Often-Overlooked Exercise von Morrison, Henry, Regens, Christopher S, Dunetz, Joshua R, Lapina, Olga, Shah, Nisha P, Burke, Brenda J, Wenderski, Todd, Asselin, Sylvie M, Vieira, Tiago

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Chiral separation of amides using supercritical fluid chromatography von Xiang, Yanqiao, Dunetz, Joshua R., Lovdahl, Michael

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Rapid Enabling of Negishi Couplings for a Pair of mGluR5 Negative Allosteric Modulators von Gontcharov, Alexander, Dunetz, Joshua R

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Discovery and Characterization of (R)‑6-Neopentyl-2-(pyridin-2-ylmethoxy)-6,7-dihydropyrimido[2,1‑c][1,4]oxazin-4(9H)‑one (PF-06462894), an Alkyne-Lacking Metabotropic Glutamate Re... von Stepan, Antonia F, Claffey, Michelle M, Reese, Matthew R, Balan, Gayatri, Barreiro, Gabriela, Barricklow, Jason, Bohanon, Michael J, Boscoe, Brian P, Cappon, Gregg D, Chenard, Lois K, Cianfrogna, Julie, Chen, Laigao, Coffman, Karen J, Drozda, Susan E, Dunetz, Joshua R, Ghosh, Somraj, Hou, Xinjun, Houle, Christopher, Karki, Kapil, Lazzaro, John T, Mancuso, Jessica Y, Marcek, John M, Miller, Emily L, Moen, Mark A, O’Neil, Steven, Sakurada, Isao, Skaddan, Marc, Parikh, Vinod, Smith, Deborah L, Trapa, Patrick, Tuttle, Jamison B, Verhoest, Patrick R, Walker, Daniel P, Won, Annie, Wright, Ann S, Whritenour, Jessica, Zasadny, Kenneth, Zaleska, Margaret M, Zhang, Lei, Shaffer, Christopher L

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Sonogashira Reactions with Propyne: Facile Synthesis of 4-Hydroxy-2-methylbenzofurans from Iodoresorcinols von Berliner, Martin A, Cordi, Eric M, Dunetz, Joshua R, Price, Kristin E

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Concerning the Synthesis of the Tedanolide C(13)−C(23) Fragment via Anti-Aldol Reaction von Dunetz, Joshua R, Roush, William R

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Multikilogram Synthesis of a Hepatoselective Glucokinase Activator von Dunetz, Joshua R, Berliner, Martin A, Xiang, Yanqiao, Houck, Timothy L, Salingue, Fabrice H, Chao, Wang, Yuandong, Chen, Shenghua, Wang, Huang, Yun, Farrand, Douglas, Boucher, Steven J, Damon, David B, Makowski, Teresa W, Barrila, Mark T, Chen, Raymond, Martínez, Isamir

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[2+2] Cycloaddition of ketenes with ynamides. A general method for the synthesis of 3-aminocyclobutenone derivatives von Kohnen, Amanda L., Mak, Xiao Yin, Lam, Tin Yiu, Dunetz, Joshua R., Danheiser, Rick L.

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Self-Assembling Porphyrin-Modified Peptides von Dunetz, Joshua R, Sandstrom, Claire, Young, Elizabeth R, Baker, Paul, Van Name, Steven A, Cathopolous, Terry, Fairman, Robert, de Paula, Julio C, Åkerfeldt, Karin S

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Pictet-Spengler reactions in multiphasic supercritical carbon dioxide/CO2-expanded liquid media. In situ generation of carbamates as a strategy for reactions of amines in supercrit... von Dunetz, Joshua R, Ciccolini, Rocco P, Fröling, Morgan, Paap, Scott M, Allen, Andrew J, Holmes, Andrew B, Tester, Jefferson W, Danheiser, Rick L

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Spotlight on Non-Precious Metal Catalysis von Dunetz, Joshua R., Fandrick, Daniel, Federsel, Hans-Jürgen

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ChemInform Abstract: Recent Large-Scale Applications of Transition Metal-Catalyzed Couplings for the Synthesis of Pharmaceuticals von Magano, Javier, Dunetz, Joshua R.

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