GAL-021, a new intravenous BKCa-channel blocker, is well tolerated and stimulates ventilation in healthy volunteers von McLeod, J.F., Leempoels, J.M., Peng, S.X., Dax, S.L., Myers, L.J., Golder, F.J.

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Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloi... von Swanson, Devin M, Dubin, Adrienne E, Shah, Chandra, Nasser, Nadia, Chang, Leon, Dax, Scott L, Jetter, Michele, Breitenbucher, J. Guy, Liu, Changlu, Mazur, Curt, Lord, Brian, Gonzales, Lisa, Hoey, Kenway, Rizzolio, Michele, Bogenstaetter, Michael, Codd, Ellen E, Lee, Doo H, Zhang, Sui-Po, Chaplan, Sandra R, Carruthers, Nicholas I

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Quinolone antibacterials: a hydroxymethylation-intramolecular cyclization route to pyrido[3,2,1-ij]-1,3,4-benzoxadiazines von Dax, S. L, Wei, C. C

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α-Substituted N-(Sulfonamido)alkyl-β-aminotetralins:  Potent and Selective Neuropeptide Y Y5 Receptor Antagonists von Youngman, Mark A, McNally, James J, Lovenberg, Timothy W, Reitz, Allen B, Willard, Nicole M, Nepomuceno, Diane H, Wilson, Sandy J, Crooke, Jeffrey J, Rosenthal, Daniel, Vaidya, Anil H, Dax, Scott L

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Dual-action penems and carbapenems von Corraz, Alfred J, Dax, Scott L, Dunlap, Norma K, Georgopapadakou, Nafsika H, Keith, Dennis D, Pruess, David L, Rossman, Pamela L, Then, Rudolf, Unowsky, Joel, Wei, Chung Chen

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Aminopyrazoles with high affinity for the human neuropeptide Y5 receptor von Kordik, Cheryl P, Luo, Chi, Zanoni, Brian C, Dax, Scott L, McNally, James J, Lovenberg, Timothy W, Wilson, Sandy J, Reitz, Allen B

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N-(sulfonamido)alkyl[tetrahydro-1H-benzo[e]indol-2-yl]amines : Potent antagonists of human neuropeptide Y Y5 receptor von MCNALLY, J. J, YOUNGMAN, M. A, LOVENBERG, T. W, NEPOMUCENO, D. H, WILSON, S. J, DAX, S. L

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Synthesis and in vitro evaluation of a novel iodinated resiniferatoxin derivative that is an agonist at the human vanilloid VR1 receptor von MCDONNELL, Mark E, ZHANG, Sui-Po, DUBIN, Adrienne E, DAX, Scott L

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Benzo[d]imidazole Transient Receptor Potential Vanilloid 1 Antagonists for the Treatment of Pain: Discovery of trans-2-(2-{2-[2-(4-Trifluoromethyl-phenyl)-vinyl]‑1H‑benzimidazol-5-... von Parsons, William H, Calvo, Raul R, Cheung, Wing, Lee, Yu-Kai, Patel, Sharmila, Liu, Jian, Youngman, Mark A, Dax, Scott L, Stone, Dennis, Qin, Ning, Hutchinson, Tasha, Lubin, Mary Lou, Zhang, Sui-Po, Finley, Michael, Liu, Yi, Brandt, Michael R, Flores, Christopher M, Player, Mark R

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Indoloquinones from azomethine ylides via the 4-oxazoline route von Vedejs, Edwin, Dax, Scott L.

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Synthesis and mechanistic studies of a ‘tetrazole-tethered” cephalosporin-quinolone hybrid von Dax, S.L., Pruess, D.L., Rossman, P.L., Wei, C.-c.

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Mannich reactions of resin-bound substrates: 2. A versatile three-component solid-phase organic synthesis methodology von McNally, James J., Youngman, Mark A., Dax, Scott L.

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N-Isoquinolin-5-yl- N′-aralkyl-urea and -amide antagonists of human vanilloid receptor 1 von Jetter, Michele C., Youngman, Mark A., McNally, James J., Zhang, Sui-Po, Dubin, Adrienne E., Nasser, Nadia, Dax, Scott L.

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N-Acylated α-(3-pyridylmethyl)-β-aminotetralin antagonists of the human neuropeptide Y Y5 receptor von McNally, James J, Youngman, Mark A, Lovenberg, Timothy W, Nepomuceno, Diane, Wilson, Sandy, Dax, Scott L

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Mannich Reactions of a Resin-Bound Terminal Alkyne von Youngman, Mark A., Dax, Scott L.

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7-Hydroxynaphthalen-1-yl-urea and -amide antagonists of human vanilloid receptor 1 von McDonnell, Mark E., Zhang, Sui-Po, Nasser, Nadia, Dubin, Adrienne E., Dax, Scott L.

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Parallel methods for the preparation and SAR exploration of N-ethyl-4-[(8-alkyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-aryl-methyl]-benzamides, powerful mu and delta opioid agonists von Coats, Steven J., Schulz, Mark J., Carson, John R., Codd, Ellen E., Hlasta, Dennis J., Pitis, Philip M., Stone, Dennis J., Zhang, Sui-Po, Colburn, Ray W., Dax, Scott L.

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N-acylated alpha-(3-pyridylmethyl)-beta-aminotetralin antagoinists of the human neuropeptide Y Y5 receptor von McNally, J J, Youngman, M A, Lovenberg, T W, Nepomuceno, D, Wilson, S, Dax, S L

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Design and synthesis of novel pyrrolidine-containing bradykinin antagonists von Lee, Jung, Reynolds, Charles, Jetter, Michele C, Youngman, Mark A, Hlasta, Dennis J, Dax, Scott L, Stone, Dennis J, Zhang, Sui-Po, Codd, Ellen E

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Synthesis and structure–Activity relationships of aroylpyrrole alkylamide bradykinin (B 2) antagonists von Youngman, Mark A., Carson, John R., Lee, Jung S., Dax, Scott L., Zhang, Sui-Po, Colburn, Ray W., Stone, Dennis J., Codd, Ellen E., Jetter, Michele C.

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