Aminomethyl Salicylaldehydes Lock onto a Surface Lysine by Forming an Extended Intramolecular Hydrogen Bond Network von Weaver, Jacqueline, Craven, Gregory B., Tram, Linh, Chen, Hao, Taunton, Jack

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Reversible lysine-targeted probes reveal residence time-based kinase selectivity von Yang, Tangpo, Cuesta, Adolfo, Wan, Xiaobo, Craven, Gregory B., Hirakawa, Brad, Khamphavong, Penney, May, Jeffrey R., Kath, John C., Lapek, John D., Niessen, Sherry, Burlingame, Alma L., Carelli, Jordan D., Taunton, Jack

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Signal peptide mimicry primes Sec61 for client-selective inhibition von Rehan, Shahid, Tranter, Dale, Sharp, Phillip P., Craven, Gregory B., Lowe, Eric, Anderl, Janet L., Muchamuel, Tony, Abrishami, Vahid, Kuivanen, Suvi, Wenzell, Nicole A., Jennings, Andy, Kalyanaraman, Chakrapani, Strandin, Tomas, Javanainen, Matti, Vapalahti, Olli, Jacobson, Matthew P., McMinn, Dustin, Kirk, Christopher J., Huiskonen, Juha T., Taunton, Jack, Paavilainen, Ville O.

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Direct mapping of ligandable tyrosines and lysines in cells with chiral sulfonyl fluoride probes von Chen, Ying, Craven, Gregory B., Kamber, Roarke A., Cuesta, Adolfo, Zhersh, Serhii, Moroz, Yurii S., Bassik, Michael C., Taunton, Jack

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High‐Throughput Kinetic Analysis for Target‐Directed Covalent Ligand Discovery von Craven, Gregory B., Affron, Dominic P., Allen, Charlotte E., Matthies, Stefan, Greener, Joe G., Morgan, Rhodri M. L., Tate, Edward W., Armstrong, Alan, Mann, David J.

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Synthesis and Configurational Assignment of Vinyl Sulfoximines and Sulfonimidamides von Craven, Gregory B, Briggs, Edward L, Zammit, Charlotte M, McDermott, Alexander, Greed, Stephanie, Affron, Dominic P, Leinfellner, Charlotte, Cudmore, Hannah R, Tweedy, Ruth R, Luisi, Renzo, Bull, James A, Armstrong, Alan

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Unexpected structures formed by the kinase RET C634R mutant extracellular domain suggest potential oncogenic mechanisms in MEN2A von Liu, Yixin, De Castro Ribeiro, Orquidea, Haapanen, Outi, Craven, Gregory B., Sharma, Vivek, Muench, Stephen P., Goldman, Adrian

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Structure of eukaryotic purine/H+ symporter UapA suggests a role for homodimerization in transport activity von Alguel, Yilmaz, Amillis, Sotiris, Leung, James, Lambrinidis, George, Capaldi, Stefano, Scull, Nicola J., Craven, Gregory, Iwata, So, Armstrong, Alan, Mikros, Emmanuel, Diallinas, George, Cameron, Alexander D., Byrne, Bernadette

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Mutant-selective AKT inhibition through lysine targeting and neo-zinc chelation von Craven, Gregory B, Chu, Hang, Sun, Jessica D, Carelli, Jordan D, Coyne, Brittany, Chen, Hao, Chen, Ying, Ma, Xiaolei, Das, Subhamoy, Kong, Wayne, Zajdlik, Adam D, Yang, Kin S, Reisberg, Solomon H, Thompson, Peter A, Lipford, J Russell, Taunton, Jack

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Intramolecular hydride transfer onto arynes: redox-neutral and transition metal-free C(sp)-H functionalization of amines von Idiris, Fahima I. M, Majesté, Cécile E, Craven, Gregory B, Jones, Christopher R

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Quantitative Irreversible Tethering (qIT) for Target-directed Covalent Fragment Screening von Craven, Gregory B, Armstrong, Alan, Mann, David J

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Reversible lysine-targeted probes reveal residence time-based kinase selectivity von Yang, Tangpo, Cuesta, Adolfo, Wan, Xiaobo, Craven, Gregory B., Hirakawa, Brad, Khamphavong, Penney, May, Jeffrey R., Kath, John C., Lapek, John D., Niessen, Sherry, Burlingame, Alma L., Carelli, Jordan D., Taunton, Jack

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Multiparameter Kinetic Analysis for Covalent Fragment Optimization by Using Quantitative Irreversible Tethering (qIT) von Craven, Gregory B., Affron, Dominic P., Kösel, Teresa, Wong, Tsz Lam M., Jukes, Zoë H., Liu, Chun‐Ting, Morgan, Rhodri M. L., Armstrong, Alan, Mann, David J.

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Acrylamide fragment inhibitors that induce unprecedented conformational distortions in enterovirus 71 3C and SARS-CoV-2 main protease von Qin, Bo, Craven, Gregory B., Hou, Pengjiao, Chesti, Julian, Lu, Xinran, Child, Emma S., Morgan, Rhodri M.L., Niu, Wenchao, Zhao, Lina, Armstrong, Alan, Mann, David J., Cui, Sheng

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Identification of the first structurally validated covalent ligands of the small GTPase RAB27A von Jamshidiha, Mostafa, Lanyon-Hogg, Thomas, Sutherell, Charlotte L, Craven, Gregory B, Tersa, Montse, De Vita, Elena, Brustur, Delia, Pérez-Dorado, Inmaculada, Hassan, Sarah, Petracca, Rita, Morgan, Rhodri M, Sanz-Hernández, Máximo, Norman, Jim C, Armstrong, Alan, Mann, David J, Cota, Ernesto, Tate, Edward W

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Vinyl sulfonamide synthesis for irreversible tethering via a novel α-selenoether protection strategy von Craven, Gregory B, Affron, Dominic P, Raymond, Philip N, Mann, David J, Armstrong, Alan

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High‐Throughput Kinetic Analysis for Target‐Directed Covalent Ligand Discovery von Craven, Gregory B., Affron, Dominic P., Allen, Charlotte E., Matthies, Stefan, Greener, Joe G., Morgan, Rhodri M. L., Tate, Edward W., Armstrong, Alan, Mann, David J.

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Intramolecular hydride transfer onto arynes: redox-neutral and transition metal-free C(sp3)–H functionalization of amines† †Electronic supplementary information (ESI) available. Se... von Idiris, Fahima I. M., Majesté, Cécile E., Craven, Gregory B., Jones, Christopher R.

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High-throughput kinetic analysis for target-directed covalent ligand discovery von Craven, Gregory

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Vinyl sulfonamide synthesis for irreversible tethering a novel α-selenoether protection strategy von Craven, Gregory B, Affron, Dominic P, Raymond, Philip N, Mann, David J, Armstrong, Alan

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