Identification of the First Synthetic Steroidogenic Factor 1 Inverse Agonists: Pharmacological Modulation of Steroidogenic Enzymes von Del Tredici, Andria L., Andersen, Carsten B., Currier, Erika A., Ohrmund, Steven R., Fairbain, Luke C., Lund, Birgitte W., Nash, Norman, Olsson, Roger, Piu, Fabrice

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Oral RKS262 reduces tumor burden in a neuroblastoma xenograft animal model and mediates cytotoxicity through SAPK/JNK and ROS activation in vitro von Singh, Rakesh K., Dorf, Lee, DeMartino, Angelica, Illenye, Sharon, Koto, Karen, Currier, Erika A., Ashikaga, Takamaru, Kim, Kyu Kwang, Brard, Laurent, Saulnier Sholler, Giselle L.

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Optimization of isochromanone based urotensin II receptor agonists von Lehmann, Fredrik, Currier, Erika A., Olsson, Roger, Ma, Jian-Nong, Burstein, Ethan S., Hacksell, Uli, Luthman, Kristina

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Identification of novel subtype selective RAR agonists von Piu, Fabrice, Gauthier, Natalie K., Olsson, Roger, Currier, Erika A., Lund, Birgitte W., Croston, Glenn E., Hacksell, Uli, Brann, Mark R.

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Identification of the Atypical L-Type Ca2+ Channel Blocker Diltiazem and Its Metabolites As Ghrelin Receptor Agonists von Ma, Jian-Nong, Schiffer, Hans H., Knapp, Anne E., Wang, Jean, Wong, Kenneth K., Currier, Erika A., Owens, Michelle, Nash, Norman R., Gardell, Luis R., Brann, Mark R., Olsson, Roger, Burstein, Ethan S.

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Discovery of Potent and Selective Small-Molecule PAR-2 Agonists von Seitzberg, Jimmi Gerner, Knapp, Anne Eeg, Lund, Birgitte Winther, Mandrup Bertozzi, Sine, Currier, Erika A, Ma, Jian-Nong, Sherbukhin, Vladimir, Burstein, Ethan S, Olsson, Roger

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Design, parallel synthesis and SAR of novel urotensin II receptor agonists von Lehmann, Fredrik, Lake, Lisa, Currier, Erika A., Olsson, Roger, Hacksell, Uli, Luthman, Kristina

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Synthesis and Evaluation of Dibenzothiazepines: A Novel Class of Selective Cannabinoid-1 Receptor Inverse Agonists von Pettersson, Hanna, Bülow, Anne, Ek, Fredrik, Jensen, Jacob, Ottesen, Lars K, Fejzic, Alma, Ma, Jian-Nong, Del Tredici, Andria L, Currier, Erika A, Gardell, Luis R, Tabatabaei, Ali, Craig, Darren, McFarland, Krista, Ott, Thomas R, Piu, Fabrice, Burstein, Ethan S, Olsson, Roger

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Discovery of non-peptidergic MrgX1 and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesis von Malik, Leila, Kelly, Nicholas M, Ma, Jian-Nong, Currier, Erika A, Burstein, Ethan S, Olsson, Roger

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Novel Potent and Efficacious Nonpeptidic Urotensin II Receptor Agonists von Lehmann, Fredrik, Pettersen, Anna, Currier, Erika A, Sherbukhin, Vladimir, Olsson, Roger, Hacksell, Uli, Luthman, Kristina

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Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols von Gustafsson, Magnus, Jensen, Jacob, Bertozzi, Sine M., Currier, Erika A., Ma, Jian-Nong, Burstein, Ethan S., Olsson, Roger

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Novel and potent small-molecule urotensin II receptor agonists von Lehmann, Fredrik, Currier, Erika A., Clemons, Bryan, Hansen, Lars K., Olsson, Roger, Hacksell, Uli, Luthman, Kristina

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Isochromanone-based urotensin-II receptor agonists von Lehmann, Fredrik, Currier, Erika A., Olsson, Roger, Hacksell, Uli, Luthman, Kristina

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Discovery of the First Nonpeptide Agonist of the GPR14/Urotensin-II Receptor:  3-(4-Chlorophenyl)-3-(2- (dimethylamino)ethyl)isochroman-1-one (AC-7954) von Croston, Glenn E, Olsson, Roger, Currier, Erika A, Burstein, Ethan S, Weiner, David, Nash, Norman, Severance, Daniel, Allenmark, Stig G, Thunberg, Linda, Ma, Jian-Nong, Mohell, Nina, O'Dowd, Brian, Brann, Mark R, Hacksell, Uli

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Identification of novel selective v2 receptor non-peptide agonists von DEL TREDID, Andria L, VANOVER, Kim E, MOHELL, Nina, OLSSON, Roger, PIN, Fabrice, KNAPP, Anne E, BERTOZZI, Sine M, NASH, Norman R, BURSTEIN, Ethan S, LAMEH, Jelveh, CURRIER, Erika A, DAVIS, Robert E, BRANN, Mark R

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Discovery of novel peptide/receptor interactions: identification of PHM-27 as a potent agonist of the human calcitonin receptor von Ma, Jian-Nong, Currier, Erika A, Essex, Anthony, Feddock, Michele, Spalding, Tracy A, Nash, Norman R, Brann, Mark R, Burstein, Ethan S

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The ras-related GTPase rac1 regulates a proliferative pathway selectively utilized by G-protein coupled receptors von BURSTEIN, E. S, HESTERBERG, D. J, GUTKIND, J. S, BRANN, M. R, CURRIER, E. A, MESSIER, T. L

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Discovery of an Ectopic Activation Site on the M 1 Muscarinic Receptor von Spalding, Tracy A., Trotter, Carol, Skjærbæk, Niels, Messier, Terri L., Currier, Erika A., Burstein, Ethan S., Li, Donghui, Hacksell, Uli, Brann, Mark R.

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Abstract 5260: Bortezomib and HDAC inhibitor PCI-24781 combination therapy for neuroblastoma von Currier, Erika A., Illenye, Sharon A., Ashikaga, Takamaru, Lescault, Pamela J., Bond, Jeffrey P., Sholler, Giselle L. Saulnier

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Discovery of non-peptidergic MrgXl and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesis von MALIK, Leila, KELLY, Nicholas M, MA, Jian-Nong, CURRIER, Erika A, BURSTEIN, Ethan S, OLSSON, Roger

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