Discovery of Potent Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors Using Fragment-Based Methods and Structure-Based Design von Friberg, Anders, Vigil, Dominico, Zhao, Bin, Daniels, R. Nathan, Burke, Jason P, Garcia-Barrantes, Pedro M, Camper, DeMarco, Chauder, Brian A, Lee, Taekyu, Olejniczak, Edward T, Fesik, Stephen W

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Approach for targeting Ras with small molecules that activate SOS-mediated nucleotide exchange von Burns, Michael C., Qi Sun, Daniels, R. Nathan, Camper, DeMarco, Kennedy, J. Phillip, Phan, Jason, Olejniczak, Edward T., Lee, Taekyu, Waterson, Alex G., Rossanese, Olivia W., Fesik, Stephen W.

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Cytochromes P450 1A2 and 3A4 Catalyze the Metabolic Activation of Sunitinib von Amaya, Gracia M, Durandis, Rebecca, Bourgeois, David S, Perkins, James A, Abouda, Arsany A, Wines, Kahari J, Mohamud, Mohamed, Starks, Samuel A, Daniels, R. Nathan, Jackson, Klarissa D

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Classics in Chemical Neuroscience: Levodopa von Whitfield, A. Connor, Moore, Ben T, Daniels, R. Nathan

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Classics in Chemical Neuroscience: Amitriptyline von McClure, Elliot W, Daniels, R. Nathan

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DARK Classics in Chemical Neuroscience: Psilocybin von Geiger, Haden A, Wurst, Madeline G, Daniels, R. Nathan

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Classics in Chemical Neuroscience: Dextromethorphan (DXM) von McClure, Elliot W., Daniels, R. Nathan

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Synthesis and SAR of analogues of the M1 allosteric agonist TBPB. Part I: Exploration of alternative benzyl and privileged structure moieties von Bridges, Thomas M., Brady, Ashley E., Phillip Kennedy, J., Nathan Daniels, R., Miller, Nicole R., Kim, Kwango, Breininger, Micah L., Gentry, Patrick R., Brogan, John T., Jones, Carrie K., Jeffrey Conn, P., Lindsley, Craig W.

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Classics in Chemical Neuroscience: Pramipexole von Wilson, Sean M, Wurst, Madeline G, Whatley, Michael F, Daniels, R. Nathan

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In Vivo Structure−Activity Relationship Study of Dorsomorphin Analogues Identifies Selective VEGF and BMP Inhibitors von Hao, Jijun, Ho, Joshua N, Lewis, Jana A, Karim, Kaleh A, Daniels, R. Nathan, Gentry, Patrick R, Hopkins, Corey R, Lindsley, Craig W, Hong, Charles C

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Total Synthesis of Ciliatamides A-C: Stereochemical Revision and the Natural Product-Guided Synthesis of Unnatural Analogs von Lewis, Jana A, Daniels, R. Nathan, Lindsley, Craig W

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Discovery of Aminopiperidine Indoles That Activate the Guanine Nucleotide Exchange Factor SOS1 and Modulate RAS Signaling von Abbott, Jason R, Hodges, Timothy R, Daniels, R. Nathan, Patel, Pratiq A, Kennedy, J. Phillip, Howes, Jennifer E, Akan, Denis T, Burns, Michael C, Sai, Jiqing, Sobolik, Tammy, Beesetty, Yugandhar, Lee, Taekyu, Rossanese, Olivia W, Phan, Jason, Waterson, Alex G, Fesik, Stephen W

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Total synthesis of polemannones B and C von Fadeyi, Olugbeminiyi O., Nathan Daniels, R., DeGuire, Sean M., Lindsley, Craig W.

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Corrigendum to “Novel GlyT1 inhibitor chemotypes by scaffold hopping. Part 2: Development of a [3.3.0]-based series and other piperidine bioisosteres” [Bioorg. Med. Chem. Lett. 24... von Sheffler, Douglas J., Nedelcovych, Michael T., Williams, Richard, Turner, Stephen C., Duerk, Brittany B., Robbins, Megan R., Jadhav, Sataya B., Niswender, Colleen M., Jones, Carrie K., Conn, P. Jeffrey, Nathan Daniels, R., Lindsley, Craig W.

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A New Catalytic Cu(II)/Sparteine Oxidant System for β,β-Phenolic Couplings of Styrenyl Phenols: Synthesis of Carpanone and Unnatural Analogs von Daniels, R. Nathan, Fadeyi, Olugbeminiyi O, Lindsley, Craig W

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Novel GlyT1 inhibitor chemotypes by scaffold hopping. Part 2: development of a [3.3.0]-based series and other piperidine bioisosteres von Sheffler, Douglas J, Nedelcovych, Michael T, Williams, Richard, Turner, Stephen C, Duerk, Brittany B, Robbins, Megan R, Jadhav, Sataya B, Niswender, Colleen M, Jones, Carrie K, Conn, P Jeffrey, Daniels, R Nathan, Lindsley, Craig W

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Synthesis and SAR of analogs of the M1 allosteric agonist TBPB. Part II: Amides, sulfonamides and ureas—The effect of capping the distal basic piperidine nitrogen von Miller, Nicole R., Daniels, R. Nathan, Bridges, Thomas M., Brady, Ashley E., Conn, P. Jeffrey, Lindsley, Craig W.

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Progress toward the Total Synthesis of Lucentamycin A: Total Synthesis and Biological Evaluation of 8-epi-Lucentamycin A von Daniels, R. Nathan, Melancon, Bruce J, Wang, Emily A, Crews, Brenda C, Marnett, Lawrence J, Sulikowski, Gary A, Lindsley, Craig W

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Synthesis and SAR of N-(4-(4-alklylpiperazin-1-yl)phenyl)benzamides as muscarinic acetylcholine receptor subtype 1 (M 1) anatgonists von Miller, Nicole R., Daniels, R. Nathan, Lee, David, Conn, P. Jeffrey, Lindsley, Craig W.

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Abstract 4911: Metabolic activation of sunitinib: Implications for sunitinib-induced toxicities von Jackson, Klarissa D., Amaya, Gracia M., Durandis, Rebecca, Wines, Kahari J., Abouda, Arsany A., Starks, Samuel A., Daniels, R. Nathan

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