Rational Design, Synthesis, and Biological Evaluation of 7‑Azaindole Derivatives as Potent Focused Multi-Targeted Kinase Inhibitors von Daydé-Cazals, Bénédicte, Fauvel, Bénédicte, Singer, Mathilde, Feneyrolles, Clémence, Bestgen, Benoit, Gassiot, Fanny, Spenlinhauer, Aurélia, Warnault, Pierre, Van Hijfte, Nathalie, Borjini, Nozha, Chevé, Gwénaël, Yasri, Abdelaziz

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Design, synthesis, and biological evaluation of bifunctional thyrointegrin inhibitors: new anti-angiogenesis analogs von Bridoux, Alexandre, Khan, Riaz A., Chen, Celei, Chevé, Gwenaël, Cui, Huadong, Dyskin, Evgeny, Yasri, Aziz, Mousa, Shaker A.

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Structural elucidation of the DFG-Asp in and DFG-Asp out states of TAM kinases and insight into the selectivity of their inhibitors von Messoussi, Abdellah, Peyronnet, Lucile, Feneyrolles, Clémence, Chevé, Gwénaël, Bougrin, Khalid, Yasri, Aziz

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Axl kinase as a key target for oncology: focus on small molecule inhibitors von Feneyrolles, Clémence, Spenlinhauer, Aurélia, Guiet, Léa, Fauvel, Bénédicte, Daydé-Cazals, Bénédicte, Warnault, Pierre, Chevé, Gwénaël, Yasri, Aziz

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Discovering novel 7-azaindole-based series as potent AXL kinase inhibitors von Feneyrolles, Clémence, Guiet, Léa, Singer, Mathilde, Van Hijfte, Nathalie, Daydé-Cazals, Bénédicte, Fauvel, Bénédicte, Chevé, Gwénaël, Yasri, Abdelaziz

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Comparative Protein Modeling of 1-Deoxy-d-xylulose-5-phosphate Reductoisomerase Enzyme from Plasmodium falciparum:  A Potential Target for Antimalarial Drug Discovery von SINGH, Nidhi, CHEVé, Gwénaël, AVERY, Mitchell A., MCCURDY, Christopher R.

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Recent Progress in the Design, Study, and Development of c-Jun N-Terminal Kinase Inhibitors as Anticancer Agents von Messoussi, Abdellah, Feneyrolles, Clémence, Bros, Aurélie, Deroide, Arthur, Daydé-Cazals, Bénédicte, Chevé, Gwénaël, Van Hijfte, Nathalie, Fauvel, Bénédicte, Bougrin, Khalid, Yasri, Aziz

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Determination and validation of mTOR kinase-domain 3D structure by homology modeling von Lakhlili, Wiame, Chevé, Gwénaël, Yasri, Abdelaziz, Ibrahimi, Azeddine

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A combined ligand-based and target-based drug design approach for G-protein coupled receptors: application to salvinorin A, a selective kappa opioid receptor agonist von Singh, Nidhi, Chevé, Gwénaël, Ferguson, David M, McCurdy, Christopher R

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Structure–activity relationships of neuropeptide FF and related peptidic and non-peptidic derivatives von Vyas, Neha, Mollereau, Catherine, Chevé, Gwénaël, McCurdy, Christopher R.

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Melatonin related compounds inhibit lipid peroxidation during copper or free radical-induced LDL oxidation von Bonnefont-Rousselot, Dominique, Chevé, Gwénaël, Gozzo, Andrea, Tailleux, Anne, Guilloz, Virginie, Caisey, Stéphanie, Teissier, Elisabeth, Fruchart, Jean-Charles, Delattre, Jacques, Jore, Daniel, Lesieur, Daniel, Duriez, Patrick, Gardès-Albert, Monique

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De novo design, synthesis and pharmacological evaluation of new azaindole derivatives as dual inhibitors of Abl and Src kinases von Chevé, Gwénaël, Bories, Cédric, Fauvel, Bénédicte, Picot, François, Tible, Alix, Daydé-Cazals, Bénédicte, Loget, Olivier, Yasri, Aziz

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A Quantitative Structure Activity Relationship approach to probe the influence of the functionalization on the drug encapsulation of porous metalorganic frameworks von Gaudin, Cédric, Cunha, Denise, Ivanoff, Emilie, Horcajada, Patricia, Chevé, Gwenael, Yasri, Aziz, Loget, Olivier, Serre, C., Maurin, Guillaume

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Increased Susceptibility of Low-Density Lipoprotein to Ex Vivo Oxidation in Mice Transgenic for Human Apolipoprotein B Treated with 1 Melatonin-Related Compound Is Not Associated w... von Tailleux, Anne, Gozzo, Andrea, Torpier, Gérard, Martin-Nizard, Françoise, Bonnefont-Rousselot, Dominique, Lemdani, Mohamed, Furman, Christophe, Foricher, Rachel, Chevé, Gwenaël, Yous, Saïd, Micard, Florence, Bordet, Régis, Gardes-Albert, Monique, Lesieur, Daniel, Teissier, Elisabeth, Fruchart, Jean-Charles, Fiévet, Catherine, Duriez, Patrick

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Structure–activity relationship of phenytoinergic antiepileptic drugs related to ameltolide von Philip, Ashok E., Poupaert, Jacques H., Chevé, Gwénaël, Muccioli, Giulio, Lambert, Didier, McCurdy, Christopher R.

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Comparative Protein Modeling of 1-Deoxy-d-xylulose-5-phosphate Reductoisomerase Enzyme from Plasmodium f alciparum:  A Potential Target for Antimalarial Drug Discovery von Singh, Nidhi, Chevé, Gwénaël, Avery, Mitchell A, McCurdy, Christopher R

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DERIVATIVES OF AZAINDOLES AS INHIBITORS OF PROTEIN KINASES ABL AND SRC von YASRI, Abdelaziz, BORIES, Cedric, CHEVE, Gwenaël, DELON, Louis

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Structure-activity relationships of neuropeptide FF and related peptidic and non-peptidic derivatives: RFamide peptides von VYAS, Neha, MOLLEREAU, Catherine, CHEVE, Gwénaël, MCCURDY, Christopher R

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Derivatives of azaindoles as inhibitors of protein kinases Abl and Src von YASRI, ABDELAZIZ, DELON, LOUIS, CHEVE, GWENAEL, BORIES, CEDRIC

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ANTI-AXL ANTIBODIES AND USES THEREOF von YASRI, Aziz, CHARDES, Thierry, PELEGRIN, André, CHEVE, Gwénaël, FAUVEL, Bénédicte, LARROQUE, Christian, LECONET, Wilhem, LARBOURET, Christel, ROBERT, Bruno

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