Alternative oxidase inhibitors: Mitochondrion‐targeting as a strategy for new drugs against pathogenic parasites and fungi von Ebiloma, Godwin U., Balogun, Emmanuel O., Cueto‐Díaz, Eduardo J., Koning, Harry P., Dardonville, Christophe

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Crystal structure of the HMGA AT-hook 1 domain bound to the minor groove of AT-rich DNA and inhibition by antikinetoplastid drugs von Nué-Martinez, J. Jonathan, Maturana, Marta, Lagartera, Laura, Rodríguez-Gutiérrez, Juan-Antonio, Boer, Roeland, Campos, J. Lourdes, Saperas, Núria, Dardonville, Christophe

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New Benzophenone-Derived Bisphosphonium Salts as Leishmanicidal Leads Targeting Mitochondria through Inhibition of Respiratory Complex II von Luque-Ortega, J. Román, Reuther, Peter, Rivas, Luis, Dardonville, Christophe

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Conjugates of 2,4-Dihydroxybenzoate and Salicylhydroxamate and Lipocations Display Potent Antiparasite Effects by Efficiently Targeting the Trypanosoma brucei and Trypanosoma congo... von Fueyo González, Francisco José, Ebiloma, Godwin U, Izquierdo García, Carolina, Bruggeman, Victor, Sánchez Villamañán, José María, Donachie, Anne, Balogun, Emmanuel Oluwadare, Inaoka, Daniel Ken, Shiba, Tomoo, Harada, Shigeharu, Kita, Kiyoshi, de Koning, Harry P, Dardonville, Christophe

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Antiprotozoal Activity and DNA Binding of Dicationic Acridones von Montalvo-Quirós, Sandra, Taladriz-Sender, Andrea, Kaiser, Marcel, Dardonville, Christophe

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Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei von Alghamdi, Ali H., Munday, Jane C., Campagnaro, Gustavo Daniel, Gurvic, Dominik, Svensson, Fredrik, Okpara, Chinyere E., Kumar, Arvind, Quintana, Juan, Abril, Maria Esther Martin, Milic, Patrik, Watson, Laura, Paape, Daniel, Settimo, Luca, Dimitriou, Anna, Wielinska, Joanna, Smart, Graeme, Anderson, Laura F., Woodley, Christopher M., Kelly, Siu Pui Ying, Ibrahim, Hasan M. S., Hulpia, Fabian, Al-Salabi, Mohammed, Eze, Anthonius A., Sprenger, Teresa, Teka, Ibrahim A., Gudin, Simon, Weyand, Simone, Field, Mark, Dardonville, Christophe, Tidwell, Richard R., Carrington, Mark, O'Neill, Paul, Boykin, David W., Zachariae, Ulrich, De Koning, Harry P.

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Automated techniques in pKa determination: Low, medium and high-throughput screening methods von Dardonville, Christophe

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Trypanocidal action of bisphosphonium salts through a mitochondrial target in bloodstream form Trypanosoma brucei von Alkhaldi, Abdulsalam A.M., Martinek, Jan, Panicucci, Brian, Dardonville, Christophe, Zíková, Alena, de Koning, Harry P.

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Discovery of nitroheterocycles active against African trypanosomes. In vitro screening and preliminary SAR studies von Arán, Vicente J., Kaiser, Marcel, Dardonville, Christophe

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SAR of 4‑Alkoxybenzoic Acid Inhibitors of the Trypanosome Alternative Oxidase von Meco-Navas, Alejandro, Ebiloma, Godwin U, Martín-Domínguez, Ana, Martínez-Benayas, Irene, Cueto-Díaz, Eduardo J, Alhejely, Amani Saud, Balogun, Emmanuel O, Saito, Machi, Matsui, Miho, Arai, Natsumi, Shiba, Tomoo, Harada, Shigeharu, de Koning, Harry P, Dardonville, Christophe

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Aqueous pKa prediction for tautomerizable compounds using equilibrium bond lengths von Caine, Beth A., Bronzato, Maddalena, Fraser, Torquil, Kidley, Nathan, Dardonville, Christophe, Popelier, Paul L. A.

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Prediction of Aqueous pKa Values for Guanidine-Containing Compounds Using Ab Initio Gas-Phase Equilibrium Bond Lengths von Caine, Beth A., Dardonville, Christophe, Popelier, Paul L. A.

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SAR Studies of Diphenyl Cationic Trypanocides: Superior Activity of Phosphonium over Ammonium Salts von Dardonville, Christophe, Alkhaldi, Abdulsalam A. M, De Koning, Harry P

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Automated techniques in pK a determination: Low, medium and high-throughput screening methods von Dardonville, Christophe

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Antiprotozoal Activity of 1-Phenethyl-4-Aminopiperidine Derivatives von DARDONVILLE, Christophe, FERNANDEZ-FERNANDEZ, Cristina, GIBBONS, Sarah-Louise, JAGEROVIC, Nadine, NIETO, Lidia, RYAN, Gary, KAISER, Marcel, BRUN, Reto

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Methyl N-(tert-butoxycarbonyl)pyridine-2-carbimidothioate: A new reagent for the synthesis of N-phenylpyridinecarboxamidine (“arylimidamide”) DNA-minor groove binders from poorly n... von Nué-Martinez, J. Jonathan, Cisneros, David, Dardonville, Christophe

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Imidazoline binding sites and their ligands: An overview of the different chemical structures von Dardonville, Christophe, Rozas, Isabel

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Observation of diastereotopic signals in (15) N NMR spectroscopy von Alkorta, Ibon, Dardonville, Christophe, Elguero, José

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Observation of Diastereotopic Signals in 15 N NMR Spectroscopy von Alkorta, Ibon, Dardonville, Christophe, Elguero, José

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Observation of Diastereotopic Signals in 15NNMR Spectroscopy von Alkorta, Ibon, Dardonville, Christophe, Elguero, José

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