Gatorbulin-1, a distinct cyclodepsipeptide chemotype, targets a seventh tubulin pharmacological site von Matthew, Susan, Chen, Qi-Yin, Ratnayake, Ranjala, Fermaintt, Charles S., Lucena-Agell, Daniel, Bonato, Francesca, Prota, Andrea E., Lim, Seok Ting, Wang, Xiaomeng, Díaz, J. Fernando, Risinger, April L., Paul, Valerie J., Oliva, Maria Ángela, Luesch, Hendrik

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Deconvolution of Buparlisib’s mechanism of action defines specific PI3K and tubulin inhibitors for therapeutic intervention von Bohnacker, Thomas, Prota, Andrea E., Beaufils, Florent, Burke, John E., Melone, Anna, Inglis, Alison J., Rageot, Denise, Sele, Alexander M., Cmiljanovic, Vladimir, Cmiljanovic, Natasa, Bargsten, Katja, Aher, Amol, Akhmanova, Anna, Díaz, J. Fernando, Fabbro, Doriano, Zvelebil, Marketa, Williams, Roger L., Steinmetz, Michel O., Wymann, Matthias P.

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Taxanes convert regions of perturbed microtubule growth into rescue sites von Rai, Ankit, Liu, Tianyang, Glauser, Simon, Katrukha, Eugene A., Estévez-Gallego, Juan, Rodríguez-García, Ruddi, Fang, Wei-Shuo, Díaz, J. Fernando, Steinmetz, Michel O., Altmann, Karl-Heinz, Kapitein, Lukas C., Moores, Carolyn A., Akhmanova, Anna

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High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design von Bueno, Oskía, Estévez Gallego, Juan, Martins, Solange, Prota, Andrea E., Gago, Federico, Gómez-SanJuan, Asier, Camarasa, María-José, Barasoain, Isabel, Steinmetz, Michel O., Díaz, J. Fernando, Pérez-Pérez, María-Jesús, Liekens, Sandra, Priego, Eva-María

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Neuronal Subtype Specification within a Lineage by Opposing Temporal Feed-Forward Loops von Baumgardt, Magnus, Karlsson, Daniel, Terriente, Javier, Díaz-Benjumea, Fernando J., Thor, Stefan

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Structural model for differential cap maturation at growing microtubule ends von Estevez-Gallego, Juan, Josa-Prado, Fernando, Ku, Siou, Buey, Ruben M., Balaguer, Francisco A., Prota, Andrea E., Lucena-Agell, Daniel, Kamma-Lorger, Christina, Yagi, Toshiki, Iwamoto, Hiroyuki, Duchesne, Laurence, Barasoain, Isabel, Steinmetz, Michel O., Chretien, Denis, Kamimura, Shinji, Fernando Diaz, J., Oliva, Maria A.

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A fluorescence anisotropy assay to discover and characterize ligands targeting the maytansine site of tubulin von Menchon, Grégory, Prota, Andrea E., Lucena-Agell, Daniel, Bucher, Pascal, Jansen, Rolf, Irschik, Herbert, Müller, Rolf, Paterson, Ian, Díaz, J. Fernando, Altmann, Karl-Heinz, Steinmetz, Michel O.

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Lateral wedge insoles and their use in ankle instability von Palomo‐Fernández, Inés, Martín‐Casado, Laura, Marcos‐Tejedor, Félix, Aldana‐Caballero, Alberto, Rubio‐Arias, Jacobo. Á., Jiménez‐Díaz, J. Fernando

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Structural insight into the stabilization of microtubules by taxanes von Prota, Andrea E, Lucena-Agell, Daniel, Ma, Yuntao, Estevez-Gallego, Juan, Li, Shuo, Bargsten, Katja, Josa-Prado, Fernando, Altmann, Karl-Heinz, Gaillard, Natacha, Kamimura, Shinji, Mühlethaler, Tobias, Gago, Federico, Oliva, Maria A, Steinmetz, Michel O, Fang, Wei-Shuo, Díaz, J Fernando

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PM534, an Optimized Target-Protein Interaction Strategy through the Colchicine Site of Tubulin von Lucena-Agell, Daniel, Guillén, María José, Matesanz, Ruth, Álvarez-Bernad, Beatriz, Hortigüela, Rafael, Avilés, Pablo, Martínez-Díez, Marta, Santamaría-Núñez, Gema, Contreras, Julia, Plaza-Menacho, Iván, Giménez-Abián, Juan F., Oliva, María A., Cuevas, Carmen, Díaz, J. Fernando

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Synthesis, Characterization, and Application in HeLa Cells of an NIR Light Responsive Doxorubicin Delivery System Based on NaYF4:Yb,Tm@SiO2‑PEG Nanoparticles von Alonso-Cristobal, Paulino, Oton-Fernandez, Olalla, Mendez-Gonzalez, Diego, Díaz, J. Fernando, Lopez-Cabarcos, Enrique, Barasoain, Isabel, Rubio-Retama, Jorge

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Synthesis and Antimitotic and Tubulin Interaction Profiles of Novel Pinacol Derivatives of Podophyllotoxins von Abad, Andrés, López-Pérez, José L, del Olmo, Esther, García-Fernández, Luis F, Francesch, Andrés, Trigili, Chiara, Barasoain, Isabel, Andreu, José M, Díaz, J. Fernando, San Feliciano, Arturo

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Targeting the tubulin C-terminal tail by charged small molecules von Li, Shuo, Mori, Mattia, Yang, Mingyan, Elfazazi, Soumia, Hortigüela, Rafael, Chan, Peter, Feng, Xinyue, Risinger, April, Yang, Zhiyou, Oliva, María Ángela, Fernando Díaz, J, Fang, Wei-Shuo

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Design and Synthesis of Pironetin Analogue/Colchicine Hybrids and Study of Their Cytotoxic Activity and Mechanisms of Interaction with Tubulin von Vilanova, Concepción, Díaz-Oltra, Santiago, Murga, Juan, Falomir, Eva, Carda, Miguel, Redondo-Horcajo, Mariano, Díaz, J. Fernando, Barasoain, Isabel, Marco, J. Alberto

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Self-Organization of FtsZ Polymers in Solution Reveals Spacer Role of the Disordered C-Terminal Tail von Huecas, Sonia, Ramírez-Aportela, Erney, Vergoñós, Albert, Núñez-Ramírez, Rafael, Llorca, Oscar, Díaz, J. Fernando, Juan-Rodríguez, David, Oliva, María A., Castellen, Patricia, Andreu, José M.

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Development of Potent Microtubule Targeting Agent by Structural Simplification of Natural Diazonamide von Kalnins, Toms, Vitkovska, Viktorija, Kazak, Mihail, Zelencova-Gopejenko, Diana, Ozola, Melita, Narvaiss, Nauris, Makrecka-Kuka, Marina, Domračeva, Ilona, Kinens, Artis, Gukalova, Baiba, Konrad, Nele, Aav, Riina, Bonato, Francesca, Lucena-Agell, Daniel, Díaz, J. Fernando, Liepinsh, Edgars, Suna, Edgars

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Semiempirical model for the estimation of site amplification in northern South America von Mercado, Vicente, Pajaro, Cesar A, Arteta, Carlos A, Díaz, Fernando J, Montejo, Julián, Arcila, Mónica, Abrahamson, Norman A

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Identification of the guanine nucleotide exchange factor for SAR1 in the filamentous fungal model Aspergillus nidulans von Bravo-Plaza, Ignacio, Hernández-González, Miguel, Pinar, Mario, Díaz, J. Fernando, Peñalva, Miguel A.

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Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands von Balaguer, Francisco de Asís, Mühlethaler, Tobias, Estévez-Gallego, Juan, Calvo, Enrique, Giménez-Abián, Juan Francisco, Risinger, April L, Sorensen, Erik J, Vanderwal, Christopher D, Altmann, Karl-Heinz, Mooberry, Susan L, Steinmetz, Michel O, Oliva, María Ángela, Prota, Andrea E, Díaz, J Fernando

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Alternative Approaches to Understand Microtubule Cap Morphology and Function von Oliva, María Ángela, Gago, Federico, Kamimura, Shinji, Díaz, J. Fernando

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