C–H activation reactions as useful tools for medicinal chemists von Caro-Diaz, Eduardo J.E., Urbano, Mariangela, Buzard, Daniel J., Jones, Robert M.

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GPR119 agonists for the treatment of type 2 diabetes von Jones, Robert M, Leonard, James N, Buzard, Daniel J, Lehmann, Juerg

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Therapeutic Utility of Cannabinoid Receptor Type 2 (CB2) Selective Agonists von Han, Sangdon, Thatte, Jayant, Buzard, Daniel J, Jones, Robert M

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Identification of 2-arylbenzimidazoles as potent human histamine H4 receptor ligands von LEE-DUTRA, Alice, ARIENTI, Kristen L, BREITENBUCHER, J. Guy, BUZARD, Daniel J, HACK, Michael D, KHATUYA, Haripada, DESAI, Pragnya J, NGUYEN, Steven, THURMOND, Robin L, KARLSSON, Lars, EDWARDS, James P

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Recent progress in the development of selective S1P1 receptor agonists for the treatment of inflammatory and autoimmune disorders von Buzard, Daniel J, Thatte, Jayant, Lerner, Michael, Edwards, Jeffrey, Jones, Robert M

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Kinetics of 5-HT2B receptor signaling: profound agonist-dependent effects on signaling onset and duration von Unett, David J, Gatlin, Joel, Anthony, Todd L, Buzard, Daniel J, Chang, Steve, Chen, Chuan, Chen, Xiaohua, Dang, Huong T-M, Frazer, John, Le, Minh K, Sadeque, Abu J M, Xing, Charles, Gaidarov, Ibragim

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Design and synthesis of new tricyclic indoles as potent modulators of the S1P1 receptor von Buzard, Daniel J., Schrader, Thomas O., Zhu, Xiuwen, Lehmann, Juerg, Johnson, Ben, Kasem, Michelle, Kim, Sun Hee, Kawasaki, Andrew, Lopez, Luis, Moody, Jeanne, Han, Sangdon, Gao, Yinghong, Edwards, Jeff, Barden, Jeremy, Thatte, Jayant, Gatlin, Joel, Jones, Robert M.

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Discovery of APD334: Design of a Clinical Stage Functional Antagonist of the Sphingosine-1-phosphate‑1 Receptor von Buzard, Daniel J, Kim, Sun Hee, Lopez, Luis, Kawasaki, Andrew, Zhu, Xiuwen, Moody, Jeanne, Thoresen, Lars, Calderon, Imelda, Ullman, Brett, Han, Sangdon, Lehmann, Juerg, Gharbaoui, Tawfik, Sengupta, Dipanjan, Calvano, Lorene, Montalban, Antonio Garrido, Ma, You-An, Sage, Carleton, Gao, Yinghong, Semple, Graeme, Edwards, Jeff, Barden, Jeremy, Morgan, Michael, Chen, Weichao, Usmani, Khawja, Chen, Chuan, Sadeque, Abu, Christopher, Ronald J, Thatte, Jayant, Fu, Lixia, Solomon, Michelle, Mills, David, Whelan, Kevin, Al-Shamma, Hussien, Gatlin, Joel, Le, Minh, Gaidarov, Ibragim, Anthony, Todd, Unett, David J, Blackburn, Anthony, Rueter, Jaimie, Stirn, Scott, Behan, Dominic P, Jones, Robert M

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An Efficient Scale-Up Process for the Preparation of the APD334 Precursor 4‑Chloromethyl-1-cyclopentyl-2-(trifluoromethyl)benzene von Sengupta, Dipanjan, Gharbaoui, Tawfik, Krishnan, Ashwin, Buzard, Daniel J, Jones, Robert M, Ma, You-An, Burda, Robert, Garrido Montalban, Antonio, Semple, Graeme

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Discovery of a novel trans-1,4-dioxycyclohexane GPR119 agonist series von Han, Sangdon, Narayanan, Sanju, Kim, Sun Hee, Calderon, Imelda, Zhu, Xiuwen, Kawasaki, Andrew, Yue, Dawei, Lehmann, Juerg, Wong, Amy, Buzard, Daniel J., Semple, Graeme, Carroll, Chris, Chu, Zhi-Liang, Al-Sharmma, Hussein, Shu, Hsin-Hui, Tung, Shiu-Feng, Unett, David J., Behan, Dominic P., Yoon, Woo Hyun, Morgan, Michael, Usmani, Khawja A., Chen, Chuan, Sadeque, Abu, Leonard, James N., Jones, Robert M.

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Discovery and optimization of 5-fluoro-4,6-dialkoxypyrimidine GPR119 agonists von Buzard, Daniel J., Kim, Sun Hee, Lehmann, Juerg, Han, Sangdon, Calderon, Imelda, Wong, Amy, Kawasaki, Andrew, Narayanan, Sanju, Bhat, Rohit, Gharbaoui, Tawfik, Lopez, Luis, Yue, Dawei, Whelan, Kevin, Al-Shamma, Hussien, Unett, David J., Shu, Hsin-Hui, Tung, Shiu-Feng, Chang, Steve, Chuang, Ching-Fen, Morgan, Michael, Sadeque, Abu, Chu, Zhi-Liang, Leonard, James N., Jones, Robert M.

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Agonist/antagonist modulation in a series of 2-aryl benzimidazole H4 receptor ligands von Savall, Brad M., Edwards, James P., Venable, Jennifer D., Buzard, Daniel J., Thurmond, Robin, Hack, Michael, McGovern, Patricia

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(7‑Benzyloxy-2,3-dihydro-1H-pyrrolo[1,2‑a]indol-1-yl)acetic Acids as S1P1 Functional Antagonists von Buzard, Daniel J, Lopez, Luis, Moody, Jeanne, Kawasaki, Andrew, Schrader, Thomas O, Kasem, Michelle, Johnson, Ben, Zhu, Xiuwen, Thoresen, Lars, Kim, Sun Hee, Gharbaoui, Tawfik, Sengupta, Dipanjan, Calvano, Lorene, Krishnan, Ashwin, Gao, Yinghong, Semple, Graeme, Edwards, Jeff, Barden, Jeremy, Morgan, Michael, Usmani, Khawja, Chen, Chuan, Sadeque, Abu, Chen, Weichao, Christopher, Ronald J, Thatte, Jayant, Fu, Lixia, Solomon, Michelle, Whelan, Kevin, Al-Shamma, Hussien, Gatlin, Joel, Gaidarov, Ibragim, Anthony, Todd, Le, Minh, Unett, David J, Stirn, Scott, Blackburn, Anthony, Behan, Dominic P, Jones, Robert M

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Synthesis of a Broad Array of Highly Functionalized, Enantiomerically Pure Cyclohexanecarboxylic Acid Derivatives by Microbial Dihydroxylation of Benzoic Acid and Subsequent Oxidat... von Myers, Andrew G, Siegel, Dionicio R, Buzard, Daniel J, Charest, Mark G

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Fused tricyclic indoles as S1P1 agonists with robust efficacy in animal models of autoimmune disease von Buzard, Daniel J., Han, Sangdon, Lopez, Luis, Kawasaki, Andrew, Moody, Jeanne, Thoresen, Lars, Ullman, Brett, Lehmann, Juerg, Calderon, Imelda, Zhu, Xiuwen, Gharbaoui, Tawfik, Sengupta, Dipanjan, Krishnan, Ashwin, Gao, Yinghong, Edwards, Jeff, Barden, Jeremy, Morgan, Michael, Usmani, Khawja, Chen, Chuan, Sadeque, Abu, Thatte, Jayant, Solomon, Michelle, Fu, Lixia, Whelan, Kevin, Liu, Ling, Al-Shamma, Hussien, Gatlin, Joel, Le, Minh, Xing, Charles, Espinola, Sheryll, Jones, Robert M.

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Design and synthesis of new tricyclic indoles as potent modulators of the S1P sub(1) receptor von Buzard, Daniel J, Schrader, Thomas O, Zhu, Xiuwen, Lehmann, Juerg, Johnson, Ben, Kasem, Michelle, Kim, Sun Hee, Kawasaki, Andrew, Lopez, Luis, Moody, Jeanne, Han, Sangdon, Gao, Yinghong, Edwards, Jeff, Barden, Jeremy, Thatte, Jayant, Gatlin, Joel, Jones, Robert M

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ChemInform Abstract: C—H Activation Reactions as Useful Tools for Medicinal Chemists von Caro‐Diaz, Eduardo J. E., Urbano, Mariangela, Buzard, Daniel J., Jones, Robert M.

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Identification of 2-arylbenzimidazoles as potent human histamine H 4 receptor ligands von Lee-Dutra, Alice, Arienti, Kristen L., Buzard, Daniel J., Hack, Michael D., Khatuya, Haripada, Desai, Pragnya J., Nguyen, Steven, Thurmond, Robin L., Karlsson, Lars, Edwards, James P., Breitenbucher, J. Guy

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Agonist/antagonist modulation in a series of 2-aryl benzimidazole H sub(4) receptor ligands von Savall, Brad M, Edwards, James P, Venable, Jennifer D, Buzard, Daniel J, Thurmond, Robin, Hack, Michael, McGovern, Patricia

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(7-Benzyloxy-2,3-dihydro- 1H -pyrrolo[1,2- a ]indol-1-yl)acetic Acids as S1P 1 Functional Antagonists von Buzard, Daniel J., Lopez, Luis, Moody, Jeanne, Kawasaki, Andrew, Schrader, Thomas O., Kasem, Michelle, Johnson, Ben, Zhu, Xiuwen, Thoresen, Lars, Kim, Sun Hee, Gharbaoui, Tawfik, Sengupta, Dipanjan, Calvano, Lorene, Krishnan, Ashwin, Gao, Yinghong, Semple, Graeme, Edwards, Jeff, Barden, Jeremy, Morgan, Michael, Usmani, Khawja, Chen, Chuan, Sadeque, Abu, Chen, Weichao, Christopher, Ronald J., Thatte, Jayant, Fu, Lixia, Solomon, Michelle, Whelan, Kevin, Al-Shamma, Hussien, Gatlin, Joel, Gaidarov, Ibragim, Anthony, Todd, Le, Minh, Unett, David J., Stirn, Scott, Blackburn, Anthony, Behan, Dominic P., Jones, Robert M.

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