Large-Scale Carbonyl Reductions in the Pharmaceutical Industry von Magano, Javier, Dunetz, Joshua R

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Large-Scale Applications of Transition Metal-Catalyzed Couplings for the Synthesis of Pharmaceuticals von Magano, Javier, Dunetz, Joshua R

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Large-Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals von Dunetz, Joshua R, Magano, Javier, Weisenburger, Gerald A

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Rapid Enabling of Negishi Couplings for a Pair of mGluR5 Negative Allosteric Modulators von Gontcharov, Alexander, Dunetz, Joshua R

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Concerning the Synthesis of the Tedanolide C(13)−C(23) Fragment via Anti-Aldol Reaction von Dunetz, Joshua R, Roush, William R

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Discovery and Preclinical Characterization of 1‑Methyl‑3-(4‑methylpyridin‑3‑yl)‑6‑(pyridin‑2‑ylmethoxy)‑1H‑pyrazolo-[3,4‑b]­pyrazine (PF470): A Highly Potent, Selective, and Efficacious Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator von Zhang, Lei, Balan, Gayatri, Barreiro, Gabriela, Boscoe, Brian P, Chenard, Lois K, Cianfrogna, Julie, Claffey, Michelle M, Chen, Laigao, Coffman, Karen J, Drozda, Susan E, Dunetz, Joshua R, Fonseca, Kari R, Galatsis, Paul, Grimwood, Sarah, Lazzaro, John T, Mancuso, Jessica Y, Miller, Emily L, Reese, Matthew R, Rogers, Bruce N, Sakurada, Isao, Skaddan, Marc, Smith, Deborah L, Stepan, Antonia F, Trapa, Patrick, Tuttle, Jamison B, Verhoest, Patrick R, Walker, Daniel P, Wright, Ann S, Zaleska, Margaret M, Zasadny, Kenneth, Shaffer, Christopher L

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Copper-Mediated N-Alkynylation of Carbamates, Ureas, and Sulfonamides. A General Method for the Synthesis of Ynamides von Dunetz, Joshua R, Danheiser, Rick L

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General and Scalable Amide Bond Formation with Epimerization-Prone Substrates Using T3P and Pyridine von Dunetz, Joshua R, Xiang, Yanqiao, Baldwin, Aaron, Ringling, Justin

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Total Syntheses of (+)-Tedanolide and (+)-13-Deoxytedanolide von Dunetz, Joshua R, Julian, Lisa D, Newcom, Jason S, Roush, William R

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Chiral separation of amides using supercritical fluid chromatography von Xiang, Yanqiao, Dunetz, Joshua R., Lovdahl, Michael

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Mapping Polymorphic Behavior of Process Intermediates, an Often-Overlooked Exercise von Morrison, Henry, Regens, Christopher S, Dunetz, Joshua R, Lapina, Olga, Shah, Nisha P, Burke, Brenda J, Wenderski, Todd, Asselin, Sylvie M, Vieira, Tiago

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ChemInform Abstract: Large‐Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals von Dunetz, Joshua R., Magano, Javier, Weisenburger, Gerald A.

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ChemInform Abstract: Recent Large-Scale Applications of Transition Metal-Catalyzed Couplings for the Synthesis of Pharmaceuticals von Magano, Javier, Dunetz, Joshua R.

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Discovery and Characterization of (R)‑6-Neopentyl-2-(pyridin-2-ylmethoxy)-6,7-dihydropyrimido[2,1‑c][1,4]oxazin-4(9H)‑one (PF-06462894), an Alkyne-Lacking Metabotropic Glutamate Receptor 5 Negative Allosteric Modulator Profiled in both Rat and Nonhuman Primates von Stepan, Antonia F, Claffey, Michelle M, Reese, Matthew R, Balan, Gayatri, Barreiro, Gabriela, Barricklow, Jason, Bohanon, Michael J, Boscoe, Brian P, Cappon, Gregg D, Chenard, Lois K, Cianfrogna, Julie, Chen, Laigao, Coffman, Karen J, Drozda, Susan E, Dunetz, Joshua R, Ghosh, Somraj, Hou, Xinjun, Houle, Christopher, Karki, Kapil, Lazzaro, John T, Mancuso, Jessica Y, Marcek, John M, Miller, Emily L, Moen, Mark A, O’Neil, Steven, Sakurada, Isao, Skaddan, Marc, Parikh, Vinod, Smith, Deborah L, Trapa, Patrick, Tuttle, Jamison B, Verhoest, Patrick R, Walker, Daniel P, Won, Annie, Wright, Ann S, Whritenour, Jessica, Zasadny, Kenneth, Zaleska, Margaret M, Zhang, Lei, Shaffer, Christopher L

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Sonogashira Reactions with Propyne: Facile Synthesis of 4-Hydroxy-2-methylbenzofurans from Iodoresorcinols von Berliner, Martin A, Cordi, Eric M, Dunetz, Joshua R, Price, Kristin E

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Pictet-Spengler reactions in multiphasic supercritical carbon dioxide/CO2-expanded liquid media. In situ generation of carbamates as a strategy for reactions of amines in supercritical carbon dioxide von Dunetz, Joshua R, Ciccolini, Rocco P, Fröling, Morgan, Paap, Scott M, Allen, Andrew J, Holmes, Andrew B, Tester, Jefferson W, Danheiser, Rick L

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[2+2] Cycloaddition of ketenes with ynamides. A general method for the synthesis of 3-aminocyclobutenone derivatives von Kohnen, Amanda L., Mak, Xiao Yin, Lam, Tin Yiu, Dunetz, Joshua R., Danheiser, Rick L.

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Spotlight on Non-Precious Metal Catalysis von Dunetz, Joshua R., Fandrick, Daniel, Federsel, Hans-Jürgen

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