Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 1: Discovery and initial structure-activity relationships for 1-amino-2-phenyl-4-(piperidin-1-yl)butanes von DORN, Conrad P, FINKE, Paul E, DEMARTINO, Julie A, SICILIANO, Salvatore J, CARELLA, Anthony, CARVER, Gwen, HOLMES, Karen, DANZEISEN, Renee, HAZUDA, Daria, KESSLER, Joseph, LINEBERGER, Janet, MILLER, Michael, OATES, Bryan, SCHLEIF, William A, EMINI, Emilio A, BUDHU, Richard J, MILLS, Sander G, MACCOSS, Malcolm, MALKOWITZ, Lorraine, SPRINGER, Martin S, DAUGHERTY, Bruce L, GOULD, Sandra L

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Phosphorylated Morpholine Acetal Human Neurokinin-1 Receptor Antagonists as Water-Soluble Prodrugs von Hale, Jeffrey J, Mills, Sander G, MacCoss, Malcolm, Dorn, Conrad P, Finke, Paul E, Budhu, Richard J, Reamer, Robert A, Huskey, Su-Er W, Luffer-Atlas, Debra, Dean, Brian J, McGowan, Erin M, Feeney, William P, Chiu, Shuet-Hing Lee, Cascieri, Margaret A, Chicchi, Gary G, Kurtz, Marc M, Sadowski, Sharon, Ber, Elzbieta, Tattersall, F. David, Rupniak, Nadia M. J, Williams, Angela R, Rycroft, Wayne, Hargreaves, Richard, Metzger, Joseph M, MacIntyre, D. Euan

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Orally active .beta.-lactam inhibitors of human leukocyte elastase-1. Activity of 3,3-diethyl-2-azetidinones von Shah, Shrenik K, Dorn, Conrad P, Finke, Paul E, Hale, Jeffrey J, Hagmann, William K, Brause, Karen A, Chandler, Gilbert O, Kissinger, Amy L, Ashe, Bonnie M

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Expression and characterization of the chemokine receptor CCR2B from rhesus monkey von Jin, Hong, Vicario, Pasquale P., Zweerink, Hans, Goyal, Shefali, Hanlon, William A., Dorn, Conrad P., Mills, Sander G., DeMartino, Julie A., Cascieri, Margaret A., Struthers, Mary

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Orally active .beta.-lactam inhibitors of human leukocyte elastase. 2. Effect of C-4 substitution von Hagmann, William K, Kissinger, Amy L, Shah, Shrenik K, Finke, Paul E, Dorn, Conrad P, Brause, Karen A, Ashe, Bonnie M, Weston, Hazel, Maycock, Alan L

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Inhibition of human leukocyte elastase. 1. Inhibition by C-7-substituted cephalosporin tert-butyl esters von Doherty, James B, Ashe, Bonnie M, Barker, Peter L, Blacklock, Thomas J, Butcher, John W, Chandler, Gilbert O, Dahlgren, M. Ellen, Davies, Philip, Dorn, Conrad P

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Synthesis and immunoadjuvant activities of 2-acetamido-5-O-acetyl-6-O-acyl-2-deoxy-3-O-[(R)-2-propionyl-L-alanyl-D-isoglutamine]-D-glucofuranoses as potential prodrug forms of 6-O-... von Durette, Philippe L, Dorn, Conrad P, Friedman, Arthur, Schlabach, Abner

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Synthesis and antiinflammatory/analgesic activities of 11H-dibenzo[b,e]dioxepinacetic acids von Hagmann, William K, Dorn, Conrad P, Frankshun, Robert A, O'Grady, Laura A, Bailey, Philip J, Rackham, Anita, Dougherty, Harry W

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Proteinase inhibitors. 1. Inhibitors of elastase von Dorn, Conrad P, Zimmerman, Morris, Yang, Shu Shu, Yurewicz, Edward C, Ashe, Bonnie M, Frankshun, Robert, Jones, Howard

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Steroids XXIII. Synthesis of Some Ring A-Fused Heterocyclic Steroids von Doorenbos, Norman J., Dorn, Conrad P.

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Steroids IX: Synthesis of Some Thiazolosteroids von Doorenbos, Norman J., Dorn, Conrad P.

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LU91069I von MacCOSS Malcolm, HARRISON Timothy, HALE Jeffrey, J, DORN Conrad, P, MILLS Sander, G, SHAH Shrenik, K, WILLIAMS Brian John, LADDUWAHETTY Tamara, FINKE Paul, E, CHAMBERS Mark Stuart

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Chemical, Biochemical, Pharmacokinetic, and Biological Properties of L-680, 833: A Potent, Orally Active Monocyclic β-Lactam Inhibitor of Human Polymorphonuclear Leukocyte Elastase... von Doherty, James B., Shah, Shrenik K., Finke, Paul E., Dorn, Conrad P., Hagmann, William K., Hale, Jeffrey J., Kissinger, Amy L., Thompson, Kevan R., Brause, karen, Chandler, Gilbert O., Knight, Wilson B., Maycock, Alan L., Ashe, Bonnie M., Weston, Hazel, Gale, Paul, Mumford, Richard A., Andersen, O. Frederick, Williams, Hollis R., Nolan, Thomas E., Frankenfield, Dale L., Underwood, Dennis, Vyas, Kamlesh P., Kari, Prasad H., Dahlgren, Mary E., Mao, Jennifer, Fletcher, Daniel S., Pa. S. Dellea, Hand, Karen M., Osinga, Donald G., Peterson, Laurence B., Williams, Dorsey T., Metzger, Joseph M., Bonney, Robert J., Humes, John L., Pacholok, Steven P., Hanlon, William A., Opas, Evan, Stolk, Jan, Davies, Philip

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Cephalosporin antibiotics can be modified to inhibit human leukocyte elastase von Doherty, James B., Ashe, Bonnie M., Argenbright, Lawrence W., Barker, Peter L., Bonney, Robert J., Chandler, Gilbert O., Dahlgren, Mary Ellen, Dorn, Conrad P., Finke, Paul E., Firestone, Raymond A., Fletcher, Daniel, Hagmann, William K., Mumford, Richard, O'Grady, Laura, Maycock, Alan L., Pisano, Judith M., Shah, Shrenik K., Thompson, Kevan R., Zimmerman, Morris

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Inhibition of human leukocyte elastase. 4. Selection of a substituted cephalosporin (L-658,758) as a topical aerosol von Finke, Paul E, Shah, Shrenik K, Ashe, Bonnie M, Ball, Richard G, Blacklock, Thomas J, Bonney, Robert J, Brause, Karen A, Chandler, Gilbert O, Cotton, Meredith

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AMINOALKYLPHENOLS, METHODS OF USING AND MAKING THE SAME von WYVRATT, MATTHEW, J, DORN, CONRAD, P, POWLES, MARY, ANN, WALSH, THOMAS, F

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MORPHOLINE AND THIOMORPHOLINE TACHYKININ RECEPTOR ANTAGONISTS von SHAH, SHRENIK K, HARRISON, TIMOTHY, LADDUWAHETTY, TAMARA, WILIAMS, BRIAN JOHNS, CHAMBERS, MARK STUART, FINKE, PAUL E, DORN, CONRAD P, MACCOSS, MALCOLM, MILLS, SANDER G, HALE, JEFFREY J

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1,4-Diacylpiperazine-2-(S)-[(N-aminoalkyl)carboxamides] as novel, potent substance P receptor antagonists von Mills, Sander G., Wu, Mu Tsu, MacCoss, Malcolm, Budhu, Richard J., Dorn, Conrad P., Cascieri, Margaret A., Sadowski, Sharon, Strader, Catherine D., Greenlee, William J.

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AMINOALKYLPHENOLS, METHODS OF USING AND MAKING THE SAME von WALSH, THOMAS F, DORN, CONRAD P, WYVRATT, MATTHEW J, POWLES, MARY ANN

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Proteoglycan-Degrading Activity of Human Stromelysin-1 and Leukocyte Elastase in Rabbit Joints. Quantitation of Proteoglycan and a Stromelysin-lnduced HABR Fragment of Aggrecan in... von Olszewski, Julie M., Moore, Vernon L., McDonnell, Joseph, Williams, Hollis, Saphos, Cheryl A., Green, Barbara G., Knight, Wilson B., Chapman, Kevin T., Hagmann, William K., Dorn, Conrad P., Hale, Jeffrey J., Mumford, Richard A.

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