Locations of the Hydrophobic Side Chains of Lipoglycopeptides Bound to the Peptidoglycan of Staphylococcus aureus von Kim, Sung Joon, Tanaka, Kelly S. E, Dietrich, Evelyne, Rafai Far, Adel, Schaefer, Jacob

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CCNE1 amplification is synthetic lethal with PKMYT1 kinase inhibition von Gallo, David, Young, Jordan T. F., Fourtounis, Jimmy, Martino, Giovanni, Álvarez-Quilón, Alejandro, Bernier, Cynthia, Duffy, Nicole M., Papp, Robert, Roulston, Anne, Stocco, Rino, Szychowski, Janek, Veloso, Artur, Alam, Hunain, Baruah, Prasamit S., Fortin, Alexanne Bonneau, Bowlan, Julian, Chaudhary, Natasha, Desjardins, Jessica, Dietrich, Evelyne, Fournier, Sara, Fugère-Desjardins, Chloe, Goullet de Rugy, Theo, Leclaire, Marie-Eve, Liu, Bingcan, Bhaskaran, Vivek, Mamane, Yael, Melo, Henrique, Nicolas, Olivier, Singhania, Akul, Szilard, Rachel K., Tkáč, Ján, Yin, Shou Yun, Morris, Stephen J., Zinda, Michael, Marshall, C. Gary, Durocher, Daniel

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Discovery of an Orally Bioavailable and Selective PKMYT1 Inhibitor, RP-6306 von Szychowski, Janek, Papp, Robert, Dietrich, Evelyne, Liu, Bingcan, Vallée, Frédéric, Leclaire, Marie-Eve, Fourtounis, Jimmy, Martino, Giovanni, Perryman, Alexander L., Pau, Victor, Yin, Shou Yun, Mader, Pavel, Roulston, Anne, Truchon, Jean-Francois, Marshall, C. Gary, Diallo, Mohamed, Duffy, Nicole M., Stocco, Rino, Godbout, Claude, Bonneau-Fortin, Alexanne, Kryczka, Rosie, Bhaskaran, Vivek, Mao, Daniel, Orlicky, Stephen, Beaulieu, Patrick, Turcotte, Pascal, Kurinov, Igor, Sicheri, Frank, Mamane, Yael, Gallant, Michel, Black, W. Cameron

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Novel non-nucleobase inhibitors of Staphylococcus aureus DNA polymerase IIIC von Rose, Yannick, Ciblat, Stéphane, Reddy, Ranga, Belley, Adam C., Dietrich, Evelyne, Lehoux, Dario, McKay, Geoffrey A., Poirier, Hugo, Far, Adel Rafai, Delorme, Daniel

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Oritavancin Exhibits Dual Mode of Action to Inhibit Cell-Wall Biosynthesis in Staphylococcus aureus von Kim, Sung Joon, Cegelski, Lynette, Stueber, Dirk, Singh, Manmilan, Dietrich, Evelyne, Tanaka, Kelly S.E., Parr, Thomas R., Far, Adel Rafai, Schaefer, Jacob

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Vancomycin and Oritavancin Have Different Modes of Action in Enterococcus faecium von Patti, Gary J., Kim, Sung Joon, Yu, Tsyr-Yan, Dietrich, Evelyne, Tanaka, Kelly S.E., Parr, Thomas R., Far, Adel Rafai, Schaefer, Jacob

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Linking Bisphosphonates to the Free Amino Groups in Fluoroquinolones: Preparation of Osteotropic Prodrugs for the Prevention of Osteomyelitis von Houghton, Tom J, Tanaka, Kelly S. E, Kang, Ting, Dietrich, Evelyne, Lafontaine, Yanick, Delorme, Daniel, Ferreira, Sandra S, Viens, Frederic, Arhin, Francis F, Sarmiento, Ingrid, Lehoux, Dario, Fadhil, Ibtihal, Laquerre, Karine, Liu, Jing, Ostiguy, Valérie, Poirier, Hugo, Moeck, Gregory, Parr, Thomas R, Far, Adel Rafai

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Synthesis and evaluation of NS5A inhibitors containing diverse heteroaromatic cores von Henderson, James A., Bilimoria, Darius, Bubenik, Monica, Cadilhac, Caroline, Cottrell, Kevin M., Denis, Francois, Dietrich, Evelyne, Ewing, Nigel, Falardeau, Guy, Giroux, Simon, L’Heureux, Lucille, Liu, Bingcan, Mani, Nagraj, Morris, Mark, Nicolas, Olivier, Pereira, Oswy Z., Poisson, Carl, Reddy, T. Jagadeeswar, Selliah, Subajini, Shawgo, Rebecca S., Vaillancourt, Louis, Wang, Jian, Xu, Jinwang, Chauret, Nathalie, Berlioz-Seux, Francoise, Chan, Laval C., Das, Sanjoy K., Grillot, Anne-Laure, Bennani, Youssef L., Maxwell, John P.

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Benzimidazole-containing HCV NS5A inhibitors: Effect of 4-substituted pyrrolidines in balancing genotype 1a and 1b potency von Henderson, James A., Bilimoria, Darius, Bubenik, Monica, Cadilhac, Caroline, Cottrell, Kevin M., Dietrich, Evelyne, Denis, Francois, Ewing, Nigel, Falardeau, Guy, Giroux, Simon, Grey, Ronald, L’Heureux, Lucille, Liu, Bingcan, Mani, Nagraj, Morris, Mark, Nicolas, Olivier, Pereira, Oswy Z., Poisson, Carl, Govinda Rao, B., Reddy, T. Jagadeeswar, Selliah, Subajini, Shawgo, Rebecca S., Vaillancourt, Louis, Wang, Jian, Yannopoulos, Constantin G., Chauret, Nathalie, Berlioz-Seux, Francoise, Chan, Laval C., Das, Sanjoy K., Grillot, Anne-Laure, Bennani, Youssef L., Maxwell, John P.

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Efficient Synthesis of Enantiopure Pyrrolizidinone Amino Acid von Dietrich, Evelyne, Lubell, William D

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Discovery of thienoimidazole-based HCV NS5A inhibitors. Part 1: C sub(2)-Symmetric inhibitors with diyne and biphenyl linkers von Giroux, Simon, Bilimoria, Darius, Cadilhac, Caroline, Cottrell, Kevin M, Denis, Francois, Dietrich, Evelyne, Ewing, Nigel, Henderson, James A, L'Heureux, Lucille, Mani, Nagraj, Morris, Mark, Nicolas, Olivier, Reddy, TJagadeeswar, Selliah, Subajini, Shawgo, Rebecca S, Xu, Jinwang, Chauret, Nathalie, Berlioz-Seux, Francoise, Chan, Laval C, Das, Sanjoy K, Grillot, Anne-Laure, Bennani, Youssef L, Maxwell, John P

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Discovery of thienoimidazole-based HCV NS5A inhibitors. Part 1: C2-Symmetric inhibitors with diyne and biphenyl linkers von Giroux, Simon, Bilimoria, Darius, Cadilhac, Caroline, Cottrell, Kevin M., Denis, Francois, Dietrich, Evelyne, Ewing, Nigel, Henderson, James A., L’Heureux, Lucille, Mani, Nagraj, Morris, Mark, Nicolas, Olivier, Reddy, T. Jagadeeswar, Selliah, Subajini, Shawgo, Rebecca S., Xu, Jinwang, Chauret, Nathalie, Berlioz-Seux, Francoise, Chan, Laval C., Das, Sanjoy K., Grillot, Anne-Laure, Bennani, Youssef L., Maxwell, John P.

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Discovery of thienoimidazole-based HCV NS5A inhibitors. Part 2: Non-symmetric inhibitors with potent activity against genotype 1a and 1b von Giroux, Simon, Bilimoria, Darius, Cadilhac, Caroline, Cottrell, Kevin M., Denis, Francois, Dietrich, Evelyne, Ewing, Nigel, Henderson, James A., L’Heureux, Lucille, Mani, Nagraj, Morris, Mark, Nicolas, Olivier, Reddy, T. Jagadeeswar, Selliah, Subajini, Shawgo, Rebecca S., Xu, Jinwang, Chauret, Nathalie, Berlioz-Seux, Francoise, Chan, Laval C., Das, Sanjoy K., Grillot, Anne-Laure, Bennani, Youssef L., Maxwell, John P.

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Synthesis and in vitro evaluation of bisphosphonated glycopeptide prodrugs for the treatment of osteomyelitis von Tanaka, Kelly S.E., Dietrich, Evelyne, Ciblat, Stéphane, Métayer, Claude, Arhin, Francis F., Sarmiento, Ingrid, Moeck, Gregory, Parr, Thomas R., Far, Adel Rafai

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Bisphosphonated fluoroquinolone esters as osteotropic prodrugs for the prevention of osteomyelitis von Tanaka, Kelly S.E., Houghton, Tom J., Kang, Ting, Dietrich, Evelyne, Delorme, Daniel, Ferreira, Sandra S., Caron, Laurence, Viens, Frederic, Arhin, Francis F., Sarmiento, Ingrid, Lehoux, Dario, Fadhil, Ibtihal, Laquerre, Karine, Liu, Jing, Ostiguy, Valérie, Poirier, Hugo, Moeck, Gregory, Parr, Thomas R., Rafai Far, Adel

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A new class of small molecule RNA polymerase inhibitors with activity against Rifampicin-resistant Staphylococcus aureus von ARHIN, Francis, BELANGER, Odette, MCKAY, Geoffrey A, MOECK, Greg, REDDY, Ranga, ROSE, Yannick, SRIKUMAR, Ramakrishnan, TANAKA, Kelly S. E, WILLIAMS, Daniel M, GROS, Philippe, PELLETIER, Jerry, PARR, Thomas R, CIBLAT, Stéphane, FAR, Adel Rafai, DEHBI, Mohammed, DELORME, Daniel, DIETRICH, Evelyne, DIXIT, Dilip, LAFONTAINE, Yanick, LEHOUX, Dario, JING LIU

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Bisphosphonated Benzoxazinorifamycin Prodrugs for the Prevention and Treatment of Osteomyelitis von Reddy, Ranga, Dietrich, Evelyne, Lafontaine, Yanick, Houghton, Tom J., Belanger, Odette, Dubois, Anik, Arhin, Francis F., Sarmiento, Ingrid, Fadhil, Ibtihal, Laquerre, Karine, Ostiguy, Valerie, Lehoux, Dario, Moeck, Gregory, Parr Jr, Thomas R., Rafai Far, Adel

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TRICYCLIC HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME von VALLÉE, Frédéric, SZYCHOWSKI, Janek, DIETRICH, Evelyne

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Mannose derivatives for treating bacterial infections von Gallant, Michel, Vallee, Frederic, Dietrich, Evelyne, Vaillancourt, Louis, Truchon, Jean-Francois, Reddy, Thumkunta

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N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (THIAZOLYL)])(SUBSTITUTED)CARBOXAMIDE COMPOUNDS AND USE THEREOF FOR INHIBITING HUMAN POLYMERASE THETA von PERRYMAN, Alexander, SOW, Boubacar, LIU, Bingcan, MOCHIRIAN, Philippe, SURPRENANT, Simon, BENDAHAN, David, BUBENIK, Monica, SZYCHOWSKI, Janek, DIETRICH, Evelyne, GALLANT, Michel

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