Direct arylations on water: synthesis of 2,5-disubstituted oxazoles balsoxin and texaline von Ohnmacht, Stephan A, Mamone, Patrizia, Culshaw, Andrew J, Greaney, Michael F

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Direct Arylations of 2H-Indazoles On Water von Ohnmacht, Stephan A, Culshaw, Andrew J, Greaney, Michael F

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Potent and Orally Bioavailable Non-Peptide Antagonists at the Human Bradykinin B1 Receptor Based on a 2-Alkylamino-5-sulfamoylbenzamide Core von Ritchie, Timothy J, Dziadulewicz, Edward K, Culshaw, Andrew J, Müller, Werner, Burgess, Gillian M, Bloomfield, Graham C, Drake, Gillian S, Dunstan, Andrew R, Beattie, David, Hughes, Glyn A, Ganju, Pam, McIntyre, Peter, Bevan, Stuart J, Davis, Clare, Yaqoob, Mohammed

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Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone:  A Potent, Orally Bioavailable Human CB1/CB2 Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous Sys... von Dziadulewicz, Edward K, Bevan, Stuart J, Brain, Christopher T, Coote, Paul R, Culshaw, Andrew J, Davis, Andrew J, Edwards, Lee J, Fisher, Adrian J, Fox, Alyson J, Gentry, Clive, Groarke, Alex, Hart, Terance W, Huber, Werner, James, Iain F, Kesingland, Adam, La Vecchia, Luigi, Loong, Yvonne, Lyothier, Isabelle, McNair, Kara, O'Farrell, Cathal, Peacock, Marcus, Portmann, Robert, Schopfer, Ulrich, Yaqoob, Mohammed, Zadrobilek, Jiri

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Discovery of Orally Bioavailable Cathepsin S Inhibitors for the Reversal of Neuropathic Pain von Irie, Osamu, Kosaka, Takatoshi, Ehara, Takeru, Yokokawa, Fumiaki, Kanazawa, Takanori, Hirao, Hajime, Iwasaki, Astuko, Sakaki, Junichi, Teno, Naoki, Hitomi, Yuko, Iwasaki, Genji, Fukaya, Hiroaki, Nonomura, Kazuhiko, Tanabe, Keiko, Koizumi, Shinichi, Uchiyama, Noriko, Bevan, Stuart J, Malcangio, Marzia, Gentry, Clive, Fox, Alyson J, Yaqoob, Mohammed, Culshaw, Andrew J, Hallett, Allan

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Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2 von Irie, Osamu, Kosaka, Takatoshi, Kishida, Masashi, Sakaki, Junichi, Masuya, Keiichi, Konishi, Kazuhide, Yokokawa, Fumiaki, Ehara, Takeru, Iwasaki, Atsuko, Iwaki, Yuki, Hitomi, Yuko, Toyao, Atsushi, Gunji, Hiroki, Teno, Naoki, Iwasaki, Genji, Hirao, Hajime, Kanazawa, Takanori, Tanabe, Keiko, Hiestand, Peter C., Malcangio, Marzia, Fox, Alyson J., Bevan, Stuart J., Yaqoob, Mohammed, Culshaw, Andrew J., Hart, Terance W., Hallett, Allan

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Identification and Biological Characterization of 6-Aryl-7-isopropylquinazolinones as Novel TRPV1 Antagonists that Are Effective in Models of Chronic Pain von Culshaw, Andrew J, Bevan, Stuart, Christiansen, Martin, Copp, Prafula, Davis, Andrew, Davis, Clare, Dyson, Alex, Dziadulewicz, Edward K, Edwards, Lee, Eggelte, Hendrikus, Fox, Alyson, Gentry, Clive, Groarke, Alex, Hallett, Allan, Hart, Terance W, Hughes, Glyn A, Knights, Sally, Kotsonis, Peter, Lee, Wai, Lyothier, Isabelle, McBryde, Andrew, McIntyre, Peter, Paloumbis, George, Panesar, Moh, Patel, Sadhana, Seiler, Max-Peter, Yaqoob, Mohammed, Zimmermann, Kaspar

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Studies on the Biomimetic Synthesis of the Manzamine Alkaloids von Baldwin, Jack E., Claridge, Timothy D. W., Culshaw, Andrew J., Heupel, Florian A., Lee, Victor, Spring, David R., Whitehead, Roger C.

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A biomimetic approach to the manzamine alkaloids von Baldwin, Jack E, Claridge, Tim D.W, Culshaw, Andrew J, Heupel, Florian A, Smrcková, Svatava, Whitehead, Roger C

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Investigations into the Manzamine Alkaloid Biosynthetic Hypothesis von Baldwin, Jack E., Claridge, Timothy D. W., Culshaw, Andrew J., Heupel, Florian A., Lee, Victor, Spring, David R., Whitehead, Roger C., Boughtflower, Robert J., Mutton, Ian M., Upton, Richard J.

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Direct Arylations of 2 H -Indazoles On Water von Ohnmacht, Stephan A., Culshaw, Andrew J., Greaney, Michael F.

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Solid phase synthesis of functionalized biaryl ethers: versatile scaffolds for combinatorial chemistry von Wijkmans, J C, Culshaw, A J, Baxter, A D

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Potent and Orally Bioavailable Non-Peptide Antagonists at the Human Bradykinin B 1 Receptor Based on a 2-Alkylamino-5-sulfamoylbenzamide Core von Ritchie, Timothy J., Dziadulewicz, Edward K., Culshaw, Andrew J., Müller, Werner, Burgess, Gillian M., Bloomfield, Graham C., Drake, Gillian S., Dunstan, Andrew R., Beattie, David, Hughes, Glyn A., Ganju, Pam, McIntyre, Peter, Bevan, Stuart J., Davis, Clare, Yaqoob, Mohammed

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Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone: A Potent, Orally Bioavailable Human CB 1 /CB 2 Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous S... von Dziadulewicz, Edward K., Bevan, Stuart J., Brain, Christopher T., Coote, Paul R., Culshaw, Andrew J., Davis, Andrew J., Edwards, Lee J., Fisher, Adrian J., Fox, Alyson J., Gentry, Clive, Groarke, Alex, Hart, Terance W., Huber, Werner, James, Iain F., Kesingland, Adam, La Vecchia, Luigi, Loong, Yvonne, Lyothier, Isabelle, McNair, Kara, O'Farrell, Cathal, Peacock, Marcus, Portmann, Robert, Schopfer, Ulrich, Yaqoob, Mohammed, Zadrobilek, Jiri

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Identification and biological characterization of 6-aryl-7-isopropylquinazolinones as novel TRPV1 antagonists that are effective in models of chronicpain von CULSHAW, Andrew J, BEVAN, Stuart, FOX, Alyson, GENTRY, Clive, GROARKE, Alex, HALLETT, Allan, HART, Terance W, HUGHES, Glyn A, KNIGHTS, Sally, KOTSONIS, Peter, LEE, Wai, LYOTHIER, Isabelle, CHRISTIANSEN, Martin, MCBRYDE, Andrew, MCINTYRE, Peter, PALOUMBIS, George, PANESAR, Moh, PATEL, Sadhana, SEILER, Max-Peter, YAQOOB, Mohammed, ZIMMERMANN, Kaspar, COPP, Prafula, DAVIS, Andrew, DAVIS, Clare, DYSON, Alex, DZIADULEWICZ, Edward K, EDWARDS, Lee, EGGELTE, Hendrikus

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Potent and orally bioavailable non-peptide antagonists at the human bradykinin B(1) receptor based on a 2-alkylamino-5-sulfamoylbenzamide core von Ritchie, Timothy J, Dziadulewicz, Edward K, Culshaw, Andrew J, Müller, Werner, Burgess, Gillian M, Bloomfield, Graham C, Drake, Gillian S, Dunstan, Andrew R, Beattie, David, Hughes, Glyn A, Ganju, Pam, McIntyre, Peter, Bevan, Stuart J, Davis, Clare, Yaqoob, Mohammed

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Cycloadditions of Carbonyl Oxides: A Novel Stereoselective Approach to 1,3-Diols von Casey, Mike, Culshaw, Andrew J.

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ChemInform Abstract: Direct Arylation of 2H-Indazoles on Water von Ohnmacht, Stephen A., Culshaw, Andrew J., Greaney, Michael F.

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ChemInform Abstract: Direct Arylations on Water: Synthesis of 2,5-Disubstituted Oxazoles Balsoxin and Texaline von Ohnmacht, Stephan A., Mamone, Patrizia, Culshaw, Andrew J., Greaney, Michael F.

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Untersuchungen zur Hypothese der Manzaminalkaloid‐Biosynthese von Baldwin, Jack E., Claridge, Timothy D. W., Culshaw, Andrew J., Heupel, Florian A., Lee, Victor, Spring, David R., Whitehead, Roger C., Boughtflower, Robert J., Mutton, Ian M., Upton, Richard J.

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