Strategy to Improve the Oral Pharmacokinetics of Cyclin-Dependent Kinase 4/6 Inhibitors: Enhancing Permeability and CYP450 Inhibition by a Natural Bioenhancer von Patil, Prajakta Harish, Desai, Mrunal Pradeep, Rao, Rajat Radhakrishna, Mutalik, Srinivas, Puralae Channabasavaiah, Jagadish

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Molecular dynamics simulation and in vitro evaluation of herb–drug interactions involving dietary polyphenols and CDK inhibitors in breast cancer chemotherapy von Patil, Prajakta H., Birangal, Sumit, Shenoy, G. Gautham, Rao, Mahadev, Kadari, Sandeep, Wankhede, Amit, Rastogi, Himanshu, Sharma, Tarun, Pinjari, Jakir, Puralae Channabasavaiah, Jagadish

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Enhancing the oral bioavailability of asenapine maleate with bio-enhancer: An in-silico assisted in-vivo pharmacokinetic study von Suresh, Akhil, Narayan, Reema, Tummala, Hari Prabhath, Matcha, Saikumar, Mallayasamy, Surulivelrajan, Nayak, Yogendra, Puralae Channabasavaiah, Jagadish, Nayak, Usha Y.

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Assessment of pH-shift drug interactions of palbociclib by in vitro micro-dissolution in bio relevant media: An analytical QbD-driven RP-HPLC method optimization von Harish Patil, Prajakta, Desai, Mrunal, Radhakrishna Rao, Rajat, Mutalik, Srinivas, Gautham Shenoy, Gurupur, Rao, Mahadev, Channabasavaiah Jagadish, Puralae

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A pilot randomized controlled trial to compare the effectiveness of two 14-day primaquine regimens for the radical cure of vivax malaria in South India von Saravu, Kavitha, Tellapragada, Chaitanya, Kulavalli, Shrivathsa, Xavier, Wilbin, Umakanth, Shashikiran, Brahmarouphu, Gouthami, Srinivas, Navyasree Kola, Channabasavaiah, Jagadish Puralae, Bava, Anzil, Saadi, Abdul Vahab, Guddattu, Vasudev, Satyamoorthy, Kapaettu, Bhat, Krishnamurthy

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Evaluation of pH Dependent Solubility and Examination of Variation in Pharmacokinetic Properties of Alectinib: A Quantitative Study by Implementing Integrated Quality by Design App... von Kolasani, Durga Deepthi, Desai, Mrunal, Patil, Prajakta, Channabasavaiah, Jagadish Puralae

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Differential effects of dietary polyphenols on oral pharmacokinetics of cyclin-dependent kinase inhibitors in rats: a mechanistic framework for in vitro-in vivo extrapolation von Patil, Prajakta Harish, Desai, Mrunal Pradeep, Birangal, Sumit, Gautham Shenoy, G, Channabasavaiah, Jagadish Puralae

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Extraction, characterization and evaluation of Kaempferia galanga L. (Zingiberaceae) rhizome extracts against acute and chronic inflammation in rats von Jagadish, Puralae Channabasavaiah, Latha, Kotehal Parameshwarappa, Mudgal, Jayesh, Nampurath, Gopalan Kutty

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Estimation of CDK inhibitors by RP-HPLC: application for pharmacokinetic interactions studies with PPIs von Desai, Mrunal Pradeep, Patil, Prajakta Harish, Shenoy, Gurupur Gautham, Channabasavaiah, Jagadish Puralae

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Should the Use of Acid Reducing Agents in Conjunction with Ribociclib be Avoided? An Integrated QbD Approach for Assessment of pH-Mediated Interaction von Desai, Mrunal, Patil, Prajakta Harish, Rao, Rajat Radhakrishna, Shenoy, Gurupur Gautham, Rao, Mahadev, Mutalik, Srinivas, Jagadish, Puralae Channabasavaiah

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In-silico design, synthesis and biological evaluation of 4-aryl-4H-chromene derivatives as CDK-2 inhibitors: A molecular approach to finding a lead for breast cancer von Amin, Sk Md Sohail, Patil, Prajakta Harish, Desai, Mrunal, Channabasavaiah, Jagadish Puralae

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The prediction of pH-dependent interaction using micro-dissolution approach in bio-relevant media: Insights from model drug study of lapatinib von Rajpurohit, nithakumari Uttam Singh, Patil, Prajakta Harish, Desai, Mrunal, Channabasavaiah, Jagadish Puralae

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The Effect of Concomitant Administration of Proton Pump Inhibitors on the Pharmacokinetics of CDK4/6 Inhibitors in Rats: Implications for the Evaluation of Hepatic and Transporter-... von Patil, Prajakta Harish, Desai, Mrunal, Birangal, Sumit, Gurupur, Gautham Shenoy, Rao, Mahadev, Yadav, Anandkumar, Kurawattimath, Vishwanath, Chaudhari, Avinash, Sharma, Tarun, Pinjari, Jakir, Channabasavaiah, Jagadish Puralae

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QbD-driven HPLC method for the quantification of rivastigmine in rat plasma and brain for pharmacokinetics study von Gopalan, Divya, Patil, Prajakta H., Jagadish, Puralae Channabasavaiah, Kini, Suvarna G., Alex, Angel Treasa, Udupa, Nayanabhirama, Mutalik, Srinivas

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