Nonsteroidal antiandrogens. Synthesis and structure-activity relationships of 3-substituted derivatives of 2-hydroxypropionanilides von Tucker, Howard, Crook, J. W, Chesterson, G. J

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Resolution of the nonsteroidal antiandrogen 4'-cyano-3-[(4-fluorophenyl)sulfonyl]-2-hydroxy-2-methyl-3'-(trifluoromethyl)propionanilide and the determination of the absolute config... von TUCKER, H, CHESTERSON, G. J

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Potentiation of fasciolicidal agents by benzoyl side chains, synthesis of benzoylsalicylanilides von Brown, George R, Chesterson, Glynn J, Coles, Gerald C

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Respite care for caregivers and people with severe mental illness: literature review von Jeon, Yun-Hee, Brodaty, Henry, Chesterson, Jon

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'Give me a break'- respite care for older carers of mentally ill persons von Jeon, Yun-Hee, Brodaty, Henry, O'Neill, Colleen, Chesterson, Jon

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SERIALIZATION AND EMPIRE IN NEIL GAIMAN'S "THE SANDMAN" von MELLETTE, JUSTIN

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Cutting system for cutting profiles in air-permeable and resilient materials and method von GREENWALD JOHN A, ROTTER MARTIN J, CHESTERSON WILLIAM L, MOSLEY MICHAEL J, BECHTLE CHARLES G, PATTON JAMES S

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Synthesis of [ 14C]- and [ 3H]-labelled ICI 176,334 von Harding, JR, Bergin, JA, Tucker, H, Chesterson, G

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Discovery of AZD3514, a small-molecule androgen receptor downregulator for treatment of advanced prostate cancer von Bradbury, Robert H., Acton, David G., Broadbent, Nicola L., Brooks, A. Nigel, Carr, Gregory R., Hatter, Glenn, Hayter, Barry R., Hill, Kathryn J., Howe, Nicholas J., Jones, Rhys D.O., Jude, David, Lamont, Scott G., Loddick, Sarah A., McFarland, Heather L., Parveen, Zaieda, Rabow, Alfred A., Sharma-Singh, Gorkhn, Stratton, Natalie C., Thomason, Andrew G., Trueman, Dawn, Walker, Graeme E., Wells, Stuart L., Wilson, Joanne, Wood, J. Matthew

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The "more at home with dementia" program: a randomized controlled study protocol to determine how caregiver training affects the well-being of patients and caregivers von Birkenhäger-Gillesse, Elizabeth G, Kollen, Boudewijn J, Zuidema, Sytse U, Achterberg, Wilco P

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Cysteamine–bicalutamide combination therapy corrects proximal tubule phenotype in cystinosis von Jamalpoor, Amer, van Gelder, Charlotte AGH, Yousef Yengej, Fjodor A, Zaal, Esther A, Berlingerio, Sante P, Veys, Koenraad R, Pou Casellas, Carla, Voskuil, Koen, Essa, Khaled, Ammerlaan, Carola ME, Rega, Laura Rita, van der Welle, Reini EN, Lilien, Marc R, Rookmaaker, Maarten B, Clevers, Hans, Klumperman, Judith, Levtchenko, Elena, Berkers, Celia R, Verhaar, Marianne C, Altelaar, Maarten, Masereeuw, Rosalinde, Janssen, Manoe J

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Small-molecule androgen receptor downregulators as an approach to treatment of advanced prostate cancer von Bradbury, Robert H., Hales, Neil J., Rabow, Alfred A., Walker, Graeme E., Acton, David G., Andrews, David M., Ballard, Peter, Brooks, Nigel A.N., Colclough, Nicola, Girdwood, Alan, Hancox, Urs J., Jones, Owen, Jude, David, Loddick, Sarah A., Mortlock, Andrew A.

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Oxidative β-C-H sulfonylation of cyclic aminesElectronic supplementary information (ESI) available. See DOI: 10.1039/c7sc04900e von Griffiths, R. J, Kong, W. C, Richards, S. A, Burley, G. A, Willis, M. C, Talbot, E. P. A

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Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists von Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Vorobiev, Anton A., Kuznetsova, Irina V., Shevkun, Natalia A., Koryakova, Angela G., Karapetian, Ruben N., Trifelenkov, Andrey S., Kravchenko, Dmitry V., Veselov, Mark S., Chufarova, Nina V.

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Design, synthesis and biological profiling of aryl piperazine based scaffolds for the management of androgen sensitive prostatic disordersThe authors declare no competing interests. CSIR-CDRI Communication no. 9294.Electronic supplementary information (ESI) available: Experimental details of chemistry and biology, 1H NMR, 13C NMR spectral data, 1H NMR, 13C NMR spectra, HRMS of compounds 8a-e, 9a-n, 11a-b and 12a-g and a representative chromatogram of compound 9a. See DOI: 10.1039/c6md00426a von Gupta, Sonal, Pandey, Deepti, Mandalapu, Dhanaraju, Bala, Veenu, Sharma, Vikas, Shukla, Mahendra, Yadav, Santosh K, Singh, Nidhi, Jaiswal, Swati, Maikhuri, Jagdamba P, Lal, Jawahar, Siddiqi, Mohammad I, Gupta, Gopal, Sharma, Vishnu L

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Microarray analysis of bicalutamide action on telomerase activity, p53 pathway and viability of prostate carcinoma cell lines von Bouchal, Jan, Baumforth, Karl R. N., Šváchová, Michaela, Murray, Paul G., von Angerer, Erwin, Kolár̂, Zdenêk

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Bicalutamide dosages used in the treatment of prostate cancer von Kolvenbag, Geert J.C.M., Nash, Anthony

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Inhibition of Androgen Receptor Function and Level in Castration-Resistant Prostate Cancer Cells by 2-[(isoxazol-4-ylmethyl)thio]-1-(4-phenylpiperazin-1-yl)ethanone von Masoodi, Khalid Z, Eisermann, Kurtis, Yang, Zhenyu, Dar, Javid A, Pascal, Laura E, Nguyen, Minh, O’Malley, Katherine, Parrinello, Erica, Feturi, Firuz G, Kenefake, Alex N, Nelson, Joel B, Johnston, Paul A, Wipf, Peter, Wang, Zhou

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Bilateral widespread mechanical pain sensitivity in carpal tunnel syndrome: evidence of central processing in unilateral neuropathy von Fernández-de-las-Peñas, César, de la Llave-Rincón, Ana Isabel, Fernández-Carnero, Josué, Cuadrado, María Luz, Arendt-Nielsen, Lars, Pareja, Juan A.

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Assessment of deep dynamic mechanical sensitivity in individuals with tension‐type headache: The dynamic pressure algometry von Palacios‐Ceña, M., Wang, K., Castaldo, M., Guerrero‐Peral, Á., Caminero, A.B., Fernández‐de‐las‐Peñas, C., Arendt‐Nielsen, L.

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