Pd- and Ni-Based Systems for the Catalytic Borylation of Aryl (Pseudo)halides with B2(OH)4 von Munteanu, Charissa, Spiller, Taylor E, Qiu, Jun, DelMonte, Albert J, Wisniewski, Steven R, Simmons, Eric M, Frantz, Doug E

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A Metal-Free Reductive N‑Alkylation of Indoles with Aldehydes von Clanton, Nicholas A, Spiller, Taylor E, Ortiz, Eliezer, Gao, Zhinong, Rodriguez-Poirier, Juan Manuel, DelMonte, Albert J, Frantz, Doug E

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Mechanistic Studies of a Pd-Catalyzed Direct Arylation En Route to Beclabuvir: Dual Role of a Tetramethylammonium Cation and an Unusual Turnover-Limiting Step von Hang, Chao, Ramirez, Antonio, Chan, Collin, Hsiao, Yi, DelMonte, Albert J, Simmons, Eric M

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Direct Lewis Acid Catalyzed Conversion of Enantioenriched N‑Acyloxazolidinones to Chiral Esters, Amides, and Acids von Stevens, Jason M, Parra-Rivera, Ana Cristina, Dixon, Darryl D, Beutner, Gregory L, DelMonte, Albert J, Frantz, Doug E, Janey, Jacob M, Paulson, James, Talley, Michael R

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Cerium(III) Chloride-Mediated Stereoselective Reduction of a 4‑Substituted Cyclohexanone Using NaBH4 von Maity, Prantik, Gujjar, Manjunath, Vellingiri, Raghukumar, Lakshminarasimhan, Thirumalai, DelMonte, Albert J, Young, Ian S, Eastgate, Martin D, Vaidyanathan, Rajappa

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Coupling-Condensation Strategy for the Convergent Synthesis of an Imidazole-Fused 2‑Aminoquinoline NLRP3 Agonist von Bi, Cong, Chadwick, James, Davies, Merrill L., DelMonte, Albert J., Geng, Peng, Glace, Andrew W., Green, Rebecca A., Gurak, John A., Haley, Matthew W., He, Brian L., Inankur, Bahar, Jamison, Christopher R., Joe, Candice L., Kolotuchin, Sergei, Lin, Dong, Lou, Sha, Nye, Jeffrey, Ortiz, Adrian, Purdum, Geoffrey E., Rosso, Victor W., Shah, Mansi, Simmons, Eric M., Stevens, Jason M., Strotman, Neil A., Tan, Yichen, Zhang, Ling

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The First Kilogram Synthesis of Beclabuvir, an HCV NS5B Polymerase Inhibitor von Bien, Jeffrey, Davulcu, Akin, DelMonte, Albert J, Fraunhoffer, Kenneth J, Gao, Zhinong, Hang, Chao, Hsiao, Yi, Hu, Wenhao, Katipally, Kishta, Littke, Adam, Pedro, Aghogho, Qiu, Yuping, Sandoval, Maria, Schild, Richard, Soltani, Michelle, Tedesco, Anthony, Vanyo, Dale, Vemishetti, Purushotham, Waltermire, Robert E

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Pd- and Ni-Based Systems for the Catalytic Borylation of Aryl (Pseudo)halides with B 2 (OH) 4 von Munteanu, Charissa, Spiller, Taylor E, Qiu, Jun, DelMonte, Albert J, Wisniewski, Steven R, Simmons, Eric M, Frantz, Doug E

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Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H2O2 von Beutner, Gregory L, Cohen, Benjamin M, DelMonte, Albert J, Dixon, Darryl D, Fraunhoffer, Kenneth J, Glace, Andrew W, Lo, Ehrlic, Stevens, Jason M, Vanyo, Dale, Wilbert, Christopher

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Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor von Fraunhoffer, Kenneth J, DelMonte, Albert J, Beutner, Gregory L, Bultman, Michael S, Camacho, Kathryn, Cohen, Benjamin, Dixon, Darryl D, Fan, Yu, Fanfair, Dayne, Freitag, Adam J, Glace, Andrew W, Gonzalez-Bobes, Francisco, Gujjar, Manjunath, Haley, Matthew W, Hickey, Matthew R, Ho, Jeanne, Iyer, Vidya, Maity, Prantik, Patel, Sunil, Rosso, Victor W, Schmidt, Michael A, Stevens, Jason M, Tan, Yichen, Wilbert, Christopher, Young, Ian S, Yu, Miao

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Safe Scale-up of an Oxygen-Releasing Cleavage of Evans Oxazolidinone with Hydrogen Peroxide von Glace, Andrew W, Cohen, Benjamin M, Dixon, Darryl D, Beutner, Gregory L, Vanyo, Dale, Akpinar, Fulya, Rosso, Victor, Fraunhoffer, Kenneth J, DelMonte, Albert J, Santana, Edgar, Wilbert, Christopher, Gallo, Frank, Bartels, William

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Reinvestigation of the Isotope Effects for the Claisen and Aromatic Claisen Rearrangements:  The Nature of the Claisen Transition States von Meyer, Matthew P, DelMonte, Albert J, Singleton, Daniel A

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Small Molecule Antagonist of Leukocyte Function Associated Antigen-1 (LFA-1): Structure−Activity Relationships Leading to the Identification of 6-((5S,9R)-9-(4-Cyanophenyl)-3-(3,5-... von Watterson, Scott H, Xiao, Zili, Dodd, Dharmpal S, Tortolani, David R, Vaccaro, Wayne, Potin, Dominique, Launay, Michele, Stetsko, Dawn K, Skala, Stacey, Davis, Patric M, Lee, Deborah, Yang, Xiaoxia, McIntyre, Kim W, Balimane, Praveen, Patel, Karishma, Yang, Zheng, Marathe, Punit, Kadiyala, Pathanjali, Tebben, Andrew J, Sheriff, Steven, Chang, ChiehYing Y, Ziemba, Theresa, Zhang, Huiping, Chen, Bang-Chi, DelMonte, Albert J, Aranibar, Nelly, McKinnon, Murray, Barrish, Joel C, Suchard, Suzanne J, Murali Dhar, T. G

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Experimental and Theoretical Kinetic Isotope Effects for Asymmetric Dihydroxylation. Evidence Supporting a Rate-Limiting “(3 + 2)” Cycloaddition von DelMonte, Albert J, Haller, Jan, Houk, K. N, Sharpless, K. Barry, Singleton, Daniel A, Strassner, Thomas, Thomas, Allen A

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The Process Development of Ravuconazole: An Efficient Multikilogram Scale Preparation of an Antifungal Agent von Pesti, Jaan, Chen, Chien-Kuang, Spangler, Lori, DelMonte, Albert J, Benoit, Serge, Berglund, Derek, Bien, Jeffrey, Brodfuehrer, Paul, Chan, Yeung, Corbett, Elisabeth, Costello, Carrie, DeMena, Paul, Discordia, Robert P, Doubleday, Wendel, Gao, Zhinong, Gingras, Stephane, Grosso, John, Haas, Oscar, Kacsur, David, Lai, Chiajen, Leung, Simon, Miller, Melanie, Muslehiddinoglu, Jale, Nguyen, Nina, Qiu, Jun, Olzog, Martina, Reiff, Emily, Thoraval, Dominique, Totleben, Michael, Vanyo, Dale, Vemishetti, Purushotham, Wasylak, John, Wei, Chenkou

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Kilogram Synthesis of a Selective Serotonin Reuptake Inhibitor von Anthes, Robert, Bello, Osagie, Benoit, Serge, Chen, Chien-Kuang, Corbett, Elisabeth, Corbett, Richard M, DelMonte, Albert J, Gingras, Stephane, Livingston, Robert, Sausker, Justin, Soumeillant, Maxime

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Kilogram Synthesis of a Second-Generation LFA-1/ICAM Inhibitor von DelMonte, Albert J, Fan, Yu, Girard, Kevin P, Jones, Gregory S, Waltermire, Robert E, Rosso, Victor, Wang, Xuebao

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An Improved Synthesis of a Selective Serotonin Reuptake Inhibitor von Anthes, Robert, Benoit, Serge, Chen, Chien-Kuang, Corbett, Elisabeth A, Corbett, Richard M, DelMonte, Albert J, Gingras, Stephane, Livingston, Robert C, Pendri, Yadagiri, Sausker, Justin, Soumeillant, Maxime

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Kilogram Synthesis of a LFA-1/ICAM Inhibitor von DelMonte, Albert J, Waltermire, Robert E, Fan, Yu, McLeod, Douglas D, Gao, Zhinong, Gesenberg, Kirsten D, Girard, Kevin P, Rosingana, Miguel, Wang, Xuebao, Kuehne-Willmore, Jennifer, Braem, Alan D, Castoro, John A

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Development of a Scalable Negishi Cross-Coupling Process for the Preparation of 2-Chloro-5-(1-(tetrahydro-2 H -pyran-2-yl)-1 H -pyrazol-5-yl)aniline von Joe, Candice L., Inankur, Bahar, Chadwick, James, Lou, Sha, Nye, Jeffrey, Strotman, Neil A., DelMonte, Albert J.

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