Applications of Fluorine in Medicinal Chemistry von Gillis, Eric P, Eastman, Kyle J, Hill, Matthew D, Donnelly, David J, Meanwell, Nicholas A

Volltext

Nucleophilic (Radio)Fluorination of Redox-Active Esters via Radical-Polar Crossover Enabled by Photoredox Catalysis von Webb, Eric W, Park, John B, Cole, Erin L, Donnelly, David J, Bonacorsi, Samuel J, Ewing, William R, Doyle, Abigail G

Volltext

Small Molecule PET Tracers in Drug Discovery von Donnelly, David J.

Volltext

Radiosynthesis and preclinical PET evaluation of 89Zr-nivolumab (BMS-936558) in healthy non-human primates von Cole, Erin L., Kim, Joonyoung, Donnelly, David J., Smith, R. Adam, Cohen, Daniel, Lafont, Virginie, Morin, Paul E., Huang, Richard Y.-C., Chow, Patrick L., Hayes, Wendy, Bonacorsi, Samuel

Volltext

Heteroatom Substitution Induced Changes in Excited-State Photophysics and Singlet Oxygen Generation in Chalcogenoxanthylium Dyes:  Effect of Sulfur and Selenium Substitutions von Ohulchanskyy, Tymish Y, Donnelly, David J, Detty, Michael R, Prasad, Paras N

Volltext

Synthesis and Preclinical Evaluation of a 68Ga-Labeled Adnectin, 68Ga-BMS-986192, as a PET Agent for Imaging PD-L1 Expression von Robu, Stephanie, Richter, Antonia, Gosmann, Dario, Seidl, Christof, Leung, David, Hayes, Wendy, Cohen, Daniel, Morin, Paul, Donnelly, David J., Lipovsek, Dasa, Bonacorsi, Samuel J., Smith, Adam, Steiger, Katja, Aulehner, Christina, Krackhardt, Angela M., Weber, Wolfgang A.

Volltext

Chemoselective Methionine Bioconjugation: Site-Selective Fluorine-18 Labeling of Proteins and Peptides von Lin, Daniel, Wallace, Michael, Allentoff, Alban J, Donnelly, David J, Gomes, Erin, Voronin, Kim, Gong, Sharon, Huang, Richard Y.-C, Kim, Ho, Caceres-Cortes, Janet, Bonacorsi, Samuel

Volltext

The discovery and evaluation of [18F]BMS-986229, a novel macrocyclic peptide PET radioligand for the measurement of PD-L1 expression and in-vivo PD-L1 target engagement von Donnelly, David J., Kim, Joonyoung, Tran, Tritin, Scola, Paul M., Tenney, Daniel, Pena, Adrienne, Petrone, Thomas, Zhang, Yunhui, Boy, Kenneth M., Poss, Michael A., Cole, Erin L., Soars, Matthew G., Johnson, Benjamin M., Cohen, Daniel, Batalla, Daniel, Chow, Patrick L., Shorts, Andrea Olga, Du, Shuyan, Meanwell, Nicholas A., Bonacorsi, Samuel J.

Volltext

Synthesis and Preclinical Evaluation of a 68 Ga-Labeled Adnectin, 68 Ga-BMS-986192, as a PET Agent for Imaging PD-L1 Expression von Robu, Stephanie, Richter, Antonia, Gosmann, Dario, Seidl, Christof, Leung, David, Hayes, Wendy, Cohen, Daniel, Morin, Paul, Donnelly, David J, Lipovšek, Daša, Bonacorsi, Samuel J, Smith, Adam, Steiger, Katja, Aulehner, Christina, Krackhardt, Angela M, Weber, Wolfgang A

Volltext

Synthesis of Diverse (11)C-Labeled PET Radiotracers via Direct Incorporation of [(11)C]CO2 von Mossine, Andrew V, Brooks, Allen F, Jackson, Isaac M, Quesada, Carole A, Sherman, Phillip, Cole, Erin L, Donnelly, David J, Scott, Peter J H, Shao, Xia

Volltext

Development, Characterization, and Radiation Dosimetry Studies of 18F-BMS-986229, a 18F-Labeled PD-L1 Macrocyclic Peptide PET Tracer von Kim, Joonyoung, Donnelly, David J., Tran, Tritin, Pena, Adrienne, Shorts, Andrea Olga, Petrone, Thomas V., Zhang, Yunhui, Boy, Kenneth M., Scola, Paul M., Tenney, Daniel J., Poss, Michael A., Soars, Matthew G., Bonacorsi, Samuel J., Cole, Erin L., Grootendorst, Diederik J., Chow, Patrick L., Meanwell, Nicholas A., Du, Shuyan

Volltext

Transcriptome-wide comparison of sequence variation in divergent ecotypes of kokanee salmon von Lemay, Matthew A, Donnelly, David J, Russello, Michael A

Volltext

Radiosynthesis of [ 11 C]Ibrutinib via Pd-Mediated [ 11 C]CO Carbonylation: Preliminary PET Imaging in Experimental Autoimmune Encephalomyelitis Mice von Lindberg, Anton, Boyle, Amanda J, Tong, Junchao, Harkness, Michael B, Garcia, Armando, Tran, Tritin, Zhai, Dongxu, Liu, Fang, Donnelly, David J, Vasdev, Neil

Volltext

Synthesis and Biologic Evaluation of a Novel 18 F-Labeled Adnectin as a PET Radioligand for Imaging PD-L1 Expression von Donnelly, David J, Smith, R Adam, Morin, Paul, Lipovšek, Daša, Gokemeijer, Jochem, Cohen, Daniel, Lafont, Virginie, Tran, Tritin, Cole, Erin L, Wright, Martin, Kim, Joonyoung, Pena, Adrienne, Kukral, Daniel, Dischino, Douglas D, Chow, Patrick, Gan, Jinping, Adelakun, Olufemi, Wang, Xi-Tao, Cao, Kai, Leung, David, Bonacorsi, Jr, Samuel J, Hayes, Wendy

Volltext

Evaluation of the Lysophosphatidic Acid Receptor Type 1 Radioligand 11 C-BMT-136088 for Lung Imaging in Rhesus Monkeys von Gallezot, Jean-Dominique, Nabulsi, Nabeel B, Holden, Daniel, Lin, Shu-Fei, Labaree, David, Ropchan, Jim, Najafzadeh, Soheila, Donnelly, David J, Cao, Kai, Bonacorsi, Samuel, Seiders, Jon, Roppe, Jeffrey, Hayes, Wendy, Huang, Yiyun, Du, Shuyan, Carson, Richard E

Volltext

Synthesis of Radiopharmaceuticals via “In-Loop” 11C-Carbonylation as Exemplified by the Radiolabeling of Inhibitors of Bruton's Tyrosine Kinase von Donnelly, David J., Preshlock, Sean, Kaur, Tanpreet, Tran, Tritin, Wilson, Thomas C., Mhanna, Karim, Henderson, Bradford D., Batalla, Daniel, Scott, Peter J. H., Shao, Xia

Volltext

Synthesis of Diverse 11C‑Labeled PET Radiotracers via Direct Incorporation of [11C]CO2 von Mossine, Andrew V, Brooks, Allen F, Jackson, Isaac M, Quesada, Carole A, Sherman, Phillip, Cole, Erin L, Donnelly, David J, Scott, Peter J. H, Shao, Xia

Volltext

Synthesis, properties, and photodynamic properties in vitro of heavy-chalcogen analogues of tetramethylrosamine von Detty, Michael R, Prasad, Paras N, Donnelly, David J, Ohulchanskyy, Tymish, Gibson, Scott L, Hilf, Russell

Volltext

Stimulation of P-Glycoprotein ATPase by Analogues of Tetramethylrosamine:  Coupling of Drug Binding at the “R” Site to the ATP Hydrolysis Transition State von Tombline, Gregory, Donnelly, David J, Holt, Jason J, You, Youngjae, Ye, Mao, Gannon, Michael K, Nygren, Cara L, Detty, Michael R

Volltext

Chalcogenoxanthylium photosensitizers for the photodynamic purging of blood-borne viral and bacterial pathogens von Wagner, Stephen J., Skripchenko, Andrey, Donnelly, David J., Ramaswamy, Krishna, Detty, Michael R.

Volltext