Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs): Discovery of capromorelin von Carpino, Philip A, Lefker, Bruce A, Toler, Steven M, Pan, Lydia C, Hadcock, John R, Cook, Ewell R, DiBrino, Joseph N, Campeta, Anthony M, DeNinno, Shari L, Chidsey-Frink, Kristin L, Hada, William A, Inthavongsay, John, Mangano, F.Michael, Mullins, Michelle A, Nickerson, David F, Ng, Oicheng, Pirie, Christine M, Ragan, John A, Rose, Colin R, Tess, David A, Wright, Ann S, Yu, Li, Zawistoski, Michael P, DaSilva-Jardine, Paul A, Wilson, Theresa C, Thompson, David D

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Discovery and biological characterization of capromorelin analogues with extended half-lives von Carpino, Philip A., Lefker, Bruce A., Toler, Steven M., Pan, Lydia C., Hadcock, John R., Murray, Marianne C., Cook, Ewell R., DiBrino, Joseph N., DeNinno, Shari L., Chidsey-Frink, Kristin L., Hada, William A., Inthavongsay, John, Lewis, Sharon K., Mangano, F.Michael, Mullins, Michelle A., Nickerson, David F., Ng, Oicheng, Pirie, Christine M., Ragan, John A., Rose, Colin R., Tess, David A., Wright, Ann S., Yu, Li, Zawistoski, Michael P., Pettersen, John C., DaSilva-Jardine, Paul A., Wilson, Theresa C., Thompson, David D.

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Discovery of 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylamino-piperidine-4-carboxylic Acid Amide Hydrochloride (CP-945,598), a Novel, Potent, and Selective Cann... von GRIFFITH, David A, HADCOCK, John R, O'CONNOR, Rebecca E, SCOTT, Dennis O, BLACK, Shawn C, IREDALE, Philip A, CARPINO, Philip A, DASILVA-JARDINE, Paul, DAY, Robert, DIBRINO, Joseph, DOW, Robert L, LANDIS, Margaret S

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Discovery of 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride (CP-945,598), a Novel, Potent, and Selective Canna... von Griffith, David A, Hadcock, John R, Black, Shawn C, Iredale, Philip A, Carpino, Philip A, DaSilva-Jardine, Paul, Day, Robert, DiBrino, Joseph, Dow, Robert L, Landis, Margaret S, O’Connor, Rebecca E, Scott, Dennis O

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Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity von Brandt, Thomas A., Caron, Stéphane, Damon, David B., DiBrino, Joseph, Ghosh, Arun, Griffith, David A., Kedia, Sandeep, Ragan, John A., Rose, Peter R., Vanderplas, Brian C., Wei, Lulin

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SYNTHESIS, IN VITRO AND IN VIVO ACTIVITY OF NOVEL 9-DEOXO-9a-AZA-9a-HOMOERYTHROMYCIN A DERIVATIVES; A NEW CLASS OF MACROLIDE ANTIBIOTICS, THE AZALIDES von BRIGHT, G. MICHAEL, NAGEL, ARTHUR A., BORDNER, JON, DESAI, KISHOR A., DIBRINO, JOSEPH N., NOWAKOWSKA, JOLANTA, VINCENT, LAWRENCE, WATROUS, RICHARD M., SCIAVOLINO, FRANK C., ENGLISH, ARTHUR R., RETSEMA, JAMES A., ANDERSON, MARGARET R., BRENNAN, LORI A., BOROVOY, ROBERTA J., CIMOCHOWSKI, CAROLINE R., FAIELLA, JAMES A., GIRARD, ARTHUR E., GIRARD, DENNIS, HERBERT, CAROL, MANOUSOS, MARY, MASON, RACHEL

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Identification of novel series of pyrazole and indole-urea based DFG-out PYK2 inhibitors von Bhattacharya, Samit K., Aspnes, Gary E., Bagley, Scott W., Boehm, Markus, Brosius, Arthur D., Buckbinder, Leonard, Chang, Jeanne S., Dibrino, Joseph, Eng, Heather, Frederick, Kosea S., Griffith, David A., Griffor, Matthew C., Guimarães, Cristiano R.W., Guzman-Perez, Angel, Han, Seungil, Kalgutkar, Amit S., Klug-McLeod, Jacquelyn, Garcia-Irizarry, Carmen, Li, Jianke, Lippa, Blaise, Price, David A., Southers, James A., Walker, Daniel P., Wei, Liuqing, Xiao, Jun, Zawistoski, Michael P., Zhao, Xumiao

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New bicyclic cannabinoid receptor-1 (CB 1-R) antagonists von Carpino, Philip A., Griffith, David A., Sakya, Subas, Dow, Robert L., Black, Shawn C., Hadcock, John R., Iredale, Philip A., Scott, Dennis O., Fichtner, Michael W., Rose, Colin R., Day, Robert, Dibrino, Joseph, Butler, Mary, DeBartolo, Demetria B., Dutcher, Darrin, Gautreau, Denise, Lizano, Jeff S., O’Connor, Rebecca E., Sands, Michelle A., Kelly-Sullivan, Dawn, Ward, Karen M.

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Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity: Recent Advances in Synthetic Methodology: Development and Applications von BRANDT, Thomas A, CARON, Stéphane, LULIN WEI, DAMON, David B, DIBRINO, Joseph, GHOSH, Arun, GRIFFITH, David A, KEDIA, Sandeep, RAGAN, John A, ROSE, Peter R, VANDERPLAS, Brian C

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trans-3-benzyl-4-hydroxy-7-chromanylbenzoic acid derivatives as antagonists of the leukotriene B4 (LTB4) receptor von REITER, L. A, KOCH, K, DIBRINO, J. N, DOMINY, B. W, FARRELL, C. A, HINGORANI, G. P, MARTINELLI, G. J, RAMCHANDANI, M, WRIGHT, K. F, PISCOPIO, A. D, SHOWELL, H. J, ALPERT, R, BIGGERS, M. S, CHAMBERS, R. J, CONKLYN, M. J, COOPER, K, CORTINA, S. R

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Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs) von Carpino, Philip A, Lefker, Bruce A, Toler, Steven M, Pan, Lydia C, Hadcock, John R, Cook, Ewell R, DiBrino, Joseph N, Campeta, Anthony M, DeNinno, Shari L, Chidsey-Frink, Kristin L, Hada, William A, Inthavongsay, John, Mangano, F.Michael, Mullins, Michelle A, Nickerson, David F, Ng, Oicheng, Pirie, Christine M, Ragan, John A, Rose, Colin R, Tess, David A, Wright, Ann S, Yu, Li, Zawistoski, Michael P, DaSilva-Jardine, Paul A, Wilson, Theresa C, Thompson, David D

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trans-3-Benzyl-4-hydroxy-7-chromanylbenzoic acid derivatives as antagonists of the leukotriene B4 (LTB4) receptor von Reiter, L A, Koch, K, Piscopio, A D, Showell, H J, Alpert, R, Biggers, M S, Chambers, R J, Conklyn, M J, Cooper, K, Cortina, S R, Dibrino, J N, Dominy, B W, Farrell, C A, Hingorani, G P, Martinelli, G J, Ramchandani, M, Wright, K F

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Design and synthesis of novel FKBP inhibitors von Hauske, James R, Dorff, Peter, Julin, Susan, DiBrino, Joseph, Spencer, Robin, Williams, Rebecca

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trans-3-Benzyl-4-hydroxy-7-chromanylbenzoic acid derivatives as antagonists of the leukotriene B 4 (LTB 4) receptor von Reiter, Lawrence A., Koch, Kevin, Piscopio, Anthony D., Showell, Henry J., Alpert, Robbin, Biggers, Michael S., Chambers, Robert J., Conklyn, Maryrose J., Cooper, Kelvin, Cortina, Santo R., Dibrino, Joseph N., Dominy, Beryl W., Farrell, Cathy A., Hingorani, Gary P., Martinelli, Gary J., Ramchandani, Mukesh, Wright, Kathyrn F.

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Investigation of the effects of synthetic, non-cytotoxic immunophilin inhibitors on MDR von Hauske, James R., Kajiji, Shama, Dorff, Peter, Julin, Susan, DiBrino, Joseph, Paillet, Simone

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Ring contraction of oleandrose on the macrolide antibiotic oleandomycin with [(methoxycarbonyl)sulfamoyl]triethylammonium hydroxide inner salt von Nagel, Arthur A, DiBrino, Joseph, Vincent, Lawrence A, Retsema, James A

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Endogenous Peptides Bound to HLA-A3 Possess a Specific Combination of Anchor Residues that Permit Identification of Potential Antigenic Peptides von DiBrino, Marianne, Parker, Kenneth C., Shiloach, Joseph, Knierman, Michael, Lukszo, Jan, Turner, Richard V., Biddison, William E., Coligan, John E.

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The HLA-B14 peptide binding site can accommodate peptides with different combinations of anchor residues von DiBrino, M, Parker, K C, Margulies, D H, Shiloach, J, Turner, R V, Biddison, W E, Coligan, J E

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Endogenous peptides with distinct amino acid anchor residue motifs bind to HLA-A1 and HLA-B8 von DiBrino, M, Parker, KC, Shiloach, J, Turner, RV, Tsuchida, T, Garfield, M, Biddison, WE, Coligan, JE

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Identification of the Peptide Binding Motif for HLA-B44, One of the Most Common HLA-B Alleles in the Caucasian Population von DiBrino, Marianne, Parker, Kenneth C, Margulies, David H, Shiloach, Joseph, Turner, Richard V, Biddison, William E, Coligan, John E

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