Factors Determining the Selection of Organic Reactions by Medicinal Chemists and the Use of These Reactions in Arrays (Small Focused Libraries) von Cooper, Tony W.J, Campbell, Ian B, Macdonald, Simon J.F

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Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor von Biggadike, Keith, Bledsoe, Randy K, Coe, Diane M, Cooper, Tony W.J, House, David, Iannone, Marie A, Macdonald, Simon J.F, Madauss, Kevin P, McLay, Iain M, Shipley, Tracy J, Taylor, Simon J, Tran, Thuy B, Uings, Iain J, Weller, Victoria, Williams, Shawn P

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Circadian clock component REV-ERBα controls homeostatic regulation of pulmonary inflammation von Pariollaud, Marie, Gibbs, Julie E, Hopwood, Thomas W, Brown, Sheila, Begley, Nicola, Vonslow, Ryan, Poolman, Toryn, Guo, Baoqiang, Saer, Ben, Jones, D Heulyn, Tellam, James P, Bresciani, Stefano, Tomkinson, Nicholas Co, Wojno-Picon, Justyna, Cooper, Anthony Wj, Daniels, Dion A, Trump, Ryan P, Grant, Daniel, Zuercher, William, Willson, Timothy M, MacDonald, Andrew S, Bolognese, Brian, Podolin, Patricia L, Sanchez, Yolanda, Loudon, Andrew Si, Ray, David W

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Discovery of a potent series of non-steroidal non α-trifluoromethyl carbinol glucocorticoid receptor agonists with reduced lipophilicity von Diallo, Hawa, Angell, Davina C., Barnett, Heather A., Biggadike, Keith, Coe, Diane M., Cooper, Tony W.J., Craven, Andy, Gray, James R., House, David, Jack, Torquil I., Keeling, Steve P., Macdonald, Simon J.F., McLay, Iain M., Oliver, Samuel, Taylor, Simon J., Uings, Iain J., Wellaway, Natalie

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Registration of 'Chet' sand bluestem von Springer, T.L, Dewald, C.L, Sims, P.L, Gillen, R.L, Louthan, V.H, Cooper, W.J, Taliaferro, C.M, Wynia, R.L, Houck, M.J. Jr, Esquivel, R.G

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Fenton-Mediated Oxidation in the Presence and Absence of Oxygen von Duesterberg, Christopher K, Cooper, William J, Waite, T. David

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Gaia Early Data Release 3 The Gaia Catalogue of Nearby Stars von Smart, R.L, Sarro, L.M, Rybizki, J, Reyle, C, Robin, A.C, Hambly, N.C, Abbas, U, Barstow, M.A, de Bruijne, J.H.J, Bucciarelli, B, Carrasco, J.M, Cooper, W.J, Hodgkin, S.T, Masana, E, Michalik, D, Sahlmann, J, Sozzetti, A, Brown, A.G.A, Vallenari, A, Prusti, T, Babusiaux, C, Biermann, M, Creevey, O.L, Evans, D.W, Eyer, L, Hutton, A, Jansen, F, Jordi, C, Klioner, S.A, Lammers, U, Lindegren, L, Luri, X, Mignard, F, Panem, C, Pourbaix, D, Randich, S, Sartoretti, P, Soubiran, C, Walton, N.A, Arenou, F, Bailer-Jones, C.A.L, Bastian, U, Cropper, M, Drimmel, R, Katz, D, Lattanzi, M.G, van Leeuwen, F, Bakker, J, Castaneda, J, De Angeli, F, Ducourant, C, Fabricius, C, Fouesneau, M, Fremat, Y, Guerra, R, Guerrier, A, Guiraud, J, Piccolo, A. Jean-Antoine, Messineo, R, Mowlavi, N, Nicolas, C, Nienartowicz, K, Pailler, F, Panuzzo, P, Riclet, F, Roux, W, Seabroke, G.M, Sordo, R, Tanga, P, Thevenin, F, Gracia-Abril, G, Portell, J, Teyssier, D, Altmann, M, Andrae, R, Bellas-Velidis, I, Benson, K, Berthier, J, Blomme, R, Brugaletta, E, Burgess, P.W, Busso, G, Carry, B, Cellino, A, Cheek, N, Clementini, G, Damerdji, Y, Davidson, M, Delchambre, L, Dell'Oro, A, Fernandez-Hernandez, J, Galluccio, L, Garcia-Lario, P, Garcia-Reinaldos, M, Gonzalez-Nunez, J, Gosset, E, Haigron, R, Halbwachs, J.-L, Harrison, D.L, Hatzidimitriou, D

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Optimization of Novel Indazoles as Highly Potent and Selective Inhibitors of Phosphoinositide 3‑Kinase δ for the Treatment of Respiratory Disease von Down, Kenneth, Amour, Augustin, Baldwin, Ian R, Cooper, Anthony W. J, Deakin, Angela M, Felton, Leigh M, Guntrip, Stephen B, Hardy, Charlotte, Harrison, Zoë A, Jones, Katherine L, Jones, Paul, Keeling, Suzanne E, Le, Joelle, Livia, Stefano, Lucas, Fiona, Lunniss, Christopher J, Parr, Nigel J, Robinson, Ed, Rowland, Paul, Smith, Sarah, Thomas, Daniel A, Vitulli, Giovanni, Washio, Yoshiaki, Hamblin, J. Nicole

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Registration of 'Verl' eastern gamagrass von Springer, T.L, Dewald, C.L, Sims, P.L, Gillen, R.L, Louthan, V.H, Cooper, W.J, Taliaferro, C.M, Maura, C. Jr, Pfaff, S, Wynia, R.L

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A Turing Test for Molecular Generators von Bush, Jacob T, Pogany, Peter, Pickett, Stephen D, Barker, Mike, Baxter, Andrew, Campos, Sebastien, Cooper, Anthony W. J, Hirst, David, Inglis, Graham, Nadin, Alan, Patel, Vipulkumar K, Poole, Darren, Pritchard, John, Washio, Yoshiaki, White, Gemma, Green, Darren V. S

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Radiation induced decomposition of methyl tert-butyl ether in water in presence of chloroform: Kinetic modelling von Basfar, Ahmed A., Khan, Hasan M., Al-Shahrani, Ahmed A., Cooper, William J.

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Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening von Wellaway, Christopher R, Amans, Dominique, Bamborough, Paul, Barnett, Heather, Bit, Rino A, Brown, Jack A, Carlson, Neil R, Chung, Chun-wa, Cooper, Anthony W. J, Craggs, Peter D, Davis, Robert P, Dean, Tony W, Evans, John P, Gordon, Laurie, Harada, Isobel L, Hirst, David J, Humphreys, Philip G, Jones, Katherine L, Lewis, Antonia J, Lindon, Matthew J, Lugo, Dave, Mahmood, Mahnoor, McCleary, Scott, Medeiros, Patricia, Mitchell, Darren J, O’Sullivan, Michael, Le Gall, Armelle, Patel, Vipulkumar K, Patten, Chris, Poole, Darren L, Shah, Rishi R, Smith, Jane E, Stafford, Kayleigh A. J, Thomas, Pamela J, Vimal, Mythily, Wall, Ian D, Watson, Robert J, Wellaway, Natalie, Yao, Gang, Prinjha, Rab K

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Free Radical Destruction of N-Nitrosodimethylamine in Water von Mezyk, Stephen P, Cooper, William J, Madden, Keith P, Bartels, David M

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Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease von Amour, Augustin, Barton, Nick, Cooper, Anthony W. J, Inglis, Graham, Jamieson, Craig, Luscombe, Christopher N, Morrell, Josie, Peace, Simon, Perez, David, Rowland, Paul, Tame, Chris, Uddin, Sorif, Vitulli, Giovanni, Wellaway, Natalie

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Discovery of Potent, Efficient, and Selective Inhibitors of Phosphoinositide 3‑Kinase δ through a Deconstruction and Regrowth Approach von Barton, Nick, Convery, Máire, Cooper, Anthony W. J, Down, Kenneth, Hamblin, J. Nicole, Inglis, Graham, Peace, Simon, Rowedder, James, Rowland, Paul, Taylor, Jonathan A, Wellaway, Natalie

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Optimized Chemical Probes for REV-ERBα von Trump, Ryan P, Bresciani, Stefano, Cooper, Anthony W. J, Tellam, James P, Wojno, Justyna, Blaikley, John, Orband-Miller, Lisa A, Kashatus, Jennifer A, Boudjelal, Mohamed, Dawson, Helen C, Loudon, Andrew, Ray, David, Grant, Daniel, Farrow, Stuart N, Willson, Timothy M, Tomkinson, Nicholas C. O

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Lead Optimization Using Matched Molecular Pairs: Inclusion of Contextual Information for Enhanced Prediction of hERG Inhibition, Solubility, and Lipophilicity von Papadatos, George, Alkarouri, Muhammad, Gillet, Valerie J, Willett, Peter, Kadirkamanathan, Visakan, Luscombe, Christopher N, Bravi, Gianpaolo, Richmond, Nicola J, Pickett, Stephen D, Hussain, Jameed, Pritchard, John M, Cooper, Anthony W. J, Macdonald, Simon J. F

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Circadian clock component REV-ERB[alpha] controls homeostatic regulation of pulmonary inflammation von Pariollaud, Marie, Gibbs, Julie E, Hopwood, Thomas W, Brown, Sheila, Begley, Nicola, Vonslow, Ryan, Poolman, Toryn, Guo, Baoqiang, Saer, Ben, Jones, D. Heulyn, Tellam, James P, Bresciani, Stefano, Tomkinson, Nicholas C.O, Wojno-Picon, Justyna, Cooper, Anthony W.J, Daniels, Dion A, Trump, Ryan P, Grant, Daniel, Zuercher, William, Willson, Timothy M, MacDonald, Andrew S, Bolognese, Brian, Podolin, Patricia L, Sanchez, Yolanda, Loudon, Andrew S.I, Ray, David W

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Pyrazolopyridines as a novel structural class of potent and selective PDE4 inhibitors von Hamblin, J. Nicole, Angell, Tony D.R., Ballantine, Stuart P., Cook, Caroline M., Cooper, Anthony W.J., Dawson, John, Delves, Christopher J., Jones, Paul S., Lindvall, Mika, Lucas, Fiona S., Mitchell, Charlotte J., Neu, Margarete Y., Ranshaw, Lisa E., Solanke, Yemisi E., Somers, Don O., Wiseman, Joanne O.

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Synthesis of dibenzylamino-1-methylcyclohexanol and dibenzylamino-1-trifluoromethylcyclohexanol isomers von Jones, D Heulyn, Bresciani, Stefano, Tellam, James P, Wojno, Justyna, Cooper, Anthony W J, Kennedy, Alan R, Tomkinson, Nicholas C O

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