Crystal structures of human glycine receptor α3 bound to a novel class of analgesic potentiators von Huang, Xin, Shaffer, Paul L, Ayube, Shawn, Bregman, Howard, Chen, Hao, Lehto, Sonya G, Luther, Jason A, Matson, David J, McDonough, Stefan I, Michelsen, Klaus, Plant, Matthew H, Schneider, Stephen, Simard, Jeffrey R, Teffera, Yohannes, Yi, Shuyan, Zhang, Maosheng, DiMauro, Erin F, Gingras, Jacinthe

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Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors von Bregman, Howard, Chakka, Nagasree, Guzman-Perez, Angel, Gunaydin, Hakan, Gu, Yan, Huang, Xin, Berry, Virginia, Liu, Jingzhou, Teffera, Yohannes, Huang, Liyue, Egge, Bryan, Mullady, Erin L, Schneider, Steve, Andrews, Paul S, Mishra, Ankita, Newcomb, John, Serafino, Randy, Strathdee, Craig A, Turci, Susan M, Wilson, Cindy, DiMauro, Erin F

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Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors von DiMauro, Erin F, Altmann, Stephen, Berry, Loren M, Bregman, Howard, Chakka, Nagasree, Chu-Moyer, Margaret, Bojic, Elma Feric, Foti, Robert S, Fremeau, Robert, Gao, Hua, Gunaydin, Hakan, Guzman-Perez, Angel, Hall, Brian E, Huang, Hongbing, Jarosh, Michael, Kornecook, Thomas, Lee, Josie, Ligutti, Joseph, Liu, Dong, Moyer, Bryan D, Ortuno, Daniel, Rose, Paul E, Schenkel, Laurie B, Taborn, Kristin, Wang, Jean, Wang, Yan, Yu, Violeta, Weiss, Matthew M

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Inhibition of Inactive States of Tetrodotoxin-Sensitive Sodium Channels Reduces Spontaneous Firing of C-Fiber Nociceptors and Produces Analgesia in Formalin and Complete Freund's A... von Matson, David J, Hamamoto, Darryl T, Bregman, Howard, Cooke, Melanie, DiMauro, Erin F, Huang, Liyue, Johnson, Danielle, Li, Xingwen, McDermott, Jeff, Morgan, Carrie, Wilenkin, Ben, Malmberg, Annika B, McDonough, Stefan I, Simone, Donald A

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Structure-guided Discovery of Dual-recognition Chemibodies von Cheng, Alan C., Doherty, Elizabeth M., Johnstone, Sheree, DiMauro, Erin F., Dao, Jennifer, Luthra, Abhinav, Ye, Jay, Tang, Jie, Nixey, Thomas, Min, Xiaoshan, Tagari, Philip, Miranda, Les P., Wang, Zhulun

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Discovery of a biarylamide series of potent, state-dependent NaV1.7 inhibitors von Schenkel, Laurie B., DiMauro, Erin F., Nguyen, Hanh N., Chakka, Nagasree, Du, Bingfan, Foti, Robert S., Guzman-Perez, Angel, Jarosh, Michael, La, Daniel S., Ligutti, Joseph, Milgram, Benjamin C., Moyer, Bryan D., Peterson, Emily A., Roberts, John, Yu, Violeta L., Weiss, Matthew M.

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Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement von Marx, Isaac E, Dineen, Thomas A, Able, Jessica, Bode, Christiane, Bregman, Howard, Chu-Moyer, Margaret, DiMauro, Erin F, Du, Bingfan, Foti, Robert S, Fremeau, Robert T, Gao, Hua, Gunaydin, Hakan, Hall, Brian E, Huang, Liyue, Kornecook, Thomas, Kreiman, Charles R, La, Daniel S, Ligutti, Joseph, Lin, Min-Hwa Jasmine, Liu, Dong, McDermott, Jeff S, Moyer, Bryan D, Peterson, Emily A, Roberts, Jonathan T, Rose, Paul, Wang, Jean, Youngblood, Beth D, Yu, Violeta, Weiss, Matthew M

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Structure-Based Design of 2‑Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors von Huang, Hongbing, Guzman-Perez, Angel, Acquaviva, Lisa, Berry, Virginia, Bregman, Howard, Dovey, Jennifer, Gunaydin, Hakan, Huang, Xin, Huang, Liyue, Saffran, Doug, Serafino, Randy, Schneider, Steve, Wilson, Cindy, DiMauro, Erin F

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Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors von Sparling, Brian A., DiMauro, Erin F.

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Discovery and Optimization of a Novel Series of N-Arylamide Oxadiazoles as Potent, Highly Selective and Orally Bioavailable Cannabinoid Receptor 2 (CB2) Agonists von Cheng, Yuan, Albrecht, Brian K, Brown, James, Buchanan, John L, Buckner, William H, DiMauro, Erin F, Emkey, Renee, Fremeau, Robert T, Harmange, Jean-Christophe, Hoffman, Beth J, Huang, Liyue, Huang, Ming, Lee, Josie Han, Lin, Fen-Fen, Martin, Matthew W, Nguyen, Hung Q, Patel, Vinod F, Tomlinson, Susan A, White, Ryan D, Xia, Xiaoyang, Hitchcock, Stephen A

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Rapid Synthesis of 3-Amino-imidazopyridines by a Microwave-Assisted Four-Component Coupling in One Pot von DiMauro, Erin F, Kennedy, Joseph M

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Catalysis of the Michael Addition Reaction by Late Transition Metal Complexes of BINOL-Derived Salens von Annamalai, Venkatachalam, DiMauro, Erin F, Carroll, Patrick J, Kozlowski, Marisa C

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Discovery of a Class of Novel Tankyrase Inhibitors that Bind to Both the Nicotinamide Pocket and the Induced Pocket von Bregman, Howard, Gunaydin, Hakan, Gu, Yan, Schneider, Steve, Wilson, Cindy, DiMauro, Erin F, Huang, Xin

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Structure-Guided Discovery of Aminoquinazolines as Brain-Penetrant and Selective LRRK2 Inhibitors von Keylor, Mitchell H, Gulati, Anmol, Kattar, Solomon D, Johnson, Rebecca E, Chau, Ryan W, Margrey, Kaila A, Ardolino, Michael J, Zarate, Cayetana, Poremba, Kelsey E, Simov, Vladimir, Morriello, Gregori J, Acton, John J, Pio, Barbara, Yan, Xin, Palte, Rachel L, McMinn, Spencer E, Nogle, Lisa, Lesburg, Charles A, Adpressa, Donovon, Lin, Shishi, Neelamkavil, Santhosh, Liu, Ping, Su, Jing, Hegde, Laxminarayan G, Woodhouse, Janice D, Faltus, Robert, Xiong, Tina, Ciaccio, Paul J, Piesvaux, Jennifer, Otte, Karin M, Wood, Harold B, Kennedy, Matthew E, Bennett, David Jonathan, DiMauro, Erin F, Fell, Matthew J, Fuller, Peter H

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Enhancing the Visibility of Women in the ACS Division of Medicinal Chemistry (ACS MEDI) von Aldrich, Jane, Allen, Shelley, Araujo, Erika, Bronson, Joanne, Bryant-Friedrich, Amanda, Cyr, Shana K., DiMauro, Erin F., Dzierba, Carolyn, Garner, Amanda L., Georg, Gunda I., Goodwin, Nicole C., Haranahalli, Krupanandan, Huang, Rong, Leftheris, Katerina, May-Dracka, Tricia L., Olson, Margaret E., Blanco, Maria-Jesus

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Discovery and Optimization of N‑Heteroaryl Indazole LRRK2 Inhibitors von Logan, Kaitlyn M., Kaplan, Will, Simov, Vladimir, Zhou, Hua, Li, Derun, Torres, Luis, Morriello, Gregori J., Acton, John J., Pio, Barbara, Chen, Yi-Heng, Keylor, Mitchell H., Johnson, Rebecca, Kattar, Solomon D., Chau, Ryan, Yan, Xin, Ardolino, Michael, Zarate, Cayetana, Otte, Karin M., Palte, Rachel L., Xiong, Tina, McMinn, Spencer E., Lin, Shishi, Neelamkavil, Santhosh F., Liu, Ping, Su, Jing, Hegde, Laxminarayan G., Woodhouse, Janice D., Moy, Lily Y., Ciaccio, Paul J., Piesvaux, Jennifer, Zebisch, Matthias, Henry, Clare, Barker, John, Wood, Harold B., Kennedy, Matthew E., DiMauro, Erin F., Fell, Matthew J., Fuller, Peter H.

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Live cell screening to identify RNA-binding small molecule inhibitors of the pre-let-7-Lin28 RNA-protein interaction von Rosenblum, Sydney L, Soueid, Dalia M, Giambasu, George, Vander Roest, Steve, Pasternak, Alexander, DiMauro, Erin F, Simov, Vladimir, Garner, Amanda L

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Discovery of MK-1468: A Potent, Kinome-Selective, Brain-Penetrant Amidoisoquinoline LRRK2 Inhibitor for the Potential Treatment of Parkinson’s Disease von Kattar, Solomon D., Gulati, Anmol, Margrey, Kaila A., Keylor, Mitchell H., Ardolino, Michael, Yan, Xin, Johnson, Rebecca, Palte, Rachel L., McMinn, Spencer E., Nogle, Lisa, Su, Jing, Xiao, Dong, Piesvaux, Jennifer, Lee, Susi, Hegde, Laxminarayan G., Woodhouse, Janice D., Faltus, Robert, Moy, Lily Y., Xiong, Tina, Ciaccio, Paul J., Pearson, Kara, Patel, Mayankbhai, Otte, Karin M., Leyns, Cheryl E.G., Kennedy, Matthew E., Bennett, David Jonathan, DiMauro, Erin F., Fell, Matthew J., Fuller, Peter H.

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Discovery and characterization of novel peptide inhibitors of the NRF2/MAFG/DNA ternary complex for the treatment of cancer von Simov, Vladimir, Altman, Michael D., Bianchi, Elisabetta, DelRizzo, Sonia, DiNunzio, Edward N., Feng, Guo, Goldenblatt, Peter, Ingenito, Raffaele, Johnson, Scott A., Mansueto, My Sam, Mayhood, Todd, Mortison, Jonathan D., Serebrov, Victor, Sondey, Christopher, Sriraman, Venkat, Tucker, Thomas J., Walji, Abbas, Wan, Hui, Yue, Yingzi, Stoeck, Alexander, DiMauro, Erin F.

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Empowering Voices: Inspiring Women in Medicinal Chemistry von Blanco, Maria-Jesus, Bronson, Joanne J., DiMauro, Erin F., Dzierba, Carolyn, Eggen, MariJean, Garner, Amanda L., Georg, Gunda, Giarolla, Jeanine, Goodwin, Nicole C., Grenier-Davies, Melissa C., Haskell-Luevano, Carrie, Holzgrabe, Ulrike, Huang, Rong, Lagiakos, H. Rachel, Leftheris, Katerina, Martin, Yvonne, Matos, Maria João, May-Dracka, Tricia L., Müller, Christa E., Newman, Amy H., Parmee, Emma, Petter, Jennifer C., Tamayo, Nuria A., Wexler, Ruth R., Bolognesi, Maria Laura, Ripka, Amy, Young, Wendy

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