Design, synthesis, and biological evaluation of phenyl thiazole-based AR-V7 degraders von Bhumireddy, Archana, Bandaru, N.V.M. Rao, Raghurami Reddy, B., Gore, Suraj T., Mukherjee, Subhendu, Balasubramanian, Wesley Roy, Sumanth Kumar, V., Alapati, Krishna Satya, Venkata Gowri Chandra Sekhar, Kondapalli, Nellore, Kavitha, Abbineni, Chandrasekhar, Samajdar, Susanta

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Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Part 2 von Sasmal, Sanjita, Balasubrahmanyam, D., Kanna Reddy, Hariprasada R., Balaji, Gade, Srinivas, Gujjary, Cheera, Srisailam, Abbineni, Chandrasekhar, Sasmal, Pradip K., Khanna, Ish, Sebastian, V.J., Jadhav, Vikram P., Singh, Manvendra P., Talwar, Rashmi, Suresh, J., Shashikumar, Dhanya, Harinder Reddy, K., Sihorkar, V., Frimurer, Thomas M., Rist, Øystein, Elster, Lisbeth, Högberg, Thomas

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Targeting SWI/SNF ATPases in enhancer-addicted prostate cancer von Xiao, Lanbo, Parolia, Abhijit, Qiao, Yuanyuan, Bawa, Pushpinder, Eyunni, Sanjana, Mannan, Rahul, Carson, Sandra E., Chang, Yu, Wang, Xiaoju, Zhang, Yuping, Vo, Josh N., Kregel, Steven, Simko, Stephanie A., Delekta, Andrew D., Jaber, Mustapha, Zheng, Heng, Apel, Ingrid J., McMurry, Lisa, Su, Fengyun, Wang, Rui, Zelenka-Wang, Sylvia, Sasmal, Sanjita, Khare, Leena, Mukherjee, Subhendu, Abbineni, Chandrasekhar, Aithal, Kiran, Bhakta, Mital S., Ghurye, Jay, Cao, Xuhong, Navone, Nora M., Nesvizhskii, Alexey I., Mehra, Rohit, Vaishampayan, Ulka, Blanchette, Marco, Wang, Yuzhuo, Samajdar, Susanta, Ramachandra, Murali, Chinnaiyan, Arul M.

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Targeting the mSWI/SNF complex in POU2F-POU2AF transcription factor-driven malignancies von He, Tongchen, Xiao, Lanbo, Qiao, Yuanyuan, Klingbeil, Olaf, Young, Eleanor, Wu, Xiaoli S., Mannan, Rahul, Mahapatra, Somnath, Redin, Esther, Cho, Hanbyul, Bao, Yi, Kandarpa, Malathi, Ching-Yi Tien, Jean, Wang, Xiaoju, Eyunni, Sanjana, Zheng, Yang, Kim, NamHoon, Zheng, Heng, Hou, Siyu, Su, Fengyun, Miner, Stephanie J., Mehra, Rohit, Cao, Xuhong, Abbineni, Chandrasekhar, Samajdar, Susanta, Ramachandra, Murali, Dhanasekaran, Saravana M., Talpaz, Moshe, Parolia, Abhijit, Rudin, Charles M., Vakoc, Christopher R., Chinnaiyan, Arul M.

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Abstract 3827: Antitumor activity of ODM-207, a novel BET bromodomain inhibitor, in nonclinical models of ER+ breast cancer as single agent and as a combination treatment von Lindqvist, Julia, Björkman, Mari, Riikonen, Reetta, Nicorici, Daniel, Mattila, Elina, Jaleel, Mahaboobi, Abbineni, Chandrasekhar, Moilanen, Anu-Maarit

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Development of an orally bioavailable mSWI/SNF ATPase degrader and acquired mechanisms of resistance in prostate cancer von He, Tongchen, Cheng, Caleb, Qiao, Yuanyuan, Cho, Hanbyul, Young, Eleanor, Mannan, Rahul, Mahapatra, Somnath, Miner, Stephanie J, Zheng, Yang, Kim, NamHoon, Zeng, Victoria Z, Wisniewski, Jasmine P, Hou, Siyu, Jackson, Bailey, Cao, Xuhong, Su, Fengyun, Wang, Rui, Chang, Yu, Kuila, Bilash, Mukherjee, Subhendu, Dukare, Sandeep, Aithal, Kiran B, D S, Samiulla, Abbineni, Chandrasekhar, Vaishampayan, Ulka, Lyssiotis, Costas A, Parolia, Abhijit, Xiao, Lanbo, Chinnaiyan, Arul M

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Author Correction: Targeting SWI/SNF ATPases in enhancer-addicted prostate cancer von Xiao, Lanbo, Parolia, Abhijit, Qiao, Yuanyuan, Bawa, Pushpinder, Eyunni, Sanjana, Mannan, Rahul, Carson, Sandra E., Chang, Yu, Wang, Xiaoju, Zhang, Yuping, Vo, Josh N., Kregel, Steven, Simko, Stephanie A., Delekta, Andrew D., Jaber, Mustapha, Zheng, Heng, Apel, Ingrid J., McMurry, Lisa, Su, Fengyun, Wang, Rui, Zelenka-Wang, Sylvia, Sasmal, Sanjita, Khare, Leena, Mukherjee, Subhendu, Abbineni, Chandrasekhar, Aithal, Kiran, Bhakta, Mital S., Ghurye, Jay, Cao, Xuhong, Navone, Nora M., Nesvizhskii, Alexey I., Mehra, Rohit, Vaishampayan, Ulka, Blanchette, Marco, Wang, Yuzhuo, Samajdar, Susanta, Ramachandra, Murali, Chinnaiyan, Arul M.

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Abstract 1143: Evaluation of AU-18069, a novel small molecule CBP/p300 bromodomain inhibitor for the treatment of cancers von Abbineni, Chandrasekhar, Thiyagarajan, Saravanan, Senaiar, Ramesh S, Mukherjee, Subhendu, Jaleel, Mahaboobi, Marappan, Sivapriya, N R, Raghavendra, Renukappa, Girish Aggunda, B, Aravind A, R, Naveen Kumar, Reddy, Venkata Siva, Babu, Asha, Srinivas, Akhila, Yadlapalli, Prasad, Gore, Suraj T, Hemasankar, Pathange, Dey, Mamon, S, Samiulla D, Naik, Chandranath D, Antony, Thomas, Nellore, Kavitha, Chelur, Shekar, Daginakatte, Girish, Myllymäki, Mikko, Wohlfahrt, Gerd, Ramachandra, Murali, Samajdar, Susanta

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Abstract 1144: Orally bioavailable SMARCA2 degraders with exceptional selectivity and potency von Abbineni, Chandrasekhar, Satyam, Leena Khare, Kuila, Bilash, Ettam, Ashok, Rawoof, Khaji Abdul, MR, Sreevidya, Dukare, Sandeep Vitthal, Gore, Suraj T., Nankar, Rakesh P., Ahuja, Vijay Kamal, KB, Charamanna, Goyal, Megha, Aithal, Kiran, DS, Samiulla, Mukherjee, Subhendu, Antony, Thomas, Giri, Sanjeev, Chelur, Shekar, Nellore, Kavitha, Daginakatte, Girish, Ramachandra, Murali, Samajdar, Susanta

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Abstract 3970: Therapeutic targeting of estrogen receptor positive breast cancer with the BET bromodomain inhibitor ODM-207 von Lindqvist, Julia, Björkman, Mari, Riikonen, Reetta, Nicorici, Daniel, Mattila, Elina, Abbineni, Chandrasekhar, Jaleel, Mahaboobi, Eriksson, John, Kallio, Pekka, Moilanen, Anu-Maarit

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Abstract LB-113: Immune-mediated anti-tumor activity with a clinical stage BET bromodomain inhibitor ODM-207 in pre-clinical models von Deshpande, Pratima, Babu, Ravi Krishna, Vadnal, Prashant Yallappa, Jaleel, Mahaboobi, Ramachandra, Murali, Abbineni, Chandrasekhar, Samajdar, Susanta, Moilanen, Anu-Maarit, Kallio, Pekka

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Abstract 1753: Targeting cancer with selective cbp/p300 bromodomain inhibitors von Jaleel, Mahaboobi, Senaiar, Ramesh S., Abbineni, Chandrasekhar, Renukappa, Girish A., Mukherjee, Subhendu, Marappan, Sivapriya, Samiulla, DS, Aravind, AB, Kumar, Naveen R., Reddy, Venkata Siva N., Babu, Asha, Srinivas, Akhila P., Yadlapalli, Prasad, Tgore, Suraj, NR, Raghavendra, Naik, Chandranath D., Giri, Sanjeev, Antony, Thomas, Nellore, Kavitha, Chelur, Shekar, Daginakatte, Girish, Ravanti, laura, Myllymäki, Mikko, Wohlfahrt, Gerd, Mattila, Elina, Karlsson, Stefan, Björkman, Mari, Riikonen, Reetta, Ikonen, Tarja, Leimu, Laura, Mälmström, Chira, Korjamo, Timo, Moilanen, Anu, Ramachandra, Murali, Samajdar, Susanta

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Abstract 1754: First in class orally bioavailable BETBRD degraders von Abbineni, Chandrasekhar, Jaleel, Mahaboobi, Mukherjee, Subhendu, Marappan, Sivapriya, Tiwari, Nirbhay Kumar, Samiulla, DS, Aravind, AB, Kumar, Naveen R, Bansal, Indu, Reddy, Raghurami B, Bandaru, NVM Rao, Srinivas, Akhila, Maben, Janith Mary, Tgore, Suraj, Kumar, Avainash, Nankar, Rakesh P., Naik, Chandranath D., Antony, Thomas, Nellore, Kavitha, Giri, Sanjeev, Daginakatte, Girish, Chelur, Shekar, Törmäkangas, Olli, Wohlfahrt, Gerd, Björkman, Mari, Mattila, Elina, Ravanti, Laura, Moilanen, Anu, Ramachandra, Murali, Samajdar, Susanta

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Abstract A047: Discovery of potent and paralog selective PROTAC degraders of CBP or p300 proteins for the treatment of various cancers von Abbineni, Chandrasekhar, Thiyagarajan, Saravanan, T, Krishna Chaitanya, Apte, Achala, R, Naveen Kumar, Kumar, Avinash, Babu, Dabbeeru Madhu, S, Shwetha, Kamath, Aishwarya B, Mandal, Monalisha, Panigrahi, Rituparna, Marappan, Sivapriya, Mukherjee, Subhendu, Nellore, Kavitha, Chelur, Shekar, Ramachandra, Murali, Samajdar, Susanta

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Abstract 118: Targeting cancer with a novel BET bromodomain inhibitor ODM-207 von Moilanen, Anu-Maarit, Björkman, Mari, Riikonen, Reetta, Abbineni, Chandrasekhar, Jaleel, Mahaboobi, Marappan, Sivapriya, Ikonen, Tarja, Daginakatte, Girish, A B, Aravind, Mattila, Elina, Rantala, Juha, Samajdar, Susanta, Ramachandra, Murali, Kallio, Pekka

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Stereoselective synthesis of an advanced seco ester intermediate as a precursor toward the synthesis of amphidinolides T1, T3, and T4 von Sasmal, Pradip K., Abbineni, Chandrasekhar, Iqbal, Javed, Mukkanti, K.

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Abstract A046: Identification of paralog selective degraders of SMARCA2 and SMARCA4 for treatment of various cancers von Abbineni, Chandrasekhar, Aithal, Kiran, Khare, Leena, V, Sandeep Dukare, Kuila, Bilash, Goyal, Megha, Rawoof, Khaji Abdul, Mahadeo, Dhaytadak Bhagwan, Kumar, Bhagya M S, M, Premkumar, Sahu, Swetangini, Gore, Suraj T, N, Lavanya Krishna, KB, Charamanna, CH, Gopinath, S, Samiulla D, Mukherjee, Subhendu, Antony, Thomas, Giri, Sanjeev, Chelur, Shekar, Nellore, Kavitha, Daginakatte, Girish, Ramachandra, Murali, Samajdar, Susanta

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1313 Characterization of the anti-tumor immune activation potential of AUR107, a novel small molecule p300/CBP bromodomain inhibitor von Daginakatte, Girish, Chandrasekhar Abbineni, Thiyagarajan, Saravanan, Dey, Mamon, Basavaraj, Aravind, Dhudashiya, Amit, Marappan, Sivapriya, Patil, Sandeep Sadashiv, Naveen, Kumar R, Raghavendra, N R, Kumar, Avinash, Uma, Bharathi B, Renukappa, Girish, Venkata Siva Reddy, Amith, A, Lavanya, C S, Mukherjee, Subhendu, Samiulla, D S, Antony, Thomas, Eswarappa, Rajesh, Nellore, Kavitha, Chelur, Shekar, Ramachandra, Murali, Samajdar, Susanta

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Abstract 3729: Discovery of orally bioavailable SMARCA2/4 dual degraders for treatment of acute myeloid leukemia von Abbineni, Chandrasekhar, Khare, Leena, Kuila, Bilash, Khaji, Abdul Rawoof, Mahadeo, Dhaytadak Bhagwan, Dukare, Sandeep Vitthal, Kumar, Bhagya M S, Gore, Suraj T, Ahuja, Vijay Kamal, Dhudashiya, Amit A, N R, Raghavendra, Gowda, Nagesh, K B, Charamanna, Aithal B, Kiran, D S, Samiulla, Mukherjee, Subhendu, Antony, Thomas, Giri, Sanjeev, Chelur, Shekar, Nellore, Kavitha, Daginakatte, Girish, Ramachandra, Murali, Samajdar, Susanta

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Abstract 3592: Targeting SWI/SNF ATPases in enhancer-addicted human cancers von Parolia, Abhijit, Xiao, Lanbo, Qiao, Yuanyuan, Bawa, Pushpinder, Eyunni, Sanjana, Young, Eleanor, Mannan, Rahul, Carson, Sandra E., Chang, Yu, Zhang, Yuping, George, James, Jaber, Mustapha, Su, Fengyun, Wang, Rui, Sasmal, Sanjita, Khare, Leena, Mukerjee, Subhendu, AbbinenI, Chandrasekhar, Aithal, Kiran, Cao, Xuhong, Wang, Yuzhuo, Samajdar, Susanta, Ramachandra, Murali, Chinnaiyan, Arul M.

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