ACE2 X-Ray Structures Reveal a Large Hinge-bending Motion Important for Inhibitor Binding and Catalysis von Towler, Paul, Staker, Bart, Prasad, Sridhar G., Menon, Saurabh, Tang, Jin, Parsons, Thomas, Ryan, Dominic, Fisher, Martin, Williams, David, Dales, Natalie A., Patane, Michael A., Pantoliano, Michael W.

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Discovery of Small Molecule Splicing Modulators of Survival Motor Neuron‑2 (SMN2) for the Treatment of Spinal Muscular Atrophy (SMA) von Cheung, Atwood K, Hurley, Brian, Kerrigan, Ryan, Shu, Lei, Chin, Donovan N, Shen, Yiping, O’Brien, Gary, Sung, Moo Je, Hou, Ying, Axford, Jake, Cody, Emma, Sun, Robert, Fazal, Aleem, Tomlinson, Ronald C, Jain, Monish, Deng, Lin, Hoffmaster, Keith, Song, Cheng, Van Hoosear, Mailin, Shin, Youngah, Servais, Rebecca, Towler, Christopher, Hild, Marc, Curtis, Daniel, Dietrich, William F, Hamann, Lawrence G, Briner, Karin, Chen, Karen S, Kobayashi, Dione, Sivasankaran, Rajeev, Dales, Natalie A

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Opportunities and challenges in developing stearoyl-coenzyme A desaturase-1 inhibitors as novel therapeutics for human disease von Zhang, Zaihui, Dales, Natalie A, Winther, Michael D

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Substrate-Based Design of the First Class of Angiotensin-Converting Enzyme-Related Carboxypeptidase (ACE2) Inhibitors von Dales, Natalie A, Gould, Alexandra E, Brown, James A, Calderwood, Emily F, Guan, Bing, Minor, Charles A, Gavin, James M, Hales, Paul, Kaushik, Virendar K, Stewart, Michael, Tummino, Peter J, Vickers, Chad S, Ocain, Timothy D, Patane, Michael A

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SMN2 splice modulators enhance U1–pre-mRNA association and rescue SMA mice von Palacino, James, Swalley, Susanne E, Song, Cheng, Cheung, Atwood K, Shu, Lei, Zhang, Xiaolu, Van Hoosear, Mailin, Shin, Youngah, Chin, Donovan N, Keller, Caroline Gubser, Beibel, Martin, Renaud, Nicole A, Smith, Thomas M, Salcius, Michael, Shi, Xiaoying, Hild, Marc, Servais, Rebecca, Jain, Monish, Deng, Lin, Bullock, Caroline, McLellan, Michael, Schuierer, Sven, Murphy, Leo, Blommers, Marcel J J, Blaustein, Cecile, Berenshteyn, Frada, Lacoste, Arnaud, Thomas, Jason R, Roma, Guglielmo, Michaud, Gregory A, Tseng, Brian S, Porter, Jeffery A, Myer, Vic E, Tallarico, John A, Hamann, Lawrence G, Curtis, Daniel, Fishman, Mark C, Dietrich, William F, Dales, Natalie A, Sivasankaran, Rajeev

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Discovery and characterization of a selective IKZF2 glue degrader for cancer immunotherapy von Bonazzi, Simone, d’Hennezel, Eva, Beckwith, Rohan E.J., Xu, Lei, Fazal, Aleem, Magracheva, Anna, Ramesh, Radha, Cernijenko, Artiom, Antonakos, Brandon, Bhang, Hyo-eun C., Caro, Roxana García, Cobb, Jennifer S., Ornelas, Elizabeth, Ma, Xiaolei, Wartchow, Charles A., Clifton, Matthew C., Forseth, Ry R., Fortnam, Bethany Hughes, Lu, Hongbo, Csibi, Alfredo, Tullai, Jennifer, Carbonneau, Seth, Thomsen, Noel M., Larrow, Jay, Chie-Leon, Barbara, Hainzl, Dominik, Gu, Yi, Lu, Darlene, Meyer, Matthew J., Alexander, Dylan, Kinyamu-Akunda, Jacqueline, Sabatos-Peyton, Catherine A., Dales, Natalie A., Zécri, Frédéric J., Jain, Rishi K., Shulok, Janine, Wang, Y. Karen, Briner, Karin, Porter, Jeffery A., Tallarico, John A., Engelman, Jeffrey A., Dranoff, Glenn, Bradner, James E., Visser, Michael, Solomon, Jonathan M.

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Use of Intramolecular 1,5-Sulfur–Oxygen and 1,5-Sulfur–Halogen Interactions in the Design of N‑Methyl-5-aryl‑N‑(2,2,6,6-tetramethylpiperidin-4-yl)-1,3,4-thiadiazol-2-amine SMN2 Spl... von Axford, Jake, Sung, Moo Je, Manchester, John, Chin, Donovan, Jain, Monish, Shin, Youngah, Dix, Ina, Hamann, Lawrence G, Cheung, Atwood K, Sivasankaran, Rajeev, Briner, Karin, Dales, Natalie A, Hurley, Brian

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Discovery and Optimization of First-in-Class Molecular Glue Degraders of the WIZ Transcription Factor for Fetal Hemoglobin Induction to Treat Sickle Cell Disease von Kerrigan, John Ryan, Thomsen, Noel M., Cernijenko, Artiom, Kochanek, Sarah E., Dewhurst, Janetta, O’Brien, Gary, Ware, Nathaniel F., Sanchez, Carina C., Manning, James R., Ma, Xiaolei, Ornelas, Elizabeth, Savage, Nikolas A., Partridge, James R., Patterson, Andrew W., Lam, Philip, Dales, Natalie A., Bonazzi, Simone, Borikar, Sneha, Hinman, Amelia E., Ting, Pamela Y.

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A molecular glue degrader of the WIZ transcription factor for fetal hemoglobin induction von Ting, Pamela Y, Borikar, Sneha, Kerrigan, John Ryan, Thomsen, Noel M, Aghania, Eamon, Hinman, Amelia E, Reyes, Alejandro, Pizzato, Nicolas, Fodor, Barna D, Wu, Fabian, Belew, Muluken S, Mao, Xiaohong, Wang, Jian, Chitnis, Shripad, Niu, Wei, Hachey, Amanda, Cobb, Jennifer S, Savage, Nikolas A, Burke, Ashley, Paulk, Joshiawa, Dovala, Dustin, Lin, James, Clifton, Matthew C, Ornelas, Elizabeth, Ma, Xiaolei, Ware, Nathaniel F, Sanchez, Carina C, Taraszka, John, Terranova, Remi, Knehr, Judith, Altorfer, Marc, Barnes, S Whitney, Beckwith, Rohan E J, Solomon, Jonathan M, Dales, Natalie A, Patterson, Andrew W, Wagner, Jürgen, Bouwmeester, Tewis, Dranoff, Glenn, Stevenson, Susan C, Bradner, James E

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High fire frequency and the impact of the 2019–2020 megafires on Australian plant diversity von Gallagher, Rachael V., Allen, Stuart, Mackenzie, Berin D. E., Yates, Colin J., Gosper, Carl R., Keith, David A., Merow, Cory, White, Matthew D., Wenk, Elizabeth, Maitner, Brian S., He, Kang, Adams, Vanessa M., Auld, Tony D.

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Bacterial community mapping of the mouse gastrointestinal tract von Gu, Shenghua, Chen, Dandan, Zhang, Jin-Na, Lv, Xiaoman, Wang, Kun, Duan, Li-Ping, Nie, Yong, Wu, Xiao-Lei

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Banach Spaces of Continuous Functions as Dual Spaces von Dales, H. G

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Sequencing-based analysis of the bacterial and fungal composition of kefir grains and milks from multiple sources von Marsh, Alan J, O'Sullivan, Orla, Hill, Colin, Ross, R Paul, Cotter, Paul D

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Enzymatic Characterization of the Pancreatic Islet-specific Glucose-6-Phosphatase-related Protein (IGRP) von Petrolonis, Anthony J, Yang, Qing, Tummino, Peter J, Fish, Susan M, Prack, Andrea E, Jain, Sadhana, Parsons, Thomas F, Li, Ping, Dales, Natalie A, Ge, Lin, Langston, Steven P, Schuller, Alwin G P, An, W Frank, Tartaglia, Louis A, Chen, Hong, Hong, Suk-Bong

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Opportunities and Challenges in Developing Stearoyl-Coenzyme A Desaturase‑1 Inhibitors as Novel Therapeutics for Human Disease: Miniperspective von Zhang, Zaihui, Dales, Natalie A, Winther, Michael D

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Complexity and variability of gut commensal microbiota in polyphagous lepidopteran larvae von Tang, Xiaoshu, Freitak, Dalial, Vogel, Heiko, Ping, Liyan, Shao, Yongqi, Cordero, Erika Arias, Andersen, Gary, Westermann, Martin, Heckel, David G, Boland, Wilhelm

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Functional and Logic Programming: 17th International Symposium, FLOPS 2024, Kumamoto, Japan, May 15-17, 2024, Proceedings von Gibbons, Jeremy, Miller, Dale

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Using lidar data to analyse sinkhole characteristics relevant for understory vegetation under forest cover-case study of a high karst area in the dinaric mountains von Kobal, Milan, Bertoncelj, Irena, Pirotti, Francesco, Dakskobler, Igor, Kutnar, Lado

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Intermediate fire severity diversity promotes richness of forest carnivores in California von Furnas, Brett J., Goldstein, Benjamin R., Figura, Peter J.

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Systematic evaluation of amide bioisosteres leading to the discovery of novel and potent thiazolylimidazolidinone inhibitors of SCD1 for the treatment of metabolic diseases von Sun, Shaoyi, Zhang, Zaihui, Kodumuru, Vishnumurthy, Pokrovskaia, Natalia, Fonarev, Julia, Jia, Qi, Leung, Po-Yee, Tran, Jennifer, Ratkay, Leslie G., McLaren, David G., Radomski, Chris, Chowdhury, Sultan, Fu, Jianmin, Hubbard, Brian, Winther, Michael D., Dales, Natalie A.

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