Preclinical pharmacology and pharmacokinetics of AZD3783, a selective 5-hydroxytryptamine 1B receptor antagonist von Zhang, Minli, Zhou, Diansong, Wang, Yi, Maier, Donna L, Widzowski, Daniel V, Sobotka-Briner, Cynthia D, Brockel, Becky J, Potts, William M, Shenvi, Ashok B, Bernstein, Peter R, Pierson, M Edward

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Linear non-competitive inhibition of solubilized human gamma-secretase by pepstatin A methylester, L685458, sulfonamides, and benzodiazepines von Tian, Gaochao, Sobotka-Briner, Cynthia D, Zysk, John, Liu, Xiaodong, Birr, Cynthia, Sylvester, Mark A, Edwards, Philip D, Scott, Clay D, Greenberg, Barry D

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De Novo Design of a Picomolar Nonbasic 5-HT1B Receptor Antagonist von Nugiel, David A, Krumrine, Jennifer R, Hill, Daniel C, Damewood, James R, Bernstein, Peter R, Sobotka-Briner, Cynthia D, Liu, JianWei, Zacco, Anna, Pierson, M. Edward

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De Novo Design of a Picomolar Nonbasic 5-HT 1B Receptor Antagonist von Nugiel, David A., Krumrine, Jennifer R., Hill, Daniel C., Damewood, James R., Bernstein, Peter R., Sobotka-Briner, Cynthia D., Liu, JianWei, Zacco, Anna, Pierson, M. Edward

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Linear Non-competitive Inhibition of Solubilized Human γ-Secretase by Pepstatin A Methylester, L685458, Sulfonamides, and Benzodiazepines von Gaochao Tian, Cynthia D. Sobotka-Briner, John Zysk, Xiaodong Liu, Cynthia Birr, Mark A. Sylvester, Philip D. Edwards, Clay D. Scott, Barry D. Greenberg

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De novo design of a picomolar nonbasic 5-HT(1B) receptor antagonist von Nugiel, David A, Krumrine, Jennifer R, Hill, Daniel C, Damewood, Jr, James R, Bernstein, Peter R, Sobotka-Briner, Cynthia D, Liu, Jianwei, Zacco, Anna, Pierson, M Edward

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Non‐Competitive Inhibition of Solubilized Human γ‐Secretase by Pepstatin A Methylester, L‐685458, Sulfonamides and Benzodiazepines von Tian, Gaochao, Sobotka‐Briner, Cynthia D., Zysk, John, Liu, Xiaodong, Birr, Cynthia, Sylvester, Mark A., Edwards, Phil D., Scott, Clay W., Greenberg, Barry D.

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Mechanism of γ-Secretase Cleavage Activation:  Is γ-Secretase Regulated through Autoinhibition Involving the Presenilin-1 Exon 9 Loop? von Knappenberger, Katharine S, Tian, Gaochao, Ye, Xiaomei, Sobotka-Briner, Cynthia, Ghanekar, Smita V, Greenberg, Barry D, Scott, Clay W

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COOH-terminal methylation of lamin B and inhibition of methylation by farnesylated peptides corresponding to lamin B and other CAAX motif proteins von C Sobotka-Briner, D Chelsky

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