Fragment-Derived Selective Inhibitors of Dual-Specificity Kinases DYRK1A and DYRK1B von Lee Walmsley, David, Murray, James B, Dokurno, Pawel, Massey, Andrew J, Benwell, Karen, Fiumana, Andrea, Foloppe, Nicolas, Ray, Stuart, Smith, Julia, Surgenor, Allan E, Edmonds, Thomas, Demarles, Didier, Burbridge, Mike, Cruzalegui, Francisco, Kotschy, Andras, Hubbard, Roderick E

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Discovery of S64315, a Potent and Selective Mcl‑1 Inhibitor von Szlavik, Zoltan, Csekei, Marton, Paczal, Attila, Szabo, Zoltan B, Sipos, Szabolcs, Radics, Gabor, Proszenyak, Agnes, Balint, Balazs, Murray, James, Davidson, James, Chen, Ijen, Dokurno, Pawel, Surgenor, Allan E, Daniels, Zoe Marie, Hubbard, Roderick E, Le Toumelin-Braizat, Gaëtane, Claperon, Audrey, Lysiak-Auvity, Gaëlle, Girard, Anne-Marie, Bruno, Alain, Chanrion, Maia, Colland, Frédéric, Maragno, Ana-Leticia, Demarles, Didier, Geneste, Olivier, Kotschy, Andras

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Structure-Guided Discovery of Potent and Selective DYRK1A Inhibitors von Weber, Csaba, Sipos, Melinda, Paczal, Attila, Balint, Balazs, Kun, Vilibald, Foloppe, Nicolas, Dokurno, Pawel, Massey, Andrew J, Walmsley, David Lee, Hubbard, Roderick E, Murray, James, Benwell, Karen, Edmonds, Thomas, Demarles, Didier, Bruno, Alain, Burbridge, Mike, Cruzalegui, Francisco, Kotschy, Andras

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Structure-Guided Discovery of Selective USP7 Inhibitors with In Vivo Activity von Vasas, Attila, Ivanschitz, Lisa, Molnár, Balázs, Kiss, Árpád, Baker, Lisa, Fiumana, Andrea, Macias, Alba, Murray, James B., Sanders, Emma, Whitehead, Neil, Hubbard, Roderick E., Saunier, Carine, Monceau, Elodie, Girard, Anne Marie, Rousseau, Marion, Chanrion, Maia, Demarles, Didier, Geneste, Olivier, Weber, Csaba, Lewkowicz, Elodie, Kotschy, Andras

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Structure-Guided Discovery of a Selective Mcl‑1 Inhibitor with Cellular Activity von Szlávik, Zoltan, Ondi, Levente, Csékei, Márton, Paczal, Attila, Szabó, Zoltán B, Radics, Gábor, Murray, James, Davidson, James, Chen, Ijen, Davis, Ben, Hubbard, Roderick E, Pedder, Christopher, Dokurno, Pawel, Surgenor, Allan, Smith, Julia, Robertson, Alan, LeToumelin-Braizat, Gaetane, Cauquil, Nicolas, Zarka, Marion, Demarles, Didier, Perron-Sierra, Francoise, Claperon, Audrey, Colland, Frederic, Geneste, Olivier, Kotschy, András

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Steady-State Pharmacokinetics of Amprenavir Coadministered with Ritonavir in Human Immunodeficiency Virus Type 1-Infected Patients von GOUJARD, Cecile, VINCENT, Isabelle, MEYNARD, Jean-Luc, CHOUDET, Nathalie, BOLLENS, Diane, ROUSSEAU, Cyril, DEMARLES, Didier, GILLOTIN, Catherine, BIDAULT, Roselyne, TABURET, Anne-Marie

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Abstract LB220: The anticalin-antibody bispecific PRS-352/S095025 strongly stimulates human CD4+ T cells in a PD-L1-dependent manner von Pattarini, Lucia, Pavlidou, Marina, Morales, Aizea Kastresana, Peper-Gabriel, Janet, Riviere, Matthieu, Demarles, Didier, Scholer-Dahirel, Alix, Blanc, Veronique, Olwill, Shane

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A Comparison of the Steady-State Pharmacokinetics and Safety of Abacavir, Lamivudine, and Zidovudine Taken as a Triple Combination Tablet and as Abacavir plus a Lamivudine-Zidovudi... von Crémieux, Anne-Claude, Katlama, Christine, Gillotin, Catherine, Demarles, Didier, Yuen, Geoffrey J., Raffi, Francois

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New hydroxyester derivatives, a process for their preparation and pharmaceutical compositions containing them von Geneste, Olivier, Paczal, Attila, Davidson, James Edward Paul, Kotschy, András, Demarles, Didier, Sipos, Szabolcs, Murray, James Brooke, Chanrion, Maïa, Bálint, Balázs, Szlávik, Zoltán

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NEW AMMONIUM DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von CHANRION, Maia, SZLAVIK, Zoltan, MARAGNO, ANA LETICIA, GENESTE, Olivier, SIPOS, Szabolcs, KOTSCHY, Andras, DEMARLES, Didier, PACZAL, Attila, BALINT, Balazs

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5-[7-(3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBONYL)-1,2,3,4 TETRAHYDROISOQUINOLIN-6-Y L]-1H-PYRROLE-3-CARBOXAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES... von SANDERS, Emma, MURRAY, James Brooke, SIPOS, Zoltán, BALASSA, Annamária, BROUGH, Paul Andrew, RAY, Stuart, KOMJÁTI, Balázs, SIPOS, Melinda, SZLÁVIK, Zoltán, ROCCHETTI, Francesca, WANG, Yikang, FÖRDŐS, Eszter, MADDOX, Daniel, DEMARLES, Didier, CLAPERON, Audrey, MOLNÁR, Balázs, WALMSLEY, Claire Louise, FEJES, Imre

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NEW PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von CHANRION, Maia, VASAS, Attila, KISS, Arpad, MURRAY, James Brooke, GENESTE OLIVIER, LEWKOWICZ, Elodie, KOTSCHY, Andras, DEMARLES, Didier, WEBER, Csaba, MOLNAR, Balazs, MACIAS, Alba

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NEW (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von CHANRION, Maia, VASAS, Attila, KISS, Arpad, MURRAY, James Brooke, IVANSCHITZ, Lisa, GENESTE OLIVIER, LEWKOWICZ, Elodie, KOTSCHY, Andras, DEMARLES, Didier, WEBER, Csaba, MOLNAR, Balazs, MACIAS, Alba

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5-[7-(3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBONYL)-1,2,3,4 TETRAHYDROISOQUINOLIN-6-Y L]-1H-PYRROLE-3-CARBOXAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES... von SANDERS, Emma, MURRAY, James Brooke, SIPOS, Zoltán, BALASSA, Annamária, BROUGH, Paul Andrew, RAY, Stuart, KOMJÁTI, Balázs, SIPOS, Melinda, SZLÁVIK, Zoltán, ROCCHETTI, Francesca, WANG, Yikang, FÖRDŐS, Eszter, MADDOX, Daniel, DEMARLES, Didier, CLAPERON, Audrey, MOLNÁR, Balázs, WALMSLEY, Claire Louise, FEJES, Imre

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NEW AMMONIUM DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von MARAGNO, Ana Leticia, SZLÁVIK, Zoltán, BÁLINT, Balázs, GENESTE, Olivier, SIPOS, Szabolcs, CHANRION, Maïa, DEMARLES, Didier, PACZAL, Attila, KOTSCHY, András

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NEW HYDROXYESTER DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von Zoltan SZLAVIK, James Edward Paul DAVIDSON, Balazs BALINT, Maia CHANRION, Didier DEMARLES, Olivier GENESTE, Szabolcs SIPOS, Attila PACZAL, James Brooke MURRAY, Andras KOTSCHY

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New ammonium derivatives, a process for their preparation and pharmaceutical compositions containing them von Geneste, Olivier, Paczal, Attila, Kotschy, András, Maragno, Ana Leticia, Demarles, Didier, Sipos, Szabolcs, Chanrion, Maïa, Bálint, Balázs, Szlávik, Zoltán

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NEW AMMONIUM DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von PACZAL, ATTILA, SIPOS, SZABOLCS, CHANRION, MAIA, MARAGNO, ANA LETICIA, BALINT, BALAZS, DEMARLES, DIDIER, SZLAVIK, ZOLTAN, GENESTE, OLIVIER, KOTSCHY, ANDRAS

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NEW (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von VASAS, Attila, MURRAY, James Brooke, IVANSCHITZ, Lisa, LEWKOWICZ, Elodie, KISS, Árpád, GENESTE, Olivier, CHANRION, Maïa, DEMARLES, Didier, WÉBER, Csaba, KOTSCHY, András, MOLNÁR, Balázs, MACIAS, Alba

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AMINO-PYRIMIDONYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von VASAS, Attila, DAVIES, Nicolas, MURRAY, James Brooke, IVANSCHITZ, Lisa, KISS, Árpád, GENESTE, Olivier, WÉBER, Csaba, SELLIER, Emilie, DEMARLES, Didier, KOTSCHY, András, MOLNÁR, Balázs, FIUMANA, Andrea, MACIAS, Alba

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