A stereochemical journey around spirocyclic glutamic acid analogs von Chernykh, Anton V, Chernykh, Alla V, Radchenko, Dmytro S, Chheda, Pratik Rajesh, Rusanov, Eduard B, Grygorenko, Oleksandr O, Spies, M. Ashley, Volochnyuk, Dmitriy M, Komarov, Igor V

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Fluoroalkyl-Substituted Cyclopropane Derivatives: Synthesis and Physicochemical Properties von Chernykh, Anton V, Olifir, Oleksandr S, Kuchkovska, Yuliya O, Volochnyuk, Dmitriy M, Yarmolchuk, Vladimir S, Grygorenko, Oleksandr O

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Impact of β-perfluoroalkyl substitution of proline on the proteolytic stability of its peptide derivatives von Chernykh, Anton V, Aloshyn, Danylo, Kuchkovska, Yuliya O, Daniliuc, Constantin G, Tolmachova, Nataliya A, Kondratov, Ivan S, Zozulya, Sergey, Grygorenko, Oleksandr O, Haufe, Günter

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3‑Substituted 6‑Azabicyclo[3.1.1]heptanes: Nonclassical Piperidine Isosteres for Drug Discovery von Chernykh, Anton V., Vashchenko, Bohdan V., Shishkina, Svitlana V., Volochnyuk, Dmytro M., Grygorenko, Oleksandr O.

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3‐Fluoroalkyl (CF3, CHF2, CH2F) Cyclobutane‐Derived Building Blocks for Medicinal Chemistry: Synthesis and Physicochemical Properties von Demchuk, Oleksandr P., Bobovskyi, Bohdan V., Vashchenko, Bohdan V., Hryshchuk, Oleksandr V., Skreminskyi, Artem, Chernykh, Anton V., Moskvina, Viktoriia S., Hordiyenko, Olga V., Volochnyuk, Dmitriy M., Grygorenko, Oleksandr O.

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Last of the gem-Difluorocycloalkanes: Synthesis and Characterization of 2,2-Difluorocyclobutyl-Substituted Building Blocks von Chernykh, Anton V, Melnykov, Kostiantyn P, Tolmacheva, Nataliya A, Kondratov, Ivan S, Radchenko, Dmytro S, Daniliuc, Constantin G, Volochnyuk, Dmitriy M, Ryabukhin, Sergey V, Kuchkovska, Yuliya O, Grygorenko, Oleksandr O

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Synthesis, biological evaluation, and modeling studies of 1,3-disubstituted cyclobutane-containing analogs of combretastatin A4 von Malashchuk, Andrii, Chernykh, Anton V., Hurmach, Vasyl V., Platonov, Maxim O., Onopchenko, Oleksandra, Zozulya, Sergey, Daniliuc, Constantin G., Dobrydnev, Alexey V., Kondratov, Ivan S., Moroz, Yuriy S., Grygorenko, Oleksandr O.

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Expanding the Chemical Space of 1,2-Difunctionalized Cyclobutanes von Chernykh, Anton V., Kudryk, Oleksandr V., Olifir, Oleksandr S., Dobrydnev, Alexey V., Rusanov, Eduard, Moskvina, Viktoriia S., Volochnyuk, Dmitriy M., Grygorenko, Oleksandr O.

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2‐ and 3‐Fluorocyclobutane Building Blocks for Organic and Medicinal Chemistry von Malashchuk, Andrii, Demchuk, Oleksandr P., Razhyk, Bohdan V., Holumbievskyi, Vitalii O., Kudryk, Oleksandr V., Chernykh, Anton V., Hryshchuk, Oleksandr V., Sosunovych, Bohdan S., Volochnyuk, Dmytro M., Vashchenko, Bohdan V., Grygorenko, Oleksandr O.

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3‑((Hetera)cyclobutyl)azetidines, “Stretched” Analogues of Piperidine, Piperazine, and Morpholine: Advanced Building Blocks for Drug Discovery von Feskov, Illia O, Chernykh, Anton V, Kuchkovska, Yuliya O, Daniliuc, Constantin G, Kondratov, Ivan S, Grygorenko, Oleksandr O

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Multigram Synthesis of Advanced 6,6‐Difluorospiro[3.3]heptane‐Derived Building Blocks von Olifir, Oleksandr S., Chernykh, Anton V., Dobrydnev, Alexey V., Grygorenko, Oleksandr O., Moroz, Yuriy S., Voitenko, Zoia V., Radchenko, Dmytro S.

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Synthesis of new fluorinated proline analogues from polyfluoroalkyl β-ketoacetals and ethyl isocyanoacetate von Tolmachova, Nataliya A, Kondratov, Ivan S, Dolovanyuk, Violetta G, Pridma, Stanislav O, Chernykh, Anton V, Daniliuc, Constantin G, Haufe, Günter

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Cyclobutyl-Containing Rigid Analogues of Threonine: Synthesis and Physical Chemical Properties von Feskov, Illia O, Chernykh, Anton V, Kondratov, Ivan S, Klyachina, Mariya, Daniliuc, Constantin G, Haufe, Günter

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Synthesis of fluorinated building blocks based on spiro[3.3]heptane scaffold von Chernykh, Anton V., Feskov, Illia O., Chernykh, Alla V., Daniliuc, Constantin G., Tolmachova, Nataliya A., Volochnyuk, Dmitriy M., Radchenko, Dmytro S.

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Synthesis and Structural Analysis of Angular Monoprotected Diamines Based on Spiro[3.3]heptane Scaffold von Chernykh, Anton V, Radchenko, Dmytro S, Grygorenko, Oleksandr O, Daniliuc, Constantin G, Volochnyuk, Dmitriy M, Komarov, Igor V

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Synthesis and Physicochemical Properties of 3-Fluorocyclobutylamines von Chernykh, Anton V., Radchenko, Dmytro S., Chernykh, Alla V., Kondratov, Ivan S., Tolmachova, Nataliya A., Datsenko, Olexandr P., Kurkunov, Maxim A., Zozulya, Sergey X., Kheylik, Yuri P., Bartels, Katharina, Daniliuc, Constantin G., Haufe, Günter

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Synthesis and Physical-Chemical Properties of cis- and trans-1-Amino-3-fluoro-3-methylcyclobutanecarboxylic Acids von Chernykh, Anton V., Feskov, Illia O., Chernykh, Alla V., Kondratov, Ivan S., Tolmachova, Nataliya, Radchenko, Dmytro S., Daniliuc, Constantin G., Haufe, Günter

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Conformationally restricted glutamic acid analogues: stereoisomers of 1-aminospiro[3.3]heptane-1,6-dicarboxylic acid von Chernykh, Anton V., Radchenko, Dmytro S., Grygorenko, Oleksandr O., Volochnyuk, Dmitriy M., Shishkina, Svitlana V., Shishkin, Oleg V., Komarov, Igor V.

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3-Substituted 6-Azabicyclo3.1.1heptanes: Nonclassical Piperidine Isosteres for Drug Discovery von Chernykh, Anton V, Vashchenko, Bohdan V, Shishkina, Svitlana V, Volochnyuk, Dmytro M, Grygorenko, Oleksandr O

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Fluorine‐Labelled Spiro[3.3]heptane‐Derived Building Blocks: Is Single Fluorine the Best? von Malashchuk, Andrii, Chernykh, Anton V., Dobrydnev, Alexey V., Grygorenko, Oleksandr O.

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