Stereoselective amination of chiral enolates. A new approach to the asymmetric synthesis of .alpha.-hydrazino and .alpha.-amino acid derivatives von Evans, David A, Britton, Thomas C, Dorow, Roberta L, Dellaria, Joseph F

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A synthesis of protected aminoalkyl epoxides from .alpha.-amino acids von Luly, Jay R, Dellaria, Joseph F, Plattner, Jacob J, Soderquist, Jeffrey L, Yi, Nwe

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Enantioselective synthesis of .alpha.-amino acid derivatives via the stereoselective alkylation of a homochiral glycine enolate synthon von Dellaria, Joseph F, Santarsiero, Bernard D

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Nonsteroidal Anti-Inflammatory Drugs as Scaffolds for the Design of 5-Lipoxygenase Inhibitors von Kolasa, Teodozyj, Brooks, Clint D. W, Rodriques, Karen E, Summers, James B, Dellaria, Joseph F, Hulkower, Keren I, Bouska, Jennifer, Bell, Randy L, Carter, George W

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Biaryl Ether Retrohydroxamates as Potent, Long-lived, Orally Bioavailable MMP Inhibitors von Michaelides, Michael R., Dellaria, Joseph F., Gong, Jane, Holms, James H., Bouska, Jennifer J., Stacey, Jamie, Wada, Carol K., Heyman, H.Robin, Curtin, Michael L., Guo, Yan, Goodfellow, Carole L., Elmore, Ildiko B., Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Morgan, Douglas W., Davidsen, Steven K.

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Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties von Bruncko, Milan, McClellan, William J., Wendt, Michael D., Sauer, Daryl R., Geyer, Andrew, Dalton, Christopher R., Kaminski, Michele A., Weitzberg, Moshe, Gong, Jane, Dellaria, Joseph F., Mantei, Robert, Zhao, Xumiao, Nienaber, Vicki L., Stewart, Kent, Klinghofer, Vered, Bouska, Jennifer, Rockway, Todd W., Giranda, Vincent L.

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Efficient and versatile synthesis of dipeptide isosteres containing .gamma.- or .delta.-lactams von Zydowsky, Thomas M, Dellaria, Joseph F, Nellans, Hugh N

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Alkyl nitrite-metal halide deamination reactions. 2. Substitutive deamination of arylamines by alkyl nitrites and copper(II) halides. A direct and remarkably efficient conversion o... von Doyle, Michael P, Siegfried, Bernard, Dellaria, Joseph F

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Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770 von Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.

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The enantio- and diastereoselective synthesis of the first phospho-statine derivative von Dellaria, Joseph F, Maki, Robert G

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New inhibitors of renin that contain novel phosphostatine Leu-Val replacements von Dellaria, Joseph F, Maki, Robert G, Stein, Herman H, Cohen, Jerome, Whittern, David, Marsh, Kennan, Hoffman, Daniel J, Plattner, Jacob J, Perun, Thomas J

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Alkyl nitrite-metal halide deamination reactions. 3. Arylation of olefinic compounds in the deamination of arylamines by alkyl nitrites and copper(II) halides. A convenient and eff... von Doyle, Michael P, Siegfried, Bernard, Elliott, Robert C, Dellaria, Joseph F

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Potent, low molecular weight renin inhibitors containing a C-terminal heterocycle: hydrogen bonding at the active site von Rosenberg, Saul H, Dellaria, Joseph F, Kempf, Dale J, Hutchins, Charles W, Woods, Keith W, Maki, Robert G, De Lara, Ed, Spina, Kenneth P, Stein, Herman H

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New inhibitors of human renin that contain novel Leu-Val replacements. Examination of the P1 site von Luly, Jay R, Bolis, Giorgio, BaMaung, Nwe, Soderquist, Jeff, Dellaria, Joseph F, Stein, Herman, Cohen, Jerome, Perun, Thomas J, Greer, Jonathan, Plattner, Jacob J

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Optimization and in vivo evaluations of a series of small, potent, and specific renin inhibitors containing a novel Leu-Val replacement von Dellaria, Joseph F, Maki, Robert G, Bopp, Barbara A, Cohen, Jerome, Kleinert, Hollis D, Luly, Jay R, Merits, Ilmar, Plattner, Jacob J, Stein, Herman H

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Reductive deamination of arylamines by alkyl nitrites in N,N-dimethylformamide. A direct conversion of arylamines to aromatic hydrocarbons von Doyle, Michael P., Dellaria, Joseph F., Siegfried, Bernard, Bishop, Stephen W.

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Patent Update: Anti-Inflammatory Patents Highlights from the First Half of 1992 von Luly, Jay R, Dellaria, Joseph F, Davidsen, Steven K

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Two syntheses of dl-aplysistatin von Hoye, Thomas R, Caruso, Andrew J, Dellaria, Joseph F, Kurth, Mark J

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The asymmetric synthesis of α-amino and α-hydrazino acid derivatives via the stereoselective amination of chiral enolates with azodicarboxylate esters von Evans, David A., Britton, Thomas C., Dorow, Roberta L., Dellaria, Joseph F.

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The Facile and Efficient Preparation of Phenolic and Thiol Esters von Dellaria, Joseph F., Nordeen, Carl, Swett, Leo R.

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