8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: Water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors von Brunschweiger, Andreas, Koch, Pierre, Schlenk, Miriam, Rafehi, Muhammad, Radjainia, Hamid, Küppers, Petra, Hinz, Sonja, Pineda, Felipe, Wiese, Michael, Hockemeyer, Jörg, Heer, Jag, Denonne, Frédéric, Müller, Christa E.

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Acetamide Scanning around Bicyclic Thiazoles: SAR at the H 3 Receptor von Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean‐Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent

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Lead Optimization of Thiazolo[5,4-c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H3R Inverse Agonists von Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie

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Phenyl‐oxazoles, a New Family of Inverse Agonists at the H 3 Histamine Receptor von Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie‐Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent

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Discovery of new C3aR ligands. Part 1: Arginine derivatives von Denonne, Frédéric, Binet, Sophie, Burton, Maggi, Collart, Philippe, Dipesa, Alan, Ganguly, Tanmoy, Giannaras, Alexander, Kumar, Seema, Lewis, Timothy, Maounis, Florence, Nicolas, Jean-Marie, Mansley, Tamsin, Pasau, Patrick, Preda, Dorin, Stebbins, Karin, Volosov, Alexander, Zou, Dong

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Studies of palladium-catalyzed coupling reactions for preparation of hindered 3-arylpyrroles relevant to (-)-rhazinilam and its analogues von Ghosez, Léon, Franc, Cécile, Denonne, Frédéric, Cuisinier, Claire, Touillaux, Roland

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Discovery of a New Class of Non‐imidazole Oxazoline‐Based Histamine H 3 Receptor (H 3 R) Inverse Agonists von Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean‐Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent

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Discovery of new C3aR ligands. Part 2: Amino-piperidine derivatives von Denonne, Frédéric, Binet, Sophie, Burton, Maggi, Collart, Philippe, Defays, Sabine, Dipesa, Alan, Eckert, Maria, Giannaras, Alexander, Kumar, Seema, Levine, Beth, Nicolas, Jean-Marie, Pasau, Patrick, Pégurier, Cécile, Preda, Dorin, Van houtvin, Nathalie, Volosov, Andrew, Zou, Dong

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Towards the Synthesis of Azoacetylenes von Denonne, Frédéric, Seiler, Paul, Diederich, François

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Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor von Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean-Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent

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Lead Optimization of Thiazolo[5,4‐ c ]piperidines: 3‐Cyclobutoxy Linker as a Key Spacer for H 3 R Inverse Agonists von Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie

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Phenyl-oxazoles, a New Family of Inverse Agonists at the H3 Histamine Receptor von Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent

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A general synthesis of 2-formyl-3-arylpyrroles von Franc, Cécile, Denonne, Frédéric, Cuisinier, Claire, Ghose, Léon

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Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses von CELANIRE SYLVAIN, DENONNE FREDERIC

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Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses von Celanire, Sylvain, Denonne, Frederic

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COMPOSTO, COMPOSIÇÃO FARMACÊUTICA, E, INTERMEDIÁRIO SINTÉTICO von SYLVAIN CELANIRE, ANNE VALADE, FREDERIC DENONNE

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Compounds Comprising an Oxazole or Thiazole Moiety, Processes for Making Them, and Their Uses von CELANIRE SYLVAIN, DENONNE FREDERIC

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Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists von Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van Houtvin, Nathalie

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COMPOUNDS COMPRISING AN OXAZOLE OR THIAZOLE MOIETY, PROCESSES FOR MAKING THEM, AND THEIR USES von DENONNE, FREDERIC, CELANIRE, SYLVAIN

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Histamine H3 receptor ligands with a 3-cyclobutoxy motif: a novel and versatile constraint of the classical 3-propoxy linker von Wijtmans, Maikel, Denonne, Frédéric, Célanire, Sylvain, Gillard, Michel, Hulscher, Saskia, Delaunoy, Christel, Van houtvin, Nathalie, Bakker, Remko A., Defays, Sabine, Gérard, Julien, Grooters, Luc, Hubert, Delphine, Timmerman, Henk, Leurs, Rob, Talaga, Patrice, de Esch, Iwan J. P., Provins, Laurent

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