Novel dual LSD1/HDAC6 inhibitor for the treatment of cancer von Gajendran, Chandru, Tantry, Subramanyam Janardhan, M, Naveen Sadhu, Mohammed, Zainuddin, Dewang, Purushottam, Hallur, Mahanandeesha, Nair, Sreekala, Vaithilingam, Krishnakumar, Nagayya, Basavaprabhu, Rajagopal, Sridharan, Sivanandhan, Dhanalakshmi

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Synthesis, biological evaluation and molecular modelling of 2,4-disubstituted-5-(6-alkylpyridin-2-yl)-1H-imidazoles as ALK5 inhibitors von Park, Myoung-Soon, Park, Hyun-Ju, An, Young Jae, Choi, Joon Hun, Cha, Geunyoung, Lee, Hwa Jeong, Park, So-Jung, Dewang, Purushottam M., Kim, Dae-Kee

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Synthesis, biological evaluation and molecular modelling of 2,4-disubstituted-5-(6-alkylpyridin-2-yl)-1 H -imidazoles as ALK5 inhibitors von Park, Myoung-Soon, Park, Hyun-Ju, An, Young Jae, Choi, Joon Hun, Cha, Geunyoung, Lee, Hwa Jeong, Park, So-Jung, Dewang, Purushottam M, Kim, Dae-Kee

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Synthesis and biological evaluation of 2-pyridyl-substituted pyrazoles and imidazoles as transforming growth factor-β type 1 receptor kinase inhibitors von Dewang, Purushottam M., Kim, Dae-Kee

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Determination of ulixertinib in mice plasma by LC–MS/MS and its application to a pharmacokinetic study in mice von Kumar, Rajinish, Suresh, P.S., Rudresh, G., Zainuddin, Mohd, Dewang, Purushottam, Kethiri, Ragahava Reddy, Rajagopal, Sriram, Mullangi, Ramesh

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Synthesis and biological evaluation of 4(5)-(6-methylpyridin-2-yl)imidazoles and -pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors von Kim, Dae-Kee, Lee, Yeon-Im, Lee, Yeon Woo, Dewang, Purushottam M., Sheen, Yhun Yhong, Kim, Yeo Woon, Park, Hyun-Ju, Yoo, Jakyung, Lee, Ho Soon, Kim, Yong-Kook

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Synthesis and biological evaluation of benzenesulfonamide-substituted 4-(6-alkylpyridin-2-yl)-5-(quinoxalin-6-yl)imidazoles as transforming growth factor-β type 1 receptor kinase i... von Kim, Dae-Kee, Jung, Sun Hee, Lee, Ho Soon, Dewang, Purushottam M.

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Synthesis and biological evaluation of trisubstituted imidazole derivatives as inhibitors of p38α mitogen-activated protein kinase von Kim, Dae-Kee, Lim, Jin-Hwi, Lee, Jung A., Dewang, Purushottam M.

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Novel dual LSD1/HDAC6 inhibitors for the treatment of multiple myeloma von Naveen Sadhu, M, Sivanandhan, Dhanalakshmi, Gajendran, Chandru, Tantry, Subramanyam, Dewang, Purushottam, Murugan, Kannan, Chickamunivenkatappa, Srinatha, Zainuddin, Mohd, Nair, Sreekala, Vaithilingam, Krishnakumar, Rajagopal, Sridharan

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Abstract B150: ASN007, a novel oral ERK inhibitor, shows robust antitumor activity in RAS mutant cancer models von Reddy, Sanjeeva P., Sivanandhan, Dhanalakshmi, Dewang, Purushottam, Rao, Niranjan, Smith, Roger A., Thompson, Scott K.

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LC–MS/MS-ESI method for simultaneous quantification of darolutamide and its active metabolite, ORM-15341 in mice plasma and its application to a pharmacokinetic study von Dittakavi, Sreekanth, Nagasuri, Pavan Kumar V.S.P., Sulochana, Suresh P., Saim, Syed Mohd, Mallurwar, Sadanand R., Zainuddin, Mohd, Dewang, Purushottam, Rajagopal, Sriram, Mullangi, Ramesh

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Abstract 1382: Novel dual inhibitors of LSD1-HDAC6/8 for treatment of cancer von Dhanalakshmi, Sivanandhan, Rajagopal, Sridharan, Nair, Sreekala, Gajendran, Chandru, Ghosh, Dimpy, Tantry, Subramanyam Janardhan, Dewang, Purushottam, Hallur, Mahanandeesha, Kannan, M, KC, Srinatha, Kuntrapaku, Damodara, Dilipkumar, M, Sharma, Radha, Meghashree, S, Kumar, D P., Zainuddin, Mohd, Vinod, A B., Rajagopal, Sriram

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Abstract 11: Novel dual inhibitors of LSD1-HDAC6/8 for treatment of cancer von Sivanandhan, Dhanalakshmi, Rajagopal, Sridharan, Nair, Sreekala, Gajendran, Chandru, Ghosh, Dimpy, Nagaraj, P, Tantry, Subramanyam J., Dewang, Purushottam, Hallur, Mahanandeesha S., Murugan, Kannan, C, Srinatha K., Kuntrapaku, Damodara, Dilipkumar, M, Sharma, R, Meghashree, S, Kumar, Durga Prasanna, Ingle, Suraj P., Zainuddin, Mohd, Vinod, A B., Rajagopal, Sriram

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Eco-Friendly Pest Management Using Monoterpenoids. I. Antifungal Efficacy of Thymol Derivatives von Kumbhar, Pramod, Dewang, Purushottam M

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Abstract 187: ASN0007, a potent ERK12 inhibitor with strong antitumor activity in multiple RAS mutant models von Reddy, Sanjeeva P, Sivanandhan, Dhanalakshmi, Kethiri, Raghava Reddy, Nair, Sreekala, Dewang, Purushottam, Zainuddin, Mohd, Vaithilingam, Krishnakumar, Smith, Roger A, Gupta, Sandeep, Thompson, Scott K

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Abstract 187: ASN0007, a potent ERK1/2 inhibitor with strong antitumor activity in multiple RAS mutant models von Reddy, Sanjeeva P., Sivanandhan, Dhanalakshmi, Kethiri, Raghava Reddy, Nair, Sreekala, Dewang, Purushottam, Zainuddin, Mohd, Vaithilingam, Krishnakumar, Smith, Roger A., Gupta, Sandeep, Thompson, Scott K.

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Abstract 5860: Novel, first-in-class dual inhibitors of lysine specific demethylase 1 (LSD1) and histone deacetylatse 1 (HDAC) for treatment of cancer von Sivanandhan, Dhanalakshmi, Nair, Sreekala, Tantry, Subramaniyam, Rajagopal, Sridharan, Hallur, Mahanandeesha, M, Kannan, KC, Srinatha, K, Damodara, M, Dilipkumar, G, Chandru, Ghosh, Dimpy, N, Pradeep, Singh, Anuj Kumar, Zainuddin, Mohd, G, Rudresh, Sharma, Radha, S, Meghashree, Kumar, Durga P., Dewang, Purushottam, Rajagopal, Sriram

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Synthesis and biological evaluation of 2-pyridyl-substituted pyrazoles and imidazoles as transforming growth factor-b type 1 receptor kinase inhibitors von Dewang, Purushottam M, Kim, Dae-Kee

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Validation of an LC–MS/MS method for simultaneous detection of four HDAC inhibitors – belinostat, panobinostat, rocilinostat and vorinostat in mouse plasma and its application to a... von Giri, Kalpesh Kumar, Suresh, P. S., Saim, Syed Mohd, Zainuddin, Mohd, Bhamidipati, Ravi Kanth, Dewang, Purushottam, Hallur, Mahanandeesha S., Rajagopal, Sridharan, Rajagopal, Sriram, Mullangi, Ramesh

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Abstract 3509: Novel dual inhibitors of LSD1-HDAC for treatment of cancer von Sivanandhan, Dhanalakshmi, Rajagopalan, Sridharan, Nair, Sreekala, Dewang, Purushottam, Kumar, Durga Prasanna, Mulakala, Chandrika, Mahadevan, Lavanya, Skariah, Neema, Kavuru, Venkata Giri, Kuntrapaku, Damodara, Sajja, Suchitra, Zainuddin, Mohammad, V, Krishnakumar, Singh, Ritu, V, Swarnakumari, Gosu, Ramachandraiah, Aiyar, Jayashree, Iyer, Pravin, Rajagopal, Sriram

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